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Results for "

Paliperidone

" in MedChemExpress (MCE) Product Catalog:

3

Inhibitors & Agonists

1

Natural
Products

1

Isotope-Labeled Compounds

Cat. No. Product Name Target Research Areas Chemical Structure
  • HY-A0019
    Paliperidone
    1 Publications Verification

    9-Hydroxyrisperidone

    Dopamine Receptor 5-HT Receptor Adrenergic Receptor Neurological Disease
    Paliperidone (9-Hydroxyrisperidone), the major active metabolite of Risperidone, is a dopamine D2 antagonist and 5-HT2A antagonist. Paliperidone is also active as an antagonist at α1 and α2 adrenergic receptors and H1-histaminergic receptors. Paliperidone, a antipsychotic agent, shows efficacy against schizophrenia .
    <em>Paliperidone</em>
  • HY-A0019S

    Dopamine Receptor 5-HT Receptor Adrenergic Receptor Neurological Disease
    Paliperidone-d4 is the deuterium labeled Paliperidone. Paliperidone (9-Hydroxyrisperidone), the major active metabolite of Risperidone, is a dopamine D2 antagonist and 5-HT2A antagonist. Paliperidone is also active as an antagonist at α1 and α2 adrenergic receptors and H1-histaminergic receptors. Paliperidone, a antipsychotic agent, shows efficacy against schizophrenia[1].
    <em>Paliperidone</em>-d4
  • HY-A0019A

    9-Hydroxyrisperidone palmitate

    Dopamine Receptor 5-HT Receptor Neurological Disease
    Paliperidone palmitate (9-Hydroxyrisperidone palmitate), an atypical long-acting antipsychotic agent, is an ester proagent of Paliperidone. Paliperidone is a dopamine antagonist and 5-HT2A antagonist of the atypical antipsychotic class. Paliperidone palmitate shows efficacy against schizophrenia .
    <em>Paliperidone</em> palmitate

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