1. GPCR/G Protein
  2. GPR84
  3. GPR84 antagonist 1

GPR84 antagonist 1 is a high affinity and highly selective competitive antagonist of human GPR84.

For research use only. We do not sell to patients.

GPR84 antagonist 1 Chemical Structure

GPR84 antagonist 1 Chemical Structure

CAS No. : 2762180-28-7

Size Price Stock Quantity
Solid + Solvent (Highly Recommended)
10 mM * 1 mL in DMSO
ready for reconstitution
USD 605 In-stock
Solution
10 mM * 1 mL in DMSO USD 605 In-stock
Solid
5 mg USD 550 In-stock
10 mg USD 890 In-stock
50 mg   Get quote  
100 mg   Get quote  

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Based on 1 publication(s) in Google Scholar

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Description

GPR84 antagonist 1 is a high affinity and highly selective competitive antagonist of human GPR84.

Molecular Weight

422.48

Formula

C26H22N4O2

CAS No.
Appearance

Solid

Color

Off-white to light yellow

SMILES

COC1=CC=C(C2=C(C3=CC=C(OC)C=C3)N=C(CC4=CNC5=C4C=CC=C5)N=N2)C=C1

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 50 mg/mL (118.35 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.3670 mL 11.8349 mL 23.6698 mL
5 mM 0.4734 mL 2.3670 mL 4.7340 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • Molarity Calculator

  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
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Concentration
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Volume
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Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

×
Volume (start)

V1

=
Concentration (final)

C2

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Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

Dosage

mg/kg

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g

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Purity & Documentation
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.3670 mL 11.8349 mL 23.6698 mL 59.1744 mL
5 mM 0.4734 mL 2.3670 mL 4.7340 mL 11.8349 mL
10 mM 0.2367 mL 1.1835 mL 2.3670 mL 5.9174 mL
15 mM 0.1578 mL 0.7890 mL 1.5780 mL 3.9450 mL
20 mM 0.1183 mL 0.5917 mL 1.1835 mL 2.9587 mL
25 mM 0.0947 mL 0.4734 mL 0.9468 mL 2.3670 mL
30 mM 0.0789 mL 0.3945 mL 0.7890 mL 1.9725 mL
40 mM 0.0592 mL 0.2959 mL 0.5917 mL 1.4794 mL
50 mM 0.0473 mL 0.2367 mL 0.4734 mL 1.1835 mL
60 mM 0.0394 mL 0.1972 mL 0.3945 mL 0.9862 mL
80 mM 0.0296 mL 0.1479 mL 0.2959 mL 0.7397 mL
100 mM 0.0237 mL 0.1183 mL 0.2367 mL 0.5917 mL
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GPR84 antagonist 1 Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Product Name:
GPR84 antagonist 1
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HY-139675
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