1. TGF-beta/Smad
  2. TGF-β Receptor
  3. San78-130

San78-130 

Cat. No.: HY-101113
Handling Instructions

San78-130 is a selective and potent ALK1 inhibitor with an IC50 of 62 nM. San78-130 also inhibits FLT4/VEGFR3, KDR/VEGFR2, MEK2, and FLT3 with IC50s of 114, 162, 186.7, and 188 nM, respectively.

For research use only. We do not sell to patients.

San78-130 Chemical Structure

San78-130 Chemical Structure

CAS No. : 66018-45-9

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Description

San78-130 is a selective and potent ALK1 inhibitor with an IC50 of 62 nM. San78-130 also inhibits FLT4/VEGFR3, KDR/VEGFR2, MEK2, and FLT3 with IC50s of 114, 162, 186.7, and 188 nM, respectively[1].

IC50 & Target[1]

ALK1

62 nM (IC50)

FLT4/VEGFR3

114 nM (IC50)

KDR/VEGFR2

162 nM (IC50)

MEK2

186.7 nM (IC50)

FLT3

188 nM (IC50)

Molecular Weight

366.41

Formula

C₁₉H₂₆O₇

CAS No.

66018-45-9

SMILES

OC1=CC(OC)=CC(CCC[[email protected]@H]([[email protected]](O)C(CCC[[email protected]](C)O2)=O)O)=C1C2=O

Shipping

Room temperature in continental US; may vary elsewhere

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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