1. Signaling Pathways
  2. Protein Tyrosine Kinase/RTK
  3. Discoidin Domain Receptor
  4. Discoidin Domain Receptor Inhibitors

Discoidin Domain Receptor Inhibitors

DDR1

DDR2

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Discoidin Domain Receptor Inhibitors
Product Name DDR1 DDR2 Purity
Sitravatinib
DDR1, IC50: 29 nM
DDR2, IC50: 0.5 nM
99.59%
WRG-28  
DDR2, IC50: 230 nM
99.34%
VU6015929
DDR1, IC50: 4.67 nM
DDR2, IC50: 7.39 nM
99.26%
DDR1-IN-6
DDR1, IC50: 9.72 nM
  98.16%
FGFR1/DDR2 inhibitor 1  
DDR2, IC50: 3.2 nM
98.26%
DDR1-IN-4
DDR1, IC50: 29 nM
DDR2, IC50: 1900 nM
98.01%
DDR1-IN-5
DDR1, IC50: 7.36 nM
  99.27%
Sitravatinib malate
DDR1, IC50: 29 nM
DDR2, IC50: 0.5 nM
DDR1-IN-1 dihydrochloride
DDR1, IC50: 105 nM
DDR2, IC50: 413 nM
DDR1/2 inhibitor-2
DDR1
DDR2
ML786 dihydrochloride  
DDR2, IC50: 7.0 nM
DDR1-IN-8
DDR1
DDR2