1. Signaling Pathways
  2. Vitamin D Related/Nuclear Receptor
  3. VD/VDR
  4. VD/VDR Inhibitor

VD/VDR Inhibitor

VD/VDR Inhibitors (2):

Cat. No. Product Name Effect Purity
  • HY-12398A
    TEI-9648
    Inhibitor 99.30%
    TEI-9648, a Vitamin D3 Lactone analogue, is a potent and specific vitamin D receptor (VDR) antagonist. TEI-9648 inhibits VDR/VDRE-mediated genomic actions of 1α,25(OH)2D3. TEI-9648 also inhibits HL-60 cell differentiation induced by of 1α,25(OH)2D3. TEI-9648 has the potential for bone metabolism research.
  • HY-103053
    PS121912
    Inhibitor
    PS121912 is a selective vitamin D receptor (VDR)-coregulator inhibitor. PS121912 has acceptable metabolic stability in vivo. PS121912 can be used for the research of cancer.