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Results for "

UM-1

" in MedChemExpress (MCE) Product Catalog:

12

Inhibitors & Agonists

1

Fluorescent Dye

3

Peptides

Cat. No. Product Name Target Research Areas Chemical Structure
  • HY-129042
    Cibacron Blue 3G-A
    1 Publications Verification

    		 Fluorescent Dye Beta-lactamase Infection
    Cibacron Blue 3G-A is an anthraquinone dye, inhibits the R46 β-lactamase with a Ki value of 1.2 uM .
    Cibacron Blue 3G-A
  • HY-122577
    EN40

    		Aldehyde Dehydrogenase (ALDH) Cancer
    EN40 is a potent, selective aldehyde dehydrogenase 3A1 (ALDH3A1) inhibitor as a covalent ligand, exhibits an IC50 value of 2 uM
    EN40
  • HY-15887
    MG 149
    Maximum Cited Publications
    11 Publications Verification

    Tip60 HAT inhibitor

    		 Histone Acetyltransferase Epigenetic Reader Domain Apoptosis Cancer
    MG149 (Tip60 HAT inhibitor) is a selective and potent Tip60 inhibitor with IC50 of 74 uM, similar potentcy for MOF (IC50= 47 uM); little potent for PCAF and p300 (IC50 >200 uM) .
    MG 149
  • HY-160754
    UM-1

    		Endogenous Metabolite Others
    UM-1 is the urinary 4-hydroxymethyl metabolite of DX-8951 (HY-13631) in human [1].
    <em>UM-1</em>
  • HY-P5562
    PP102

    		Bacterial Infection
    PP102 is an antimicrobial peptide is active against gram-positive B. subtilis (MIC: 25 uM), S. aureus (MIC: 13.3 uM), S. lutea (MIC: 63 uM), and B. pumilu (MIC: 23 uM) .
    PP102
  • HY-111772A
    (R)-Elexacaftor

    (R)-VX-445

    		 CFTR Inflammation/Immunology
    (R)-Elexacaftor is an enantiomer of Elexacaftor (HY-111772). (R)-Elexacaftor is the Compound 37 from patent WO2018107100A1. (R)-Elexacaftor is a modulator of cystic fibrosis transmembrane conductance regulator (CFTR), the EC50 for CFTR dF508 is 0.29 uM .
    (R)-Elexacaftor
  • HY-102019
    NSC61610

    		Interleukin Related Inflammation/Immunology
    NSC61610 disrupts hIL-18 binding to the ectromelia virus IL-18BP. NSC61610 inhibits hIL-18:ectvIL-18BP complex formation with an IC50 about 6 uM .
    NSC61610
  • HY-123905A
    LIN28 inhibitor LI71 enantiomer

    		Others Cancer
    LIN28 inhibitor LI71 enantiomer is the enantiomer of LIN28 inhibitor LI71 with less active. LIN28 inhibitor LI71 is a potent and cell-permeable LIN28 inhibitor, which abolishes LIN28-mediated oligouridylation with an IC50 of 7 uM .
    LIN28 inhibitor LI71 enantiomer
  • HY-117535
    CDK2-IN-4
    2 Publications Verification

    		 CDK Cancer
    CDK2-IN-4 (compound 73) is a potent and selective CDK2 inhibitor with an IC50 of 44 nM for CDK2/cyclin A, shows 2,000-fold selectivity over CDK1/cyclin B (IC50=86 uM) .
    CDK2-IN-4
  • HY-P5563
    PP113

    		Bacterial Infection
    PP113 is an antimicrobial peptide is active against Gram-negative and Gram-positive bacteria, E.coli (MIC: 73.3 uM), B. subtilis (MIC: 23.3 uM), S. aureus (MIC: 13 uM), S. lutea (MIC: 16.7 uM), and B. pumilu (MIC: 23.3 uM) .
    PP113
  • HY-P5560
    PP13

    		Bacterial Infection
    PP13 is an antimicrobial peptide, and is active against Gram-negative and Gram-positive bacteria E.coli (MIC: 16.7 uM), B. subtilis (MIC: 13.3 uM), S. aureus (MIC: 23.3 uM), S. lutea (MIC: 8.0 uM), and B. pumilu (MIC: 9.0 uM) .
    PP13
  • HY-125236
    BET-IN-19

    		Epigenetic Reader Domain Cancer
    BET-IN-19 (Compound 146) is a BET inhibitor. BET-IN-19 inhibits hlL-6 mRNA transcription (IC50 ≤ 0.3 uM), and c-myc activity in human AML MV4-11 cell (IC50 ≤ 0.3 uM)。BET-IN-19 inhibits tetra-acetylated histone H4 binding to BRD4 bromodomain 1 (IC50 ≤ 0.3 uM) .
    BET-IN-19

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