1. Screening Libraries
  2. Virtual Screening
  3. Allosteric Kinase Library

Allosteric Kinase Library

Cat. No.: HY-L0063V

Allosteric kinase inhibition is among the most promising and sensitive deactivation mechanism of kinase activity. A unique collection of 4,800 carefully selected molecules via docking and visual evaluation has been offered.

Allosteric Kinase Library
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100 μL/well (10 mM solution) Get quote In-stock

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Description
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Advantages

•   A unique collection of 4,800 carefully selected molecules via docking and visual evaluation.

•   Four type of possible allosteric kinase pockets were determined by now: 1) Myristoyl pocket; 2) Inhibitor binding mode that occupies part of binding pocket adjacent to the ATP-site; 3) PIF-pocket (regulatory site targeted); 4) pocket type I 1/2 relatively allosteric regulators of kinases (library contains 500 such compounds, only).

•   Structurally diverse.

•   No PAINS (Pan Assay Interference Compounds).

•   NMR and HPLC validated to ensure high purity and quality.

•   All compounds can be readily followed with analogues either from stock or from new syntheses.

•   Databases and compounds are provided by Enamine.

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Allosteric Kinase Library
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