1. Apoptosis Protein Tyrosine Kinase/RTK
  2. Discoidin Domain Receptor c-Kit PDGFR c-Myc
  3. GW694590A

GW694590A (UNC10112731) is a MYC protein stabilizer that increases endogenous MYC protein levels. GW694590A also targets receptor tyrosine kinases, inhibiting DDR2, KIT and PDGFRα by 81% at 1 μM. , 68% and 67%. GW694590A is a protein kinase inhibitor across ATP-dependent and -independent luciferases with potential effects on the Fluc reporter gene.

For research use only. We do not sell to patients.

GW694590A Chemical Structure

GW694590A Chemical Structure

CAS No. : 948313-24-4

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Description

GW694590A (UNC10112731) is a MYC protein stabilizer that increases endogenous MYC protein levels. GW694590A also targets receptor tyrosine kinases, inhibiting DDR2, KIT and PDGFRα by 81% at 1 μM. , 68% and 67%. GW694590A is a protein kinase inhibitor across ATP-dependent and -independent luciferases with potential effects on the Fluc reporter gene[1].

Molecular Weight

417.42

Formula

C22H19N5O4

CAS No.
SMILES

O=C(NC1=CC=C(OC2=CC3=C(NC(NC(OC)=O)=N3)C=C2)C=C1)NC4=CC=CC=C4

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Room temperature in continental US; may vary elsewhere.

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Please store the product under the recommended conditions in the Certificate of Analysis.

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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GW694590A
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HY-160689
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