1. Metabolic Enzyme/Protease
    Anti-infection
  2. HCV
    HCV Protease

Vaniprevir (Synonyms: MK-7009; MK7009; MK 7009)

Cat. No.: HY-10243
Handling Instructions

Vaniprevir (MK-7009) is a non-covalent competitive inhibitor of the hepatitis C virus (HCV) NS3/4A protease.

For research use only. We do not sell to patients.
Vaniprevir Chemical Structure

Vaniprevir Chemical Structure

CAS No. : 923590-37-8

Size Price Stock Quantity
10 mM * 1 mL in DMSO $417 In-stock
5 mg $350 In-stock
10 mg $500 In-stock
50 mg   Get quote  
100 mg   Get quote  

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Description

Vaniprevir (MK-7009) is a non-covalent competitive inhibitor of the hepatitis C virus (HCV) NS3/4A protease. IC50 Value: Target: HCV NS3/4A Protease; HCV vaniprevir (MK-7009) is a macrocyclic hepatitis C virus NS3/4a protease inhibitor, is active against both the genotype 1 and genotype 2 NS3/4a protease enzymes. vaniprevir (MK-7009) has good plasma exposure and excellent liver exposure in multiple species.

Clinical Trial
Sponsor Condition Start Date Phase
Merck & Co Inc Hepatitis C virus infection 2011-09-30 Phase 3
Merck & Co Inc Hepatitis C virus infection 2011-08-31 Phase 3
Merck & Co Inc Hepatitis C virus infection 2011-06-30 Phase 3
Merck & Co Inc Hepatitis C virus infection 2009-03-31 Phase 2
Merck & Co Inc Hepatitis C virus infection 2010-06-30 Phase 2
Preparing Stock Solutions
Concentration Volume (DMSO) Mass 1 mg 5 mg 10 mg
1 mM 1.3194 mL 6.5968 mL 13.1937 mL
5 mM 0.2639 mL 1.3194 mL 2.6387 mL
10 mM 0.1319 mL 0.6597 mL 1.3194 mL
M.Wt

757.94

Formula

C₃₈H₅₅N₅O₉S

CAS No.

923590-37-8

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Shipping

Room temperature in continental US; may vary elsewhere

Solvent & Solubility

10 mM in DMSO

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Product Name:
Vaniprevir
Cat. No.:
HY-10243
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