1. Signaling Pathways
  2. Vitamin D Related/Nuclear Receptor
  3. Nuclear Hormone Receptor 4A/NR4A

Nuclear Hormone Receptor 4A/NR4A

Nerve Growth Factor IB-like Receptor

 

Nuclear Hormone Receptor 4A/NR4A Related Products (22):

Cat. No. Product Name Effect Purity Chemical Structure
  • HY-149608
    Nurr1 agonist 5
    Agonist
    Nurr1 agonist 5 (compound 5o) is a neuroprotective transcription factor Nurr1 agonist with a Kd of 0.5 μM and an EC50 of 3 μM.
    Nurr1 agonist 5
  • HY-B1322AS1
    Amodiaquine-d10 hydrochloride
    Agonist
    Amodiaquine-d10 hydrochloride is deuterated labeled Amodiaquine (HY-B1322A). Amodiaquine (Amodiaquin), a 4-aminoquinoline class of antimalarial agent, is a potent and orally active histamine N-methyltransferase inhibitor. Amodiaquine is also a Nurr1 agonist and specifically binds to Nurr1-LBD (ligand binding domain) with an EC50 of ~20 μM. Anti-inflammatory effect.
    Amodiaquine-d<sub>10</sub> hydrochloride