1. Epigenetics
  2. Histone Methyltransferase
  3. EZH2-IN-8

EZH2-IN-8 

Cat. No.: HY-142951
Handling Instructions

EZH2-IN-8 is a potent inhibitor of EZH2. EZH2 overexpression or mutations in the SET region (Y641F, Y641N, A687V, A677G point mutations) all lead to abnormal elevation of H3K27me3 and promote the growth and development of many types of tumors, such as breast cancer, prostate cancer, leukemia, etc. EZH2-IN-8 has the potential for the research of cancer diseases (extracted from patent WO2021129629A1, compound 265).

For research use only. We do not sell to patients.

EZH2-IN-8 Chemical Structure

EZH2-IN-8 Chemical Structure

CAS No. : 2659225-08-6

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Description

EZH2-IN-8 is a potent inhibitor of EZH2. EZH2 overexpression or mutations in the SET region (Y641F, Y641N, A687V, A677G point mutations) all lead to abnormal elevation of H3K27me3 and promote the growth and development of many types of tumors, such as breast cancer, prostate cancer, leukemia, etc. EZH2-IN-8 has the potential for the research of cancer diseases (extracted from patent WO2021129629A1, compound 265)[1].

Molecular Weight

570.74

Formula

C31H40F2N4O2S

CAS No.
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Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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EZH2-IN-8
Cat. No.:
HY-142951
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