2. Epigenetics
  3. Histone Methyltransferase
  4. DCPT1061 hydrochloride

DCPT1061 hydrochloride has a strong inhibitory effect on PRMT1, PRMT6, and PRMT8 in vitro, The epigenetic enzymes such as PRMT3, PRMT4 and PRMT5 had little inhibitory effect. DCPT1061 hydrochloride has antitumor effects.

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DCPT1061 hydrochloride Chemical Structure

DCPT1061 hydrochloride Chemical Structure

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Based on 1 publication(s) in Google Scholar

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Description

DCPT1061 hydrochloride has a strong inhibitory effect on PRMT1, PRMT6, and PRMT8 in vitro, The epigenetic enzymes such as PRMT3, PRMT4 and PRMT5 had little inhibitory effect. DCPT1061 hydrochloride has antitumor effects[1][2].

Molecular Weight

375.72

Formula

C17H21Cl3N2O
Appearance

Solid

Color

White to off-white

SMILES

ClC1=C(OC2=CC=CC=C2CN(C)CCNC)C=CC=C1Cl.[H]Cl
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

-20°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Solvent & Solubility
In Vitro: 

DMSO : 50 mg/mL (133.08 mM; ultrasonic and warming and heat to 60°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.6616 mL 13.3078 mL 26.6156 mL
5 mM 0.5323 mL 2.6616 mL 5.3231 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

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In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

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Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Purity & Documentation
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.6616 mL 13.3078 mL 26.6156 mL 66.5389 mL
5 mM 0.5323 mL 2.6616 mL 5.3231 mL 13.3078 mL
10 mM 0.2662 mL 1.3308 mL 2.6616 mL 6.6539 mL
15 mM 0.1774 mL 0.8872 mL 1.7744 mL 4.4359 mL
20 mM 0.1331 mL 0.6654 mL 1.3308 mL 3.3269 mL
25 mM 0.1065 mL 0.5323 mL 1.0646 mL 2.6616 mL
30 mM 0.0887 mL 0.4436 mL 0.8872 mL 2.2180 mL
40 mM 0.0665 mL 0.3327 mL 0.6654 mL 1.6635 mL
50 mM 0.0532 mL 0.2662 mL 0.5323 mL 1.3308 mL
60 mM 0.0444 mL 0.2218 mL 0.4436 mL 1.1090 mL
80 mM 0.0333 mL 0.1663 mL 0.3327 mL 0.8317 mL
100 mM 0.0266 mL 0.1331 mL 0.2662 mL 0.6654 mL
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DCPT1061 hydrochloride Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

DCPT1061DCPT 1061DCPT-1061Histone MethyltransferaseInhibitorAntitumorPRMTinhibitorinhibit

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