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AR-C155858 Data Sheet

Product Name: AR-C155858
CAS No.: 496791-37-8
Cat. No.: HY-13248
MWt: 461.53
Formula: C21H27N5O5S
Purity : >98%
Solubility: DMSO : ≥ 50 mg/mL (108.34 mM)
Mechanisms: Target: Others
Biological Activity:
AR-C155858 is a selective monocarboxylate transporter MCT1 and MCT2 inhibitor with Kis of 2.3 nM and 10 nM, respectively. IC50 & Target: Ki: 2.3 nM (MCT1), 10 nM (MCT2) In Vitro: AR-C155858 (10 nM-100 nM) inhibits MCT1/MCT2 C-terminal chimaeras[1]. AR-C155858 inhibits MCT2, and the 70% inhibition seen at 10 nM is followed by a gradually increasing inhibition which can only be explained by a Ki value of significantly less than 10 nM. AR-C155858 inhibits MCT1 expressed in Xenopus oocytes in a time- and concentration-dependent manner[2].

Caution: Not fully tested. For research purposes only

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