1. Signaling Pathways
  2. Metabolic Enzyme/Protease
  3. Isocitrate Dehydrogenase (IDH)
  4. Isocitrate Dehydrogenase (IDH) Inhibitors

Isocitrate Dehydrogenase (IDH) Inhibitors

IDH1

IDH2

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Isocitrate Dehydrogenase (IDH) Inhibitors
Product Name IDH1 IDH2 Purity
Enasidenib  
IDH2
99.97%
Vorasidenib
IDH1
IDH2
99.87%
GSK864
IDH1
  99.93%
AGI-5198
IDH1
  99.77%
BAY-1436032
IDH1
  99.48%
Enasidenib mesylate  
IDH2
99.85%
Olutasidenib
IDH1
  99.30%
Mutant IDH1-IN-1
IDH1
  99.53%
(S,R)-GSK321
IDH1
  98.78%
IDH1 Inhibitor 2
IDH1
  99.40%
(R,R)-GSK321
IDH1
  99.31%
Mutant IDH1-IN-2
IDH1
  98.50%
LY3410738
IDH1
IDH2
IDH1 Inhibitor 7
IDH1, IC50: <100 nM
  99.46%
Safusidenib
IDH1
 
TC-E 5008
R132H IDH1, Ki: 190 nM
R132C IDH1, Ki: 120 nM
WT IDH1, Ki: 12.3 μM
 
IHMT-IDH1-053
R132H IDH1, IC50: 4.7 μM