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Targets Recommended: NEDD8-activating Enzyme

Results for "2474876-09-8" in MCE Product Catalog:

Cat. No. Product Name Target Research Areas
  • HY-136571
    GSK046

    iBET-BD2

    Epigenetic Reader Domain Inflammation/Immunology
    GSK046 (iBET-BD2) is a potent, selective and orally active BD2 bromodomain inhibitor of the BET proteins, with IC50s of 264 nM (BRD2 BD2), 98 nM (BRD3 BD2), 49 nM (BRD4 BD2) and 214 nM (BRDT BD2), respectively. GSK046 has immunomodulatory activity.