2. Membrane Transporter/Ion Channel
  3. CFTR
  4. Astressin 2B TFA

Astressin 2B TFA is a potent and selective corticotropin-releasing factor receptor 2 (CRF2) antagonist, with the IC50 values of 1.3 nM and > 500 nM for CRF2 and CRF1, respectively. Astressin 2B TFA antagonizes CRF2-mediated inhibition of gastric emptying.

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Astressin 2B TFA Chemical Structure

Astressin 2B TFA Chemical Structure

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Other Forms of Astressin 2B TFA:

Astressin 2B TFA Related Antibodies

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Description

Astressin 2B TFA is a potent and selective corticotropin-releasing factor receptor 2 (CRF2) antagonist, with the IC50 values of 1.3 nM and > 500 nM for CRF2 and CRF1, respectively. Astressin 2B TFA antagonizes CRF2-mediated inhibition of gastric emptying[1][2][3].

Molecular Weight

4041.69 (free base)

Formula

C183H307N49O53.xC2HF3O2
Appearance

Solid

Sequence

Ac-Asp-Leu-Ser-{d-Phe}-His-{a-methyl-Leu}-Leu-Arg-Lys-{Nle}-Ile-Glu-Ile-Glu-Lys-Gln-Glu-Lys-Glu-Lys-Gln-Gln-Ala-{g-Glu}-Asn-Asn-Leu-Leu-Leu-Asp-{a-methyl-Leu}-Ile-NH2 (Lactam bridge: Glu24-Lys27)
Sequence Shortening

Ac-Asp-LS-{d-Phe}-H-{a-methyl-Leu}-LRK-{Nle}-IEIEKQEKEKQQA-{g-Glu}-NNKLLLD-{a-methyl-Leu}-I-NH2 (Lactam bridge:Glu24-Lys27)
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Sealed storage, away from moisture and light

Powder -80°C 2 years
-20°C 1 year

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)

Purity & Documentation
References
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Astressin 2B TFA Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Astressin 2BCFTRCystic fibrosis transmembrane conductance regulatorcorticotropin-releasing factor receptorgastric emptyingendogenous peptide agonistInhibitorinhibitorinhibit

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