1. Signaling Pathways
  2. Cell Cycle/DNA Damage
  3. PPAR
  4. PPAR Inhibitors

PPAR Inhibitors

PPARα

PPARβ/δ

PPARγ

PPAR

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

PPAR Inhibitors, Agonists, Antagonists, Activators & Modulators
Product Name PPARα PPARβ/δ PPARγ PPAR Purity
Retinoic acid
PPARα, Kd: 103 nM
PPARβ/δ, Kd: 17 nM
PPARγ, Kd: 178 nM
  99.74%
Rosiglitazone    
PPARγ1, EC50: 30 nM
PPARγ2, EC50: 100 nM
  99.54%
GW9662
PPARα, IC50: 32 nM
PPARδ, IC50: 2000 nM
PPARγ, IC50: 3.3 nM
  99.83%
Elafibranor
PPAR-α, EC50: 45 nM
PPAR-δ, EC50: 175 nM
    99.18%
GW 6471
PPARα
      98.98%
CUDA
PPARα
      >98.0%
Ciprofibrate impurity A
PPARα
     
Troglitazone    
PPARγ, EC50: 550 nM (Human PPARγ)
  99.53%
Pioglitazone
hPPARα, EC50: 100 μM
mouse PPARα, EC50: 100 μM
hPPARδ, EC50: 43 μM
hPPARγ, EC50: 0.93 μM
mouse PPARγ, EC50: 0.99 μM
  99.18%
T0070907
PPARα, Ki: 0.85 μM
PPARδ, Ki: 1.8 μM
PPARγ, Ki: 1 nM
  99.34%
Fenofibrate
PPARα, IC50: 30 μM
      99.92%
GW 501516  
PPARδ, EC50: 1.1 nM
    99.27%
Icariin
PPARα
      98.75%
Pirinixic acid
PPARα, EC50: 0.63 μM
 
PPARγ, EC50: 32 μM
  99.48%
5-Aminosalicylic Acid    
PPARγ
  >98.0%
CDDO-Im
PPARα, Ki: 232 nM
 
PPARγ, Ki: 344 nM
  98.20%
GW1929    
PPAR-γ, pEC50: 8.56 (Human PPAR-γ)
  99.77%
Daidzein
PPAR-α
 
PPAR-γ
  99.89%
Pioglitazone hydrochloride
PPARα, EC50: 0.93 μM (Human PPARα)
PPARδ, EC50: 0.01 μM (Human PPARδ)
PPARγ, EC50: 43 μM (Human PPARγ)
  96.39%
GW7647
PPARα, EC50: 6 nM (Human PPARα)
PPARδ, EC50: 6.2 μM (Human PPARδ)
PPARγ, EC50: 1.1 μM (Human PPARγ)
  98.04%
FH535      
PPAR
99.93%
GW0742
PPARα, EC50: 1.1 μM
PPARδ, EC50: 1 nM
PPARγ, EC50: 2 μM
  97.27%
Magnolol    
PPARγ, EC50: 17.7 μM
  99.72%
Bezafibrate
hPPARα, EC50: 50 μM
hPPARδ, EC50: 20 μM
hPPARγ, EC50: 60 μM
  99.43%
Astaxanthin    
PPARγ
  >98.0%
GSK3787  
PPARδ, pIC50: 6.6 nM
    99.04%
Lanifibranor
PPARα, EC50: 1537 nM (Human PPARα)
PPARδ, EC50: 866 nM (Human PPARδ)
PPARγ, EC50: 206 nM (Human PPARγ)
  98.89%
Ginsenoside Rh1    
PPAR-γ
  >98.0%
Rosiglitazone maleate    
PPARγ1, EC50: 30 nM
PPARγ2, EC50: 100 nM
  99.75%
Seladelpar sodium salt  
PPAR-δ, EC50: 2 nM
    98.52%
NXT629
hPPARα, IC50: 77 nM
hPPARδ, IC50: 6 μM
hPPARγ, IC50: 15 μM
  99.05%
Palmitelaidic Acid
PPARα
      >99.0%
Gemfibrozil
PPAR-α
      99.91%
Eupatilin
PPARα
      99.01%
Saroglitazar Magnesium
PPARα, EC50: 0.65 pM (HepG2 cell)
 
PPARγ, EC50: 3 nM (HepG2 cell)
  98.85%
Fenofibric acid
PPARα, EC50: 22.4 μM
PPARδ, EC50: 1.06 μM
PPARγ, EC50: 1.47 μM
  99.67%
Clofibrate
PPARα, EC50: 50 μM
 
PPARγ, EC50: 500 μM
  99.59%
Glabridin    
PPARγ, EC50: 6.1 μM
  99.98%
Inolitazone dihydrochloride    
PPARγ
  99.21%
Balaglitazone    
PPARγ, EC50: 351 nM (Human PPARγ)
  99.21%
L-165041  
PPARδ, Ki: 6 nM
PPARγ, Ki: 730 nM
  99.74%
Alpinetin    
PPAR-γ
  99.07%
Oleuropein    
PPARγ
  98.54%
Oleoylethanolamide
PPAR-α
      99.55%
MA-0204  
PPARδ, EC50: 0.4 nM (in human)
PPARδ, EC50: 7.9 nM (in mouse)
PPARδ, EC50: 10 nM (in rat)
    99.71%
DG172 dihydrochloride  
PPARβ/δ, IC50: 27 nM
    99.70%
BMS-687453
PPARα, IC50: 260 nM (Human PPARα)
      99.04%
Raspberry ketone
PPAR-α
      99.91%
Mifobate    
PPARγ, IC50: 140 μM
  >99.0%
Adelmidrol    
PPARγ
  >98.0%
Indeglitazar
PPARα
PPARδ
PPARγ
  99.42%
Ciprofibrate
PPARα
      99.79%
EHP-101    
PPARγ
  98.56%
Agrimol B    
PPARγ
  99.36%
Aleglitazar
PPARα, IC50: 38 nM
 
PPARγ, IC50: 19 nM
  99.30%
Gypenoside XLIX
PPAR-α
      >99.0%
15-Deoxy-Δ-12,14-prostaglandin J2    
PPARγ, EC50: 2 μM
 
Glabrone    
PPAR-γ
 
Caulophyllogenin    
PPARγ, EC50: 12.6 μM
 
Pparδ agonist 1  
PPARδ, EC50: 5.06 nM
   
Ophiopogonin D
PPARα
     
Angeloylgomisin H    
PPAR-γ
 
Fonadelpar  
PPARδ
   
KD-3010  
PPARδ
   
Ertiprotafib
PPARα, EC50: ~1 μM
PPARβ, EC50: ~1 μM
   
13-Oxo-9E,11E-octadecadienoic acid
PPARα
     
Cefminox sodium    
PPARγ
 
Mesalamine impurity P      
PPAR
Methyl oleanonate    
PPARγ
 
Bilobetin
PPARα
     
Licarin B    
PPARγ
 
Imiglitazar
PPARα, EC50: 67 nM
 
PPARγ1, EC50: 31 nM
 
4-O-Methyl honokiol    
PPARγ
 
Inolitazone    
PPARγ
 
Arhalofenate    
PPAR-γ
 
PPAR agonist 1
PPARα
 
PPARγ