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  2. Kinase Inhibitor Library

Kinase Inhibitor Library

(653 bioactive Compounds) Cat. No.: HY-L009
Library Contents: XLSX PDF

A unique collection of 653 kinase inhibitors/regulators for high throughput screening (HTS) and high content screening (HCS).

Size (Pre-dissolved DMSO or Solid) Price Stock
30 μL/well (10 mM solution) Get quote In-stock
50 μL/well (10 mM solution) Get quote In-stock
100 μL/well (10 mM solution) Get quote In-stock
250 μL/well (10 mM solution) Get quote In-stock
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  • Description

  • Product Details

  • Contents

  • Documentation

Description
& Advantages

•   A unique collection of 588 kinase inhibitors/regulators for high throughput screening (HTS) and high content screening (HCS).

•   Targets kinases such as RTKs, PI3K, Aurora Kinase, CDK, PKC, VEGFR, ROCK and Raf etc.

•   Bioactivity and safety confirmed by preclinical research and clinical trials.

•   Some inhibitors have been approved by the FDA.

•   Most are ATP competitive.

•   Structurally diverse, medicinally active, and cell permeable.

•   Rich documentation with structure, IC50, and customer reviews.

•   NMR and HPLC validated to ensure high purity.

Product Details
Formulation:
A collection of 653 kinase regulators supplied as pre-dissolved DMSO solutions
Container:
96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
Storage:
-80°C
Shipping:
Blue ice
Composition

Kinase Inhibitor Library

Source: MedChem Express

Contents of Kinase Inhibitor Library

Plate layout: HY-L009-1

1 2 3 4 5 6 7 8 9 10 11 12
a Empty 3-Methyladenine 5-Aminosalicylic acid Metformin (hydrochloride) Poloxime AG 18 Scopoletin MNS Trapidil CID755673 SP600125 Empty
b Empty RIPA-56 TDZD-8 SC-514 Resveratrol SU5416 Danthron SU9516 Phenformin (hydrochloride) CGP 57380 Piceatannol Empty
c Empty IQ-1S (free acid) NU2058 TG003 PHA-767491 (hydrochloride) kb NB 142-70 TPI-1 BMS-345541 (free base) Bakuchiol AS-605240 AICAR Empty
d Empty Necrostatin-1 SMI-16a Anisomycin Honokiol PD98059 Formononetin Apigenin Emodin Genistein SAR245409 Empty
e Empty Butein Bikinin TCS-PIM-1-4a RG14620 GW 441756 TC-DAPK 6 SC66 Indirubin-3'-monoxime TPCA-1 NU 7026 Empty
f Empty Compound 401 PP1 BX517 Tyrphostin A9 Y15 Wogonin Dihydroartemisinin Scutellarein Zoledronic acid (monohydrate) BMS-345541 Empty
g Empty CHR-6494 IRAK inhibitor 1 AG-490 [6]-Gingerol SU 5402 Poloxin SKF-86002 ID-8 Amlexanox Nocodazole Empty
h Empty PP2 Quercetin SKI II MCB-613 AG1024 AS-252424 NSC23005 (sodium) IRAK inhibitor 2 LY294002 Hydroxyfasudil Empty

Plate layout: HY-L009-2

1 2 3 4 5 6 7 8 9 10 11 12
a Empty AR-A014418 LY3177833 INK-128 TSU-68 IC261 Thiazovivin AT13148 STO-609 AG-1478 Isorhamnetin Empty
b Empty Tyrphostin AG 879 LH846 1-Naphthyl PP1 TWS119 PP121 Vps34-PIK-III Y-27632 (dihydrochloride) Triciribine SKLB1002 PS-1145 Empty
c Empty Bupivacaine (hydrochloride) XL413 (hydrochloride) RKI-1447 Kenpaullone FR 180204 Fasudil (Hydrochloride) PD158780 TTP 22 SB 202190 1-NM-PP1 Empty
d Empty KW-2449 TCS JNK 5a Oglufanide GSK1059615 ZM 306416 GDC-0879 Tideglusib SL327 DPH CC-115 Empty
e Empty AT7867 LM22A-4 Pim1/AKK1-IN-1 NVP-BVU972 PRT-060318 MSC2530818 PQ401 CCT128930 Fingolimod (hydrochloride) ETC-1002 Empty
f Empty BMS-265246 SSR128129E TG100-115 NG 52 L-779450 Ingenol CP-466722 SRPIN340 CX-4945 IPA-3 Empty
g Empty TA-01 Ro-3306 1-Naphthyl PP1 (hydrochloride) VS-5584 Roscovitine ISCK03 Coptisine (chloride) CGP60474 BIO AICAR (phosphate) Empty
h Empty CH5183284 R1530 TAS-301 SAR131675 SGX-523 SB 415286 LFM-A13 PD153035 PD 169316 A-769662 Empty

Plate layout: HY-L009-3

1 2 3 4 5 6 7 8 9 10 11 12
a Empty TCS 359 PF06650833 PHA-793887 ZLN024 (hydrochloride) AZD-7762 MLN1117 BML-277 CDK-IN-2 EMD638683 CZC24832 Empty
b Empty TGX-221 SC79 GSK180736A GW2580 MLN120B TCS PIM-1 1 APTO-253 Sanguinarine (chloride) LJI308 SB 239063 Empty
c Empty VE-821 PD168393 Tivantinib Brivanib MSDC 0160 LDC000067 SB 216763 AIM-100 SU6656 AZD-5438 Empty
d Empty CX-4945 (sodium salt) PF-04217903 Tetrahydrocurcumin SB1317 TEPP-46 CC-115 (hydrochloride) Src Inhibitor 1 Motesanib GNF-2 Linifanib Empty
e Empty WHI-P154 JNJ-38877605 IM-12 CH5132799 SB 203580 Ro 28-1675 CCT245737 BI-78D3 AZD1208 PF-4989216 Empty
f Empty ZINC00881524 SNS-032 CL-387785 LJH685 AT9283 PLX647 GSK 650394 EAI045 Losmapimod IMD-0354 Empty
g Empty Chelerythrine Chloride WP1130 PI-103 (Hydrochloride) K145 (hydrochloride) AMG319 Acumapimod TIC10 isomer TIC10 APS-2-79 BIBX 1382 Empty
h Empty CPDA Purvalanol A T56-LIMKi ZM 336372 PIK-93 PF-4708671 BI-D1870 5-Iodotubercidin Latrepirdine (dihydrochloride) Dovitinib Empty

Plate layout: HY-L009-4

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Fruquintinib Erlotinib Reversine A66 IRAK-1-4 Inhibitor I KU-55933 PD-166866 Toceranib IRAK inhibitor 6 Dinaciclib Empty
b Empty CID 2011756 IC-87114 D4476 GSK583 Sunitinib BLZ945 HLM006474 TAK-715 CVT-313 ACHP (Hydrochloride ) Empty
c Empty Acalisib Flavopiridol Dehydrocorydaline (chloride) VX-702 SGI-1776 PF-06463922 LY3023414 ANA-12 SR-3677 AZD 6482 Empty
d Empty PHT-427 Telatinib PF-670462 NVP-BKM120 AT7867 (dihydrochloride) PQR309 GS-9973 ZM323881 (hydrochloride) NT157 INCB28060 Empty
e Empty BIX02188 AZ20 AZD6738 KU-57788 PLX-4720 SB 203580 (hydrochloride) AXL1717 LTURM34 GNE-317 GSK2256098 Empty
f Empty SKLB610 CAL-101 Tomatidine GSK2656157 KRN-633 Duvelisib Duvelisib (R enantiomer) ZSTK474 CP-673451 Pexidartinib Empty
g Empty GNF-5 TP-3654 AT7519 (Hydrochloride) Vatalanib CHIR-124 Linsitinib URMC-099 HS-173 AVL-292 AM-2394 Empty
h Empty NVP-BAW2881 HMN-214 LY3009120 CC-401 (hydrochloride) PF-04691502 GSK-690693 Vps34-IN-1 U0126 Lenvatinib Afuresertib Empty

Plate layout: HY-L009-5

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Icotinib (Hydrochloride) LOXO-101 AZD5363 GSK2141795 BMS-3 ON123300 AZ191 Erlotinib (Hydrochloride) PRT062607 (Hydrochloride) AS703026 Empty
b Empty BMS-5 MK-8745 GSK429286A LDC4297 Purvalanol B VRT752271 GSK2636771 CUDC-101 LEE011 TBB Empty
c Empty VX-745 LY2603618 Pazopanib XL228 Flavopiridol (Hydrochloride) Sotrastaurin S49076 PCI-32765 BIX02189 AEE788 Empty
d Empty MEK162 Brivanib (alaninate) BYL-719 SU14813 Go 6983 AZM475271 OSI-930 Crenolanib LY2874455 Cerdulatinib Empty
e Empty PF-04979064 Erdafitinib NVP-BKM120 (Hydrochloride) Gefitinib AZD2932 Amuvatinib Quercitrin PI3K inhibitor X AZD-3463 Crizotinib Empty
f Empty Cediranib ISRIB (trans-isomer) GSK2606414 AZ 628 SUN11602 SLx-2119 AZD2858 SB-590885 ONO-4059 Tivozanib Empty
g Empty SGI-7079 GDC-0623 BRAF inhibitor ONO-4059 (analog) AZD8186 AS 602801 Selumetinib GDC-0068 AZD3759 NVP-LCQ195 Empty
h Empty GDC-0032 PHA-848125 AZD8330 Necrosulfonamide BMS-754807 AZD0156 Perifosine MK-5108 CX-6258 GSK2334470 Empty

Plate layout: HY-L009-6

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Sal003 BAY 61-3606 (dihydrochloride) AMG-337 VE-822 AZD4547 UNC2881 Afuresertib (hydrochloride) BI-847325 Tozasertib MRT67307 Empty
b Empty Sorafenib CHIR-99021 Acalabrutinib JI-101 YM-201636 Pelitinib Mubritinib PF-04217903 (methanesulfonate) HTH-01-015 BMS-794833 Empty
c Empty NVP-TAE 226 Ki8751 CP-724714 AZD-8835 Dacomitinib LY2784544 R406 (free base) ETP-46464 MRT68921 (hydrochloride) BX-912 Empty
d Empty Ro 5126766 Dorsomorphin (dihydrochloride) Rigosertib (sodium) Sapitinib Pazopanib (Hydrochloride) PF-03814735 XMD8-92 Danusertib Vandetanib UNC2025 Empty
e Empty DMAT GW843682X CI-1040 AZD7545 B-Raf inhibitor 1 CCT241533 (hydrochloride) SBE13 (Hydrochloride) Salubrinal NVS-PAK1-1 BMS-536924 Empty
f Empty MK 2206 (dihydrochloride) Irbinitinib PD0325901 Dovitinib (lactate) CH5424802 Regorafenib IKK 16 Palbociclib (hydrochloride) LY2409881 AZ-5104 Empty
g Empty Afatinib CHIR-98014 Olmutinib Crizotinib (hydrochloride) Dasatinib Bucladesine (calcium salt) PIK-75 DCC-2618 PIK-294 Vemurafenib Empty
h Empty PF-3758309 Poziotinib Bucladesine (sodium salt) PF-573228 EMD-1214063 Apatinib Imatinib Toceranib (phosphate) WZ4002 AT7519 (trifluoroacetate) Empty

Plate layout: HY-L009-7

1 2 3 4 5 6 7 8 9 10 11 12
a Empty WZ4003 CCT129202 GDC-0980 Masitinib CNX-774 CDK9-IN-1 AZD-9291 VX-11e MK-1775 Regorafenib (monohydrate) Empty
b Empty PND-1186 Cabozantinib PHA-680632 NVP-BHG712 AMG 900 TAK-733 TAK-901 GSK2126458 MLN 2480 PI-3065 Empty
c Empty AZD1152-HQPA JNK-IN-8 GSK-1070916 BLU9931 TG101209 Defactinib LY2090314 BMS 777607 SCIO-469 UNC2025 (hydrochloride) Empty
d Empty FRAX486 CCT196969 ZM-447439 GDC-0941 Enzastaurin TP-0903 PDK1 inhibitor Hesperadin CEP-32496 MGCD-265 analog Empty
e Empty ALK inhibitor 2 RAF265 Alisertib CH5424802 (Hydrochloride) Regorafenib (Hydrochloride) H-89 (dihydrochloride) Dabrafenib GW 5074 BI 2536 Tauroursodeoxycholate (Sodium) Empty
f Empty PD173074 Dasatinib (hydrochloride) ENMD-2076 (Tartrate) SNS-314 KX2-391 (Mesylate) Doramapimod IPI549 ALK-IN-1 Nilotinib AST 487 Empty
g Empty Lck Inhibitor GDC-0068 (dihydrochloride) Cobimetinib NMS-1286937 GZD824 Ponatinib GSK1838705A CFI-400945 (free base) GNF-5837 BIBF 1120 Empty
h Empty XL-147 Saracatinib GSK461364 CNX-2006 GNF-7 KU-60019 TAK-285 Pluripotin CCT 137690 AKT inhibitor VIII Empty

Plate layout: HY-L009-8

1 2 3 4 5 6 7 8 9 10 11 12
a Empty LY2801653 DDR1-IN-1 LEE011 (succinate) DCC-2036 Ro 31-8220 (mesylate) TAK-632 CO-1686 CGK733 Neratinib LDK378 Empty
b Empty SU14813 (maleate) Canertinib (dihydrochloride) NVP-BGJ398 LDC1267 Entrectinib Quizartinib PD318088 TAK-960 Flumatinib Tandutinib Empty
c Empty THZ1 Cediranib (maleate) BMS-599626 (Hydrochloride) SU11274 WH-4-023 Motesanib (Diphosphate) GSK269962A LEE011 (succinate hydrate) TGR-1202 Refametinib Empty
d Empty Palbociclib (isethionate) CHIR-99021 (trihydrochloride) Bafetinib Belizatinib CGI-1746 CEP-37440 ASP3026 Lapatinib Nilotinib (monohydrochloride monohydrate) Brigatinib Empty
e Empty AZD1152 Aurora A inhibitor I Imatinib (Mesylate) BX795 A 419259 (trihydrochloride) Masitinib (mesylate) AZD-9291 (mesylate) PI3K-IN-1 THZ1 (Hydrochloride) LY2835219 Empty
f Empty Avitinib (maleate) KRCA-0008 EG00229 Neohesperidin dihydrochalcone LY2228820 NVP-TAE 684 Trametinib Dabrafenib (Mesylate) LY-2584702 (tosylate salt) Volasertib Empty
g Empty Ginsenoside Rh2 R788(prodrug of R406) Verbascoside R406 Sitravatinib LDK378 (dihydrochloride) Centrinone-B Foretinib Centrinone E-7050 Empty
h Empty FIIN-2 CEP-28122 (mesylate salt) Cabozantinib (S-malate) CO-1686 (hydrobromide) Sorafenib (Tosylate) XMD17-109 PHA-665752 BEZ235 (Tosylate) BIBF 1120 (esylate) NVP-BGT226 Empty

Plate layout: HY-L009-9

1 2 3 4 5 6 7 8 9 10 11 12
a Empty CFI-400945 (fumarate) Flumatinib (mesylate) PF-562271 (besylate) Icariin Trametinib (DMSO solvate) c-Met inhibitor 2 GDC-0941 (dimethanesulfonate) Afatinib (dimaleate) KN-62 R788 (disodium hexahydrate) Empty
b Empty Astragaloside IV GSK1904529A Lapatinib (ditosylate) Empty Empty Empty Empty Empty Empty Empty Empty
c Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
d Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
e Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
f Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
g Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
h Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
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