1. Signaling Pathways
  2. GPCR/G Protein
    Neuronal Signaling
  3. Cannabinoid Receptor
  4. Cannabinoid Receptor Inhibitors

Cannabinoid Receptor Inhibitors

CB1

CB2

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Cannabinoid Receptor Inhibitors, Agonists, Antagonists, Activators & Modulators
Product Name CB1 CB2 Purity
Rimonabant Hydrochloride
CB1 , Ki: 1.8 nM
  99.79%
JD-5037
CB1 , IC50: 1.5 nM
  ≥98.0%
(S)-MRI-1867
CB1
 
Pregnenolone
CB1
  ≥98.0%
Pregnenolone monosulfate
CB1
  ≥98.0%
TM38837
CB1
  99.61%
N-Oleoyl glycine
CB1
  ≥99.0%
EHP-101  
CB2
98.56%
Yangonin
CB1 , IC50: 1.79 μM
CB1 , Ki: 0.72 μM
  99.72%
Bay 59-3074
CB1 , Ki: 48.3 nM
CB2 , Ki: 45.5 nM
98.85%
AZD1940
hCB1-R, pKi: 7.93
hCB2-R, pKi: 9.06
99.45%
Pregnenolone monosulfate sodium salt
CB1
 
Rimonabant
CB1 , Ki: 1.8 nM
 
AM9405
CB1 , IC50: 45.71 nM
 
LY320135
CB1 , Ki: 141 nM
CB2 , Ki: >10 μM
O-2050
CB1 , Ki: 2.5 nM
CB2 , Ki: 0.2 nM
CB2 modulator 1  
CB2
AM281
CB1 , IC50: 9.91 nM
CB2 , IC50: 13000 nM
Drinabant
rCB1-R, IC50: 10 nM
hCB1-R, IC50: 25 nM
CB2 , IC50: 10000 nM
BAY 38-7271
CB1 , Ki: 1.85 nM
CB2 , Ki: 5.96 nM
CB2R-IN-1  
CB2 , Ki: 0.9 nM
Tedalinab  
CB2
CB2R PAM  
cannabinoid type-2 receptors
2-Palmitoylglycerol
CB1
 
Ibipinabant
CB1 , Ki: 7.8 nM
CB2 , Ki: 7943 nM
Leelamine hydrochloride
CB1
 
PM226  
CB2 , EC50: 39 nM
CB2 , Ki: 13 nM
RVD-Hpα
CB1
 
Tetrahydromagnolol
CB1 , EC50: 9010 nM
CB1 , Ki: 2260 nM
CB2 , EC50: 170 nM
CB2 , Ki: 416 nM
CB1 inverse agonist 1
CB1 , IC50: 7.5 nM
CB2 , IC50: 4100 nM
RVD-Hpα TFA
CB1