1. Others
  2. Estrogen Receptor/ERR

PHTPP 

Cat. No.: HY-103456 Purity: 99.07%
Data Sheet SDS Handling Instructions

PHTPP is a selective ERβ antagonist.

For research use only. We do not sell to patients.
PHTPP Chemical Structure

PHTPP Chemical Structure

CAS No. : 805239-56-9

Size Price Stock Quantity
Free Sample (0.5-1 mg)   Apply now  
10 mM * 1 mL in DMSO USD 92 In-stock
5 mg USD 84 In-stock
10 mg USD 144 In-stock
25 mg USD 312 In-stock
50 mg USD 552 In-stock
100 mg USD 912 In-stock
200 mg   Get quote  
500 mg   Get quote  

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  • Biological Activity

  • Protocol

  • Technical Information

  • Purity & Documentation

  • References

Description

PHTPP is a selective ERβ antagonist.

IC50 & Target

ERβ[1]

In Vitro

PHTPP is a selective ERβ antagonist and displays 36-fold selectivity over ERα. PHTPP is fully effective as an ERβ antagonist while exhibiting no significant activity on ERα[1].

References
Preparing Stock Solutions
Concentration Volume Mass 1 mg 5 mg 10 mg
1 mM 2.3623 mL 11.8117 mL 23.6233 mL
5 mM 0.4725 mL 2.3623 mL 4.7247 mL
10 mM 0.2362 mL 1.1812 mL 2.3623 mL
Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

423.31

Formula

C₂₀H₁₁F₆N₃O

CAS No.

805239-56-9

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Shipping

Room temperature in continental US; may vary elsewhere

Solvent & Solubility

10 mM in DMSO

* "<1 mg/mL" means slightly soluble or insoluble. "≥" means soluble, but saturation unknown.

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PHTPP
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