Culmerciclib maleate

Cat. No.: HY-147258A Purity: 99.52%: FAQs
Data Sheet SDS COA Handling Instructions

Molarity Calculator

Culmerciclib maleate is a cyclin dependent kinase (CDK) inhibitor, and has antineoplastic activity.

For research use only. We do not sell to patients.

Culmerciclib maleate Chemical Structure

CAS No. : 2197922-55-5

Size	Price	Stock	Quantity
Free Sample (0.1 - 0.5 mg)		Apply Now
5 mg	USD 215	In-stock	Estimated Time of Arrival: December 31
10 mg	USD 350	In-stock	Estimated Time of Arrival: December 31
25 mg	USD 700	In-stock	Estimated Time of Arrival: December 31
50 mg	USD 1120	In-stock	Estimated Time of Arrival: December 31
100 mg	USD 1800	In-stock	Estimated Time of Arrival: December 31
200 mg		Get quote
500 mg		Get quote

or Bulk Inquiry

* Please select Quantity before adding items.

This product is a controlled substance and not for sale in your territory.

Customer Review

Based on 1 publication(s) in Google Scholar

Featured Recommendations

•Related Screening Libraries:

•Related Small Molecules:

•Related Proteins:

Biological Activity
Purity & Documentation
References
Customer Review

Description

Culmerciclib maleate is a cyclin dependent kinase (CDK) inhibitor, and has antineoplastic activity^[1].

Molecular Weight

562.60

Formula

C₂₈H₃₁FN₈O₄

CAS No.

2197922-55-5

Appearance

Solid

Color

Light yellow to yellow

SMILES

OC(/C=C\C(O)=O)=O.CC(C1=C2C(C=CC(C3=NC(NC4=CC=C(N5CCNCC5)C=N4)=NC=C3F)=C2)=NN1C)C

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

-20°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Solvent & Solubility

In Vitro:

DMSO : 125 mg/mL (222.18 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

1 mM	1.7775 mL	8.8873 mL	17.7746 mL
5 mM	0.3555 mL	1.7775 mL	3.5549 mL
10 mM	0.1777 mL	0.8887 mL	1.7775 mL

View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Molarity Calculator
Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

In Vivo Dissolution Calculator

Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
(per animal)

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.

Calculation results:

Working solution concentration: mg/mL

Purity & Documentation

Purity: 99.52%

Select Batch:

Data Sheet (264 KB) SDS (251 KB)

COA (244 KB) HNMR (305 KB) LCMS (93 KB)

Handling Instructions (2659 KB)

References

[1]. International Nonproprietary Names for Pharmaceutical Substances (INN)

Complete Stock Solution Preparation Table

Optional Solvent	Concentration Solvent Mass	1 mg	5 mg	10 mg	25 mg

DMSO	1 mM	1.7775 mL	8.8873 mL	17.7746 mL	44.4365 mL
	5 mM	0.3555 mL	1.7775 mL	3.5549 mL	8.8873 mL
	10 mM	0.1777 mL	0.8887 mL	1.7775 mL	4.4437 mL
	15 mM	0.1185 mL	0.5925 mL	1.1850 mL	2.9624 mL
	20 mM	0.0889 mL	0.4444 mL	0.8887 mL	2.2218 mL
	25 mM	0.0711 mL	0.3555 mL	0.7110 mL	1.7775 mL
	30 mM	0.0592 mL	0.2962 mL	0.5925 mL	1.4812 mL
	40 mM	0.0444 mL	0.2222 mL	0.4444 mL	1.1109 mL
	50 mM	0.0355 mL	0.1777 mL	0.3555 mL	0.8887 mL
	60 mM	0.0296 mL	0.1481 mL	0.2962 mL	0.7406 mL
	80 mM	0.0222 mL	0.1111 mL	0.2222 mL	0.5555 mL
	100 mM	0.0178 mL	0.0889 mL	0.1777 mL	0.4444 mL