1. Signaling Pathways
  2. GPCR/G Protein
    Neuronal Signaling
  3. mGluR
  4. mGluR Inhibitors

mGluR Inhibitors

mGluR8

mGluR6

mGluR7

mGluR5

mGluR4

mGluR2

mGluR3

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

mGluR Inhibitors, Agonists, Antagonists & Modulators
Product Name mGluR8 mGluR6 mGluR7 mGluR5 mGluR4 mGluR2 mGluR3 Purity
LY2794193          
mGluR2, EC50: 47.5
mGluR2, Ki: 412
mGluR3, EC50: 0.47 nM
mGluR3, Ki: 0.927 nM
99.88%
LY2812223          
mGluR2, Ki: 144 nM
mGluR3, Ki: 156 nM
>98.0%
CHPG sodium salt      
mGluR5
     
Foliglurax monohydrochloride        
mGlu4, EC50: 79 nM
    98.93%
L-APB
mGlu8, EC50: 0.29 μM
mGlu6, EC50: 1.0 μM
mGlu7, EC50: 249 μM
 
mGlu4, EC50: 0.13 μM
    >99.0%
Xanthurenic acid          
mGluR2
mGluR3
98.17%
(R)-ADX-47273      
mGluR5, EC50: 168 nM
      99.25%
VU6001376        
mGlu4, EC50: 50.1 nM
   
Foliglurax        
mGlu4, EC50: 79 nM
   
CHPG      
mGluR5
     
VU0652835      
mGluR5, IC50: 81 nM
     
VU0650786            
mGluR3, IC50: 392 nM
99.97%
LY3020371 hydrochloride          
mGluR2, Ki: 5.3 nM
mGluR3, Ki: 2.5 nM
Fenobam      
rat mGluR5, Kd: 54 nM
human mGluR5, Kd: 31 nM
      98.53%
LY 541850          
mGluR2, IC50: 0.161 μM
mGluR3, IC50: 1.05 μM