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AZ-5104

HY-B0793

AZ-5104

AZ-5104 Chemical Structure

AZ-5104 is a potent EGFR inhibitor, displays potent antitumor activities both in vitro and in vivo.

Size Price Stock Quantity
10 mM * 1 mL in DMSO $55 In-stock
5 mg $50 In-stock
10 mg $90 In-stock
50 mg $320 In-stock
100 mg $520 In-stock
200 mg $720 In-stock
500 mg Get quote
1 g Get quote
Size Price Stock Quantity
10 mM * 1 mL in DMSO €54 In-stock
5 mg €49 In-stock
10 mg €88 In-stock
50 mg €314 In-stock
100 mg €510 In-stock
200 mg €706 In-stock
500 mg Get quote
1 g Get quote

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Product name: AZ-5104
Cat. No.: HY-B0793

AZ-5104 Data Sheet

  • Network Version

    DataSheet

Related Compound Libraries

Biological Activity of AZ-5104

AZ-5104 is a potent EGFR inhibitor, displays potent antitumor activities both in vitro and in vivo.
Target: EGFR
AZ-5104 is an active, demethylated metabolite of AZD-9291. AZ-5104 displays similar overall activity profile with AZD-9291, but is more potent against mutant EGFR forms, while hitting the wild-type EGFR form at a lower concentration thus demonstrating a smaller selectivity margin compared with the parent.

Chemical Information

M.Wt 485.58 Storage Please store the product under the recommended conditions in the Certificate of Analysis.
Formula C27H31N7O2
CAS No 1421373-98-9
Solvent & Solubility

10 mM in DMSO

Preparing Stock Solutions

1 mg 5 mg 10 mg
1 mM 2.0594 mL 10.2970 mL 20.5939 mL
5 mM 0.4119 mL 2.0594 mL 4.1188 mL
10 mM 0.2059 mL 1.0297 mL 2.0594 mL

References on AZ-5104

Inhibitor Kit

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