1. Metabolic Enzyme/Protease
  2. FABP
  3. FABP5-IN-1

FABP5-IN-1 

Cat. No.: HY-129910
Handling Instructions

FABP5-IN-1(Compounds 4j) is a selective and high affinity fatty acid binding protein 5 (FABP5) inhibitor with a Ki value of 1.7 μM, and does not bind to both FABP3 and FABP7. FABP5-IN-1 shows potent antinociceptive effects.

For research use only. We do not sell to patients.

FABP5-IN-1 Chemical Structure

FABP5-IN-1 Chemical Structure

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Description

FABP5-IN-1(Compounds 4j) is a selective and high affinity fatty acid binding protein 5 (FABP5) inhibitor with a Ki value of 1.7 μM, and does not bind to both FABP3 and FABP7. FABP5-IN-1 shows potent antinociceptive effects[1].

IC50 & Target

Ki: 1.7 μM (FABP5)[1]

In Vivo

FABP5-IN-1 (Compounds 4j; 20 mg/kg; intraperitoneal injection; for 90 minutes; male wild-type C57BL/6 mice) treatment displays potent antinociceptive effects in CFA model[1].

Animal Model: Male wild-type C57BL/6 mice injected with complete Freund’s adjuvant (CFA)[1]
Dosage: 20 mg/kg
Administration: Intraperitoneal injection; for 90 minutes
Result: Displayed potent antinociceptive effects in CFA model.
Molecular Weight

534.60

Formula

C₃₄H₃₀O₆

SMILES

O=C(OCC1C(C=CC=C2)=C2C3=C1C=CC=C3)[[email protected]]4[[email protected]@H](C5=CC=CC=C5OC)[[email protected]](C(O)=O)[[email protected]@H]4C6=CC=CC=C6OC

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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KeyWords:

FABP5-IN-1 | FABP | Fatty acid-binding protein | Inhibitor | inhibitor | inhibit

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FABP5-IN-1
Cat. No.:
HY-129910
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