1. Signaling Pathways
  2. Cell Cycle/DNA Damage
  3. PPAR
  4. PPAR Inhibitors

PPAR Inhibitors

PPARα

PPARβ/δ

PPARγ

PPAR

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

PPAR Inhibitors, Agonists, Antagonists, Activators & Modulators
Product Name PPARα PPARβ/δ PPARγ PPAR Purity
Rosiglitazone    
PPARγ1, EC50: 30 nM
PPARγ2, EC50: 100 nM
  99.21%
GW9662
PPARα, IC50: 32 nM
PPARδ, IC50: 2000 nM
PPARγ, IC50: 3.3 nM
  99.53%
Retinoic acid
PPARα, Kd: 103 nM
PPARβ/δ, Kd: 17 nM
PPARγ, Kd: 178 nM
  98.62%
Elafibranor
PPAR-α, EC50: 45 nM
PPAR-δ, EC50: 175 nM
    99.18%
GW 501516  
PPARδ, EC50: 1.1 nM
    99.27%
VCE-​004.8    
PPARγ
 
T0070907
PPARα, Ki: 0.85 μM
PPARδ, Ki: 1.8 μM
PPARγ, Ki: 1 nM
  99.34%
Troglitazone    
PPARγ, EC50: 550 nM (Human PPARγ)
  99.53%
Pemafibrate
h-PPARα, EC50: 1 nM
PPARδ, EC50: 1.58 μM
h-PPARγ, EC50: 1.1 μM
  99.92%
Icariin
PPARα
      98.75%
Pirinixic acid
PPARα, EC50: 0.63 μM
 
PPARγ, EC50: 32 μM
  99.48%
GW 6471
PPARα
      98.98%
GW1929    
PPAR-γ, pEC50: 8.56 (Human PPAR-γ)
  99.64%
FH535      
PPAR
99.93%
Pioglitazone
PPARα, EC50: 0.93 μM (Human PPARα)
PPARδ, EC50: 0.01 μM (Human PPARδ)
PPARγ, EC50: 43 μM (Human PPARγ)
  99.18%
GW0742
PPARα, EC50: 1.1 μM
PPARδ, EC50: 1 nM
PPARγ, EC50: 2 μM
  97.27%
Daidzein
PPAR-α
 
PPAR-γ
  99.66%
Magnolol    
PPARγ, EC50: 17.7 μM
  99.72%
GW7647
PPARα, EC50: 6 nM (Human PPARα)
PPARδ, EC50: 6.2 μM (Human PPARδ)
PPARγ, EC50: 1.1 μM (Human PPARγ)
  98.04%
5-Aminosalicylic Acid    
PPARγ
  >98.0%
Saroglitazar
PPARα, EC50: 0.65 pM (HepG2 cell)
 
PPARγ, EC50: 3 nM (HepG2 cell)
  98.03%
Astragalus polysaccharide    
PPAR-γ
  >98.0%
Lanifibranor
PPARα, EC50: 1537 nM (Human PPARα)
PPARδ, EC50: 866 nM (Human PPARδ)
PPARγ, EC50: 206 nM (Human PPARγ)
  98.89%
Palmitelaidic Acid
PPARα
      >99.0%
Seladelpar sodium salt  
PPAR-δ, EC50: 2 nM
    98.52%
Ginsenoside Rh1    
PPAR-γ
  >98.0%
Clofibrate
PPARα, EC50: 50 μM
 
PPARγ, EC50: 500 μM
  99.59%
Saroglitazar Magnesium
PPARα, EC50: 0.65 pM (HepG2 cell)
 
PPARγ, EC50: 3 nM (HepG2 cell)
  98.85%
Inolitazone dihydrochloride    
PPARγ
  99.21%
GSK3787  
PPARδ, pIC50: 6.6 nM
    96.67%
Astaxanthin    
PPARγ
  >98.0%
Rosiglitazone maleate    
PPARγ1, EC50: 30 nM
PPARγ2, EC50: 100 nM
  99.25%
NXT629
hPPARα, IC50: 77 nM
hPPARδ, IC50: 6 μM
hPPARγ, IC50: 15 μM
  99.05%
BMS-687453
PPARα, IC50: 260 nM (Human PPARα)
      99.04%
Fenofibric acid
PPARα, EC50: 22.4 μM
PPARδ, EC50: 1.06 μM
PPARγ, EC50: 1.47 μM
  99.38%
Eupatilin
PPARα
      99.01%
DG172 dihydrochloride  
PPARβ/δ, IC50: 27 nM
    99.70%
L-165041  
PPARδ, Ki: 6 nM
PPARγ, Ki: 730 nM
  99.14%
Ciprofibrate
PPARα
      99.62%
MA-0204  
PPARδ, EC50: 0.4 nM (in human)
PPARδ, EC50: 7.9 nM (in mouse)
PPARδ, EC50: 10 nM (in rat)
   
Oleoylethanolamide
PPAR-α
      >98.0%
Raspberry ketone
PPAR-α
      99.91%
Balaglitazone    
PPARγ, EC50: 351 nM (Human PPARγ)
  99.21%
Adelmidrol    
PPARγ
  >98.0%
Glabridin    
PPARγ, EC50: 6.1 μM
  99.98%
Indeglitazar
PPARα
PPARδ
PPARγ
  99.42%
Seladelpar
PPAR-α, EC50: 1600 nM
PPAR-δ, EC50: 2 nM
   
Aleglitazar
PPARα, IC50: 38 nM
 
PPARγ, IC50: 19 nM
  99.30%
Pemafibrate racemate
h-PPARα, EC50: 1 nM
h-PPARδ, EC50: 1.7 μM
   
Alpinetin    
PPAR-γ
 
Glabrone    
PPAR-γ
 
Gypenoside XLIX
PPAR-α
     
LJ570
PPARα, EC50: 1.05 μM
 
PPARγ, EC50: 0.12 μM
 
Pparδ agonist 1  
PPARδ, EC50: 5.06 nM
   
Ophiopogonin D
PPARα
     
Angeloylgomisin H    
PPAR-γ
 
Fonadelpar  
PPARδ
   
Agrimol B    
PPARγ
 
Pparδ agonist 2  
PPARδ
   
KD-3010  
PPARδ
   
13-Oxo-9E,11E-octadecadienoic acid
PPARα
     
Cefminox sodium    
PPARγ
 
Bilobetin
PPARα
     
Imiglitazar
PPARα, EC50: 67 nM
 
PPARγ1, EC50: 31 nM
 
Chiglitazar
PPARα, EC50: 1.8 μM
PPARδ, EC50: 1.7 μM
PPARγ, EC50: 0.08 μM
 
Ertiprotafib
PPARα, EC50: ~1 μM
PPARβ, EC50: ~1 μM
   
4-O-Methyl honokiol    
PPARγ
 
Inolitazone    
PPARγ
 
AVE-8134
PPARα, EC50: 100 nM (Human PPARα)
     
Arhalofenate    
PPAR-γ
 
PPARα-MO-1
PPARα
     
PPAR agonist 1
PPARα
 
PPARγ