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Results for "

Baclofen

" in MedChemExpress (MCE) Product Catalog:

12

Inhibitors & Agonists

1

Peptides

1

Isotope-Labeled Compounds

Cat. No. Product Name Target Research Areas Chemical Structure
  • HY-B0007
    Baclofen
    4 Publications Verification

    		 GABA Receptor Neurological Disease
    Baclofen, a lipophilic derivative of γ-aminobutyric acid (GABA), is an orally active, selective metabotropic GABAB receptor (GABABR) agonist. Baclofen mimics the action of GABA and produces slow presynaptic inhibition through the GABAB receptor. Baclofen has high blood brain barrier penetrance. Baclofen has the potential for muscle spasticity research .
    <em>Baclofen</em>
  • HY-B0007S
    Baclofen-d4

    		GABA Receptor Neurological Disease
    Baclofen-d4 is the deuterium labeled Baclofen. Baclofen, a lipophilic derivative of γ-aminobutyric acid (GABA), is an orally active, selective metabotropic GABAB receptor (GABABR) agonist. Baclofen mimics the action of GABA and produces slow presynaptic inhibition through the GABAB receptor. Baclofen has high blood brain barrier penetrance. Baclofen has the potential for muscle spasticity research[1][2][3].
    <em>Baclofen</em>-d4
  • HY-17354
    (R)-Baclofen
    2 Publications Verification

    ArBaclofen; STX209

    		 GABA Receptor Neurological Disease
    (R)-Baclofen (Arbaclofen) is a selective GABAB receptor agonist .
    (R)-<em>Baclofen</em>
  • HY-B0007R
    Baclofen (Standard)

    		GABA Receptor Neurological Disease
    Baclofen (Standard) is the analytical standard of Baclofen. This product is intended for research and analytical applications. Baclofen, a lipophilic derivative of γ-aminobutyric acid (GABA), is an orally active, selective metabotropic GABAB receptor (GABABR) agonist. Baclofen mimics the action of GABA and produces slow presynaptic inhibition through the GABAB receptor. Baclofen has high blood brain barrier penetrance. Baclofen has the potential for muscle spasticity research .
    <em>Baclofen</em> (Standard)
  • HY-B0007C
    Baclofen hydrochloride

    		GABA Receptor Neurological Disease
    Baclofen hydrochloride, a lipophilic derivative of γ-aminobutyric acid (GABA), is an orally active, selective metabotropic GABAB receptor (GABABR) agonist. Baclofen hydrochloride mimics the action of GABA and produces slow presynaptic inhibition through the GABAB receptor. Baclofen hydrochloride has high blood brain barrier penetrance. Baclofen hydrochloride has the potential for muscle spasticity research .
    <em>Baclofen</em> hydrochloride
  • HY-17354A
    (R)-Baclofen hydrochloride

    ArBaclofen hydrochloride; STX 209 hydrochloride

    		 GABA Receptor Neurological Disease
    (R)-Baclofen hydrochloride (Arbaclofen hydrochloride) is a selective GABAB receptor agonist .
    (R)-<em>Baclofen</em> hydrochloride
  • HY-14735
    Arbaclofen placarbil

    XP 19986

    		 GABA Receptor Neurological Disease
    Arbaclofen placarbil is a novel transported proagent of the active R-isomer of baclofen. Baclofen is a racemic GABAB receptor agonist
    Arbaclofen placarbil
  • HY-100798
    Phaclofen

    Phaclofen is a selective GABAB receptor antagonist. Phaclofen is a peripheral and central baclofen antagonist. Phaclofen maybe a potential compound in determining the physiological significance of central and peripheral bicuculline-insensitive receptors with which GABA and (-)-baclofen interact .
    Phaclofen
  • HY-103516
    CGP55845 hydrochloride

    		GABA Receptor Neurological Disease
    CGP55845 hydrochloride is a potent and selective GABAB receptor antagonist with an IC50 of 6 nM. CGP55845 hydrochloride can be used for neurological research .
    CGP55845 hydrochloride
  • HY-W105694
    3-Aminopropylphosphonic acid

    (3-Aminopropyl)phosphonic acid

    		 GABA Receptor Neurological Disease
    3-Aminopropylphosphonic acid is a GABAB receptor agonist with IC50 value of 1.5 μM .
    3-Aminopropylphosphonic acid
  • HY-103532
    CGP46381

    		GABA Receptor Neurological Disease
    CGP 46381 is an orally active GABAB receptor antagonist with IC50 of 4.9 μM. CGP 46381 blocks the neuronal depression induced by iontophoretically applied baclofen (HY-B0007) .
    CGP46381
  • HY-103502
    CGP7930

    		GABA Receptor Neurological Disease
    CGP7930 (3-(3’,5’-Di-tert-butyl-4’-hydroxy) phenyl-2, 2-dimethylpropanol) is a positive metabotropic GABAB receptor allosteric modulator. CGP7930 enhances the inhibitory effect of l-baclofen on the oscillatory activity of cultured cortical neurons .
    CGP7930

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