1. GPCR/G Protein
  2. Leukotriene Receptor
  3. Pranlukast-d5

Pranlukast-d5 

Cat. No.: HY-B0290S
Handling Instructions

Pranlukast-d5 (ONO-1078-d5) is the deuterium labeled Pranlukast. Pranlukast is a highly potent, selective and competitive antagonist of peptide leukotrienes. Pranlukast inhibits [3H]LTE4, [3H]LTD4, and [3H]LTC4 bindings to lung membranes with Kis of 0.63, 0.99, and 5640 nM, respectively.

For research use only. We do not sell to patients.

Pranlukast-d5 Chemical Structure

Pranlukast-d5 Chemical Structure

CAS No. : 1216719-50-4

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Description

Pranlukast-d5 (ONO-1078-d5) is the deuterium labeled Pranlukast. Pranlukast is a highly potent, selective and competitive antagonist of peptide leukotrienes. Pranlukast inhibits [3H]LTE4, [3H]LTD4, and [3H]LTC4 bindings to lung membranes with Kis of 0.63, 0.99, and 5640 nM, respectively.

In Vitro

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

486.53

Formula

C₂₇H₁₈D₅N₅O₄

CAS No.
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Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Pranlukast-d5
Cat. No.:
HY-B0290S
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