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Signaling Pathway

WH-4-023

HY-12299

(Dual LCK/SRC inhibitor)

WH-4-023

WH-4-023 Chemical Structure

WH-4-023 is a potent and selective dual Lck/Src inhibitor with IC50 of 2 nM/6 nM for Lck and Src kinase respectively; little inhibition on p38α and KDR.

Size Price Stock Quantity
Free sample   Apply now  
10 mM * 1 mL in DMSO $100 In-stock
5 mg $80 In-stock
10 mg $120 In-stock
50 mg $400 In-stock
100 mg $650 In-stock
200 mg Get quote
500 mg Get quote
Size Price Stock Quantity
Free sample   Apply now  
10 mM * 1 mL in DMSO €98 In-stock
5 mg €78 In-stock
10 mg €118 In-stock
50 mg €392 In-stock
100 mg €637 In-stock
200 mg Get quote
500 mg Get quote

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Inquiry Information
Product name: WH-4-023
Cat. No.: HY-12299

WH-4-023 Data Sheet

  • View current batch:

    Purity: 99.93%

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    DataSheet

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    MSDS

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    COA

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    NMR

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    LCMS

Related Compound Libraries

Biological Activity of WH-4-023

WH-4-023 is a potent and selective dual Lck/Src inhibitor with IC50 of 2 nM/6 nM for Lck and Src kinase respectively; little inhibition on p38α and KDR.
IC50 value: 2 nM/6 nM(Lck/Src) [1]
Target: Lck/Src inhibitor

Protocol (Extracted from published papers and Only for reference)

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Chemical Information

M.Wt 568.67 Storage Please store the product under the recommended conditions in the Certificate of Analysis.
Formula C32H36N6O4
CAS No 837422-57-8
Solvent & Solubility

DMSO: ≥ 46.8 mg/mL

Preparing Stock Solutions

1 mg 5 mg 10 mg
1 mM 1.7585 mL 8.7924 mL 17.5849 mL
5 mM 0.3517 mL 1.7585 mL 3.5170 mL
10 mM 0.1758 mL 0.8792 mL 1.7585 mL

References on WH-4-023

Inhibitor Kit

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