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DUBs-IN-3

HY-50737

DUBs-IN-3

DUBs-IN-3 Chemical Structure

DUBs-IN-3 is a potent deubiquitinase enzyme inhibitor with IC50s of 3.1 uM for USP8; >30 fold selectivity over USP7 (IC50 > 100 uM).

Size Price Stock Quantity
10 mM * 1 mL in DMSO $385 In-stock
5 mg $350 In-stock
10 mg $500 In-stock
50 mg $1500 In-stock
100 mg $2100 In-stock
200 mg Get quote
500 mg Get quote
Size Price Stock Quantity
10 mM * 1 mL in DMSO €377 In-stock
5 mg €343 In-stock
10 mg €490 In-stock
50 mg €1470 In-stock
100 mg €2058 In-stock
200 mg Get quote
500 mg Get quote

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Product name: DUBs-IN-3
Cat. No.: HY-50737

DUBs-IN-3 Data Sheet

  • View current batch:

    Purity: 99.20%

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    DataSheet

    Pdf Version Network Version

    MSDS

    Pdf Version

    COA

Related Compound Libraries

Biological Activity of DUBs-IN-3

DUBs-IN-3 is a potent deubiquitinase enzyme inhibitor with IC50s of 3.1 uM for USP8; >30 fold selectivity over USP7 (IC50 > 100 uM).
IC50 value: 3.1 uM(USP8) [1]
Target: USP8

Chemical Information

M.Wt 287.28 Storage Please store the product under the recommended conditions in the Certificate of Analysis.
Formula C16H9N5O
CAS No 924296-17-3
Solvent & Solubility

DMSO: ≥ 20 mg/mL

Preparing Stock Solutions

1 mg 5 mg 10 mg
1 mM 3.4809 mL 17.4046 mL 34.8092 mL
5 mM 0.6962 mL 3.4809 mL 6.9618 mL
10 mM 0.3481 mL 1.7405 mL 3.4809 mL

References on DUBs-IN-3

Other Forms

Inhibitor Kit

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