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Oxazoloazepin

" in MedChemExpress (MCE) Product Catalog:
Cat. No. Product Name Target Research Areas Chemical Structure
  • HY-103212

    B-HT 933 dihydrochloride; Oxazoloazepin dihydrochloride

    Adrenergic Receptor Cardiovascular Disease Endocrinology
    Azepexole (B-HT 933) dihydrochloride is a potent and selective alpha 2-adrenoceptor agonist with pKis of 8.3, 7.6, and 7.5 for α2A-, α2B- and α2C-adrenoceptor subtypes, resepctively . Azepexole dihydrochloride causes concentration-dependent inhibition of peristaltic contractions (IC50= 78.72 nM) .
    Azepexole dihydrochloride

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