1. Signaling Pathways
  2. Metabolic Enzyme/Protease
  3. Glutaminase
  4. Glutaminase Degrader

Glutaminase Degrader

Glutaminase Degrader (1):

Cat. No. Product Name Effect Purity
  • HY-155102
    PROTAC TG2 degrader-2
    Degrader
    PROTAC TG2 degrader-2 (compound 7) is a selective, competitive degrader targeting Transglutaminase 2 (TG2), with Kd > 100 μM. PROTAC TG2 degrader-2 inhibits the cell migration and decreases the level of TG2 in ovarian cancer cells. PROTAC TG2 degrader-2 can be used for ovarian cancer study.