1. Search Result

Search Result

Targets Recommended: PI4K MAP4K Oct3/4 FXR Serotonin Transporter
Results for "


" in MCE Product Catalog:
Cat. No. Product Name Target Research Areas
  • HY-141547

    Sodium Channel Cytochrome P450 Inflammation/Immunology
    Nav1.7-IN-8 is a potent blockage of NaV1.7 with high selectivity for the inhibition of NaV1.7 over the subtypes hNaV1.1 and hNaV1.5. Nav1.7-IN-8 inhibits CYP2C9 and CYP3A4 with an IC50 of 0.17 μM and 0.077 μM, respectively. Nav1.7-IN-8 displays significant analgesic effects in rodent models of acute and inflammatory pain.