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Products are for research use only. Not for human use. We do not sell to patients.

Signaling Pathway

Zaurategrast

HY-70073

(CDP-323; CDP 323; CDP323)

Zaurategrast

Zaurategrast Chemical Structure

Zaurategrast(CDP-323) is an oral α4-integrin inhibitor.

Size Price Stock Quantity
Free sample   Apply now  
10 mM * 1 mL in DMSO $195 In-stock
5 mg $170 In-stock
10 mg $300 In-stock
25 mg $590 In-stock
50 mg Get quote
100 mg Get quote
Size Price Stock Quantity
Free sample   Apply now  
10 mM * 1 mL in DMSO €191 In-stock
5 mg €167 In-stock
10 mg €294 In-stock
25 mg €578 In-stock
50 mg Get quote
100 mg Get quote

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Inquiry Information
Product name: Zaurategrast
Cat. No.: HY-70073

Zaurategrast Data Sheet

  • View current batch:

    Purity: 99.53%

  • Pdf Version Network Version

    DataSheet

    Pdf Version Network Version

    MSDS

    Pdf Version

    COA

Related Compound Libraries

Biological Activity of Zaurategrast

Zaurategrast(CDP-323) is an oral α4-integrin inhibitor.
IC50 value:
Target: α4-integrin
CDP323 significantly decreased the capacity of lymphocytes to bind vascular adhesion molecule-1 (VCAM-1) and the expression of α4-integrin on VCAM-1-binding cells.CDP323 at daily doses of 1000 or 2000 mg induced significant increases in total lymphocyte count and suppressed VCAM-1 binding by reducing unbound very late antigen-4 expression on lymphocytes.

Protocol (Extracted from published papers and Only for reference)

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Chemical Information

M.Wt 521.41 Storage Please store the product under the recommended conditions in the Certificate of Analysis.
Formula C26H25BrN4O3
CAS No 455264-31-0
Solvent & Solubility

10 mM in DMSO

Preparing Stock Solutions

1 mg 5 mg 10 mg
1 mM 1.9179 mL 9.5894 mL 19.1788 mL
5 mM 0.3836 mL 1.9179 mL 3.8358 mL
10 mM 0.1918 mL 0.9589 mL 1.9179 mL

References on Zaurategrast

Inhibitor Kit

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