1. Screening Libraries
  2. Protein Tyrosine Kinase Compound Library

Protein Tyrosine Kinase Compound Library

(271 bioactive Compounds) Cat. No.: HY-L016
Library Contents: XLSX PDF

A unique collection of 271 tyrosine kinase inhibitors for high throughput screening (HTS) and high content screening (HCS).

Size (Pre-dissolved DMSO or Solid) Price Stock
30 μL/well (10 mM solution) Get quote In-stock
50 μL/well (10 mM solution) Get quote In-stock
100 μL/well (10 mM solution) Get quote In-stock
250 μL/well (10 mM solution) Get quote In-stock
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  • Description

  • Product Details

  • Composition

  • Contents

  • Documentation

Description
& Advantages

•   A unique collection of 271 tyrosine kinase inhibitors for high throughput screening (HTS) and high content screening (HCS).

•   Bioactivity and safety confirmed by preclinical research and clinical trials.

•   Some tyrosine kinase inhibitors have been approved by FDA.

•   Targets such as Ack1, ALK, Btk, c-Fms, c-Met/HGFR, EGFR, FGFR, Insulin Receptor, JAK,PDGFR etc.

•   Structurally diverse, medicinally active and cell permeable.

•   Rich documentation with structure, IC50 and summary.

•   NMR and HPLC to ensure the high purity.

Product Details
Formulation:
A collection of 271 tyrosine kinase inhibitors supplied as pre-dissolved DMSO solutions
Container:
96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
Storage:
-80°C
Shipping:
Blue ice
Composition

Protein Tyrosine Kinase Compound Library

Source: MedChem Express

Contents of Protein Tyrosine Kinase Compound Library

Plate layout: HY-L016-1

1 2 3 4 5 6 7 8 9 10 11 12
a Empty AG 18 MNS Trapidil SU5416 Piceatannol TPI-1 Formononetin Genistein Butein RG14620 Empty
b Empty GW 441756 PP1 Tyrphostin A9 Y15 Scutellarein IRAK inhibitor 1 AG-490 SU 5402 ID-8 Nocodazole Empty
c Empty PP2 MCB-613 AG1024 IRAK inhibitor 2 TSU-68 AG-1478 Tyrphostin AG 879 1-Naphthyl PP1 PP121 SKLB1002 Empty
d Empty PD158780 KW-2449 Oglufanide ZM 306416 DPH LM22A-4 NVP-BVU972 PRT-060318 PQ401 SSR128129E Empty
e Empty 1-Naphthyl PP1 (hydrochloride) ISCK03 CH5183284 R1530 SAR131675 SGX-523 LFM-A13 PD153035 TCS 359 PF06650833 Empty
f Empty GW2580 PD168393 Tivantinib Brivanib MSDC 0160 AIM-100 SU6656 PF-04217903 SB1317 Src Inhibitor 1 Empty
g Empty Motesanib GNF-2 Linifanib ENMD-2076 WHI-P154 JNJ-38877605 TAK-659 (hydrochloride) CL-387785 PLX647 EAI045 Empty
h Empty WP1130 BIBX 1382 CPDA Dovitinib Fruquintinib Erlotinib IRAK-1-4 Inhibitor I PD-166866 Toceranib IRAK inhibitor 6 Empty

Plate layout: HY-L016-2

1 2 3 4 5 6 7 8 9 10 11 12
a Empty BLZ945 PF-06463922 ANA-12 Telatinib GS-9973 ZM323881 (hydrochloride) NT157 INCB28060 AXL1717 GSK2256098 Empty
b Empty SKLB610 KRN-633 CP-673451 Pexidartinib GNF-5 Vatalanib CHIR-124 Linsitinib AVL-292 NVP-BAW2881 Empty
c Empty Lenvatinib Afuresertib Icotinib (Hydrochloride) LOXO-101 AZD5363 AZ191 Erlotinib (Hydrochloride) PRT062607 (Hydrochloride) CUDC-101 Pazopanib Empty
d Empty XL228 S49076 PCI-32765 AEE788 Brivanib (alaninate) SU14813 AZM475271 OSI-930 Crenolanib LY2874455 Empty
e Empty Cerdulatinib Erdafitinib Gefitinib AZD2932 Amuvatinib AZD-3463 Crizotinib Cediranib SUN11602 ONO-4059 Empty
f Empty Tivozanib SGI-7079 ONO-4059 (analog) AZD3759 BMS-754807 BAY 61-3606 (dihydrochloride) AMG-337 AZD4547 UNC2881 Afuresertib (hydrochloride) Empty
g Empty Sorafenib Acalabrutinib JI-101 Pelitinib Mubritinib PF-04217903 (methanesulfonate) BMS-794833 NVP-TAE 226 Ki8751 CP-724714 Empty
h Empty Dacomitinib LY2784544 R406 (free base) Sapitinib Pazopanib (Hydrochloride) Vandetanib UNC2025 NVS-PAK1-1 BMS-536924 Irbinitinib Empty

Plate layout: HY-L016-3

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Dovitinib (lactate) CH5424802 Regorafenib AZ-5104 Afatinib Olmutinib Crizotinib (hydrochloride) Dasatinib Bucladesine (calcium salt) DCC-2618 Empty
b Empty Poziotinib Bucladesine (sodium salt) PF-573228 EMD-1214063 Apatinib Imatinib Toceranib (phosphate) WZ4002 Masitinib CNX-774 Empty
c Empty AZD-9291 Regorafenib (monohydrate) PND-1186 Cabozantinib NVP-BHG712 PF-562271 BLU9931 TG101209 Defactinib BMS 777607 Empty
d Empty UNC2025 (hydrochloride) TP-0903 MGCD-265 analog ALK inhibitor 2 RAF265 CH5424802 (Hydrochloride) Regorafenib (Hydrochloride) H-89 (dihydrochloride) PD173074 Dasatinib (hydrochloride) Empty
e Empty ENMD-2076 (Tartrate) LOXO-101 (sulfate) KX2-391 (Mesylate) ALK-IN-1 Nilotinib AST 487 Lck Inhibitor Ponatinib GZD824 GSK1838705A Empty
f Empty GNF-5837 BIBF 1120 Saracatinib CNX-2006 GNF-7 TAK-285 LY2801653 DDR1-IN-1 DCC-2036 CO-1686 Empty
g Empty Neratinib LDK378 SU14813 (maleate) Canertinib (dihydrochloride) NVP-BGJ398 LDC1267 Entrectinib Quizartinib Flumatinib Tandutinib Empty
h Empty Cediranib (maleate) BMS-599626 (Hydrochloride) SU11274 WH-4-023 Motesanib (Diphosphate) Bafetinib CGI-1746 CEP-37440 ASP3026 Lapatinib Empty

Plate layout: HY-L016-4

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Nilotinib (monohydrochloride monohydrate) Brigatinib Imatinib (Mesylate) A 419259 (trihydrochloride) Masitinib (mesylate) AZD-9291 (mesylate) Avitinib (maleate) KRCA-0008 EG00229 Neohesperidin dihydrochalcone Empty
b Empty NVP-TAE 684 Ginsenoside Rh2 R406 Sitravatinib LDK378 (dihydrochloride) Foretinib FIIN-2 CEP-28122 (mesylate salt) Cabozantinib (S-malate) CO-1686 (hydrobromide) Empty
c Empty Sorafenib (Tosylate) PHA-665752 BIBF 1120 (esylate) Flumatinib (mesylate) GDC-0853 PF-562271 (besylate) c-Met inhibitor 2 Afatinib (dimaleate) R788 (disodium hexahydrate) GSK1904529A Empty
d Empty Lapatinib (ditosylate) Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
e Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
f Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
g Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
h Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
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