2. GPCR/G Protein Neuronal Signaling
  3. Opioid Receptor
  4. UFP-101

UFP-101 is a potent, selective, and competitive antagonist of the NOP receptor, with a pKi of 10.24. UFP-101 displays >3000-fold selectivity over δ, μ and κ opioid receptors. UFP-101 shows antidepressant-like effect.

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UFP-101 Chemical Structure

UFP-101 Chemical Structure

CAS No. : 849024-68-6

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Description

UFP-101 is a potent, selective, and competitive antagonist of the NOP receptor, with a pKi of 10.24. UFP-101 displays >3000-fold selectivity over δ, μ and κ opioid receptors. UFP-101 shows antidepressant-like effect[1][2].

IC50 & Target

NOP Receptor/ORL1

 

In Vivo

UFP-101 elicits a pronounced acute and dosedependent antidepressant-like effect in mice submitted to the forced swimming test (FST)[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Molecular Weight

1908.17

Formula

C82H138N32O21
CAS No.
Sequence Shortening

{Bn}-GGGFTGARKSARKRKNQ-NH2
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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UFP-101 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

UFP-101849024-68-6UFP101UFP 101Opioid Receptorselectivecompetitiveantidepressantforcedswimmingtestligand,Inhibitorinhibitorinhibit

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