1. Metabolic Enzyme/Protease
  2. Dipeptidyl Peptidase
  3. DPP-IV-IN-1

DPP-IV-IN-1 

Cat. No.: HY-U00346
Handling Instructions

DPP-IV-IN-1 is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV), a highly specific serine protease, with an IC50 of 4.6 nM.

For research use only. We do not sell to patients.

DPP-IV-IN-1 Chemical Structure

DPP-IV-IN-1 Chemical Structure

CAS No. : 625110-37-4

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Description

DPP-IV-IN-1 is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV), a highly specific serine protease, with an IC50 of 4.6 nM.

In Vivo

DPP-IV-IN-1 (0.1 and 0.3 mg/kg, p.o.) reduces the increase in plasma glucose beginning 30 min after glucose loading, and significantly suppresses hyperglycemia at the dose of 0.3 mg/kg in a rat model of obesity and impaired glucose tolerance. The effect is based on its inhibitory effect on plasma DPP-IV activity[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

243.28

Formula

C₁₁H₁₈FN₃O₂

CAS No.
SMILES

N#C[[email protected]]1N(C(CNC(C)(C)CO)=O)C[[email protected]@H](F)C1

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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Keywords:

DPP-IV-IN-1Dipeptidyl PeptidaseDPPInhibitorinhibitorinhibit

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