1. GPCR/G Protein
    Neuronal Signaling
  2. Somatostatin Receptor
  3. Paltusotine

Paltusotine (Synonyms: CRN00808)

Cat. No.: HY-109155 Purity: 99.06%
Handling Instructions

Paltusotine (CRN00808) is an orally active, nonpeptide selective somatostatin type 2 (SST2) receptor agonist. Paltusotine has the potential for maintaining GH and IGF-1 levels after depot somatostatin receptor ligand therapy.

For research use only. We do not sell to patients.

Paltusotine Chemical Structure

Paltusotine Chemical Structure

CAS No. : 2172870-89-0

Size Price Stock Quantity
5 mg USD 760 In-stock
Estimated Time of Arrival: December 31
10 mg USD 1150 In-stock
Estimated Time of Arrival: December 31
25 mg USD 2300 In-stock
Estimated Time of Arrival: December 31
50 mg USD 3650 In-stock
Estimated Time of Arrival: December 31
100 mg USD 5400 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

* Please select Quantity before adding items.

Customer Review

Based on 1 publication(s) in Google Scholar

Top Publications Citing Use of Products
  • Biological Activity

  • Purity & Documentation

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  • Customer Review

Description

Paltusotine (CRN00808) is an orally active, nonpeptide selective somatostatin type 2 (SST2) receptor agonist. Paltusotine has the potential for maintaining GH and IGF-1 levels after depot somatostatin receptor ligand therapy[1][2].

Clinical Trial
Molecular Weight

456.49

Formula

C27H22F2N4O

CAS No.
SMILES

N#CC1=CC=CC(C2=CC=C3N=CC(C4=CC(F)=CC(F)=C4)=C(N5CCC(N)CC5)C3=C2)=C1O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 20 mg/mL (43.81 mM; ultrasonic and warming and heat to 60°C)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.1906 mL 10.9531 mL 21.9063 mL
5 mM 0.4381 mL 2.1906 mL 4.3813 mL
10 mM 0.2191 mL 1.0953 mL 2.1906 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.5 mg/mL (5.48 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2 mg/mL (4.38 mM); Clear solution

*All of the co-solvents are available by MCE.
Purity & Documentation

Purity: 99.06%

References
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The dilution calculator equation

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This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
Paltusotine
Cat. No.:
HY-109155
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