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  4. Estrogen Receptor/ERR Inhibitors

Estrogen Receptor/ERR Inhibitors

Estrogen receptor

ERα

ERβ

ERRα

ERRβ

ERRγ

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Estrogen Receptor/ERR Inhibitors, Agonists, Antagonists, Activators & Modulators
Product Name Estrogen receptor ERα ERβ ERRα ERRβ ERRγ Purity
Tamoxifen
Estrogen receptor
          99.92%
4-Hydroxytamoxifen
Estrogen receptor, IC50: 3.3 nM
          99.95%
Kaempferol  
ERα
        99.62%
GSK5182          
ERRγ, IC50: 79 nM
FLTX1  
ERα, IC50: 87.5 nM
        99.71%
Tamoxifen Citrate
Estrogen receptor
          ≥99.0%
DPN    
ERβ, EC50: 0.85 nM
      ≥98.0%
Giredestrant
ER
          99.52%
SAR439859  
ERα, EC50: 0.2 nM
        99.59%
Propyl pyrazole triol  
ERα
        ≥99.0%
XCT790      
ERRα, IC50: 0.37 μM
    99.66%
Saikosaponin D    
ERβ
      ≥98.0%
Prinaberel  
hERα, IC50: 1200 nM
mouse ERα, IC50: 750 nM
rat ERα, IC50: 620 nM
hERβ, IC50: 5.4 nM
rat ERβ, IC50: 3.1 nM
mouse ERβ, IC50: 3.7 nM
      98.62%
(E/Z)-4-Hydroxytamoxifen
Estrogen receptor
          99.60%
DY131        
ERRβ
ERRγ
99.72%
ERRα antagonist-1      
ERRα
    ≥98.0%
H3B-5942  
ERαY537S, Ki: 0.41 nM
ERαWT, Ki: 1 nM
        99.31%
PROTAC ERα Degrader-2  
ERα
        98.41%
Hexestrol  
ERα, Ki: 0.06 nM
ERβ, Ki: 0.06 nM
      ≥98.0%
Erteberel    
ERβ, Ki: 1.54 nM
ERβ, EC50: 3.61 nM
      ≥99.0%
OP-1074  
ERα
ERβ
     
Endoxifen  
ERα
       
Acolbifene  
ERα, IC50: 2 nM (E2-induced transcriptional activity)
ERβ, IC50: 0.4 nM (E2-induced transcriptional activity)
      98.86%
Zearalanone
Estrogen receptor
          98.11%
ERα degrader-2  
ERα, IC50: 4.6 nM
       
PROTAC ER Degrader-4
ER
         
PROTAC ERRα Degrader-1      
ERRα
   
ERRγ Inverse Agonist 1  
ERα, IC50: 1.240 μM
   
ERRβ, IC50: 1.330 μM
ERRγ, IC50: 0.040 μM
Giredestrant tartrate
Estrogen receptor
         
4',2-Dihydroxy-4,6-dimethoxydihydrochalcone
Estrogen receptor
         
(E)-4-Hydroxytamoxifen
Estrogen receptor
         
CMP8  
MGERα, IC50: 29 nM
MGRERα, IC50: 41 nM
hERα, IC50: 1100 nM
hERβ, IC50: 2200 nM
     
Raloxifene
Estrogen receptor
         
(+)-Medicarpin    
ERβ
     
Tamoxifen-​d5
Estrogen receptor
         
LY117018
Estrogen receptor
         
Acolbifene hydrochloride  
ERα, IC50: 2 nM (E2-induced transcriptional activity)
ERβ, IC50: 0.4 nM (E2-induced transcriptional activity)
      98.48%
Estrogen receptor modulator 6  
ERα, Ki: 8.4 nM
ERβ, Ki: 0.44 nM
     
PROTAC ERRα ligand 1      
ERRα, IC50: 0.04 μM
 
ERRγ, IC50: 2.8 μM