1. TGF-beta/Smad
  2. TGF-β Receptor
  3. TGFβRI-IN-3

TGFβRI-IN-3 

Cat. No.: HY-132290
Handling Instructions

TGFβRI-IN-3 inhibits TGFβR1 at an IC50 of 0.79 nM with 2000-fold selectivity against MAP4K4. TGFβRI-IN-3 represents a highly selective TGFβR1 inhibitor that has potential applications in immuno-oncology.

For research use only. We do not sell to patients.

TGFβRI-IN-3 Chemical Structure

TGFβRI-IN-3 Chemical Structure

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Description

TGFβRI-IN-3 inhibits TGFβR1 at an IC50 of 0.79 nM with 2000-fold selectivity against MAP4K4. TGFβRI-IN-3 represents a highly selective TGFβR1 inhibitor that has potential applications in immuno-oncology[1].

IC50 & Target

IC50: 0.79 nM (TGFβR1)[1]

In Vitro

TGFβRI-IN-3 inhibits TGFβR1 at an IC50 of 0.79 nM with 2000-fold selectivity against MAP4K4[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

465.57

Formula

C₂₈H₂₃N₃O₂S

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Product Name:
TGFβRI-IN-3
Cat. No.:
HY-132290
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