1. GPCR/G Protein
  2. Protease-Activated Receptor (PAR)

Vorapaxar (Synonyms: SCH 530348)

Cat. No.: HY-10119 Purity: 99.90%
Handling Instructions

Vorapaxar is a thrombin receptor (protease-activated receptor, PAR-1) antagonist.

For research use only. We do not sell to patients.
Vorapaxar Chemical Structure

Vorapaxar Chemical Structure

CAS No. : 618385-01-6

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 185 In-stock
5 mg USD 168 In-stock
10 mg USD 288 In-stock
25 mg USD 600 In-stock
50 mg USD 900 In-stock
100 mg   Get quote  
200 mg   Get quote  

* Please select Quantity before adding items.

Customer Review

  • Biological Activity

  • Protocol

  • Technical Information

  • Purity & Documentation

  • References

Description

Vorapaxar is a thrombin receptor (protease-activated receptor, PAR-1) antagonist. Target: PAR-1 Vorapaxar is an oral protease-activated receptor antagonist, is a novel antiplatelet drug that has been recently approved to provide further risk reduction. Vorapaxar has a high bioavailability after oral administration of >90% with a half-life of 126 h-296 h. It binds reversibly to a PAR-1; however, it slowly dissociates making it functionally irreversible. Vorapaxar is a potential antithrombotic drug.

Clinical Trial
References
Preparing Stock Solutions
Concentration Volume Mass 1 mg 5 mg 10 mg
1 mM 2.0301 mL 10.1506 mL 20.3013 mL
5 mM 0.4060 mL 2.0301 mL 4.0603 mL
10 mM 0.2030 mL 1.0151 mL 2.0301 mL
Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

492.58

Formula

C₂₉H₃₃FN₂O₄

CAS No.

618385-01-6

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Shipping

Room temperature in continental US; may vary elsewhere

Solvent & Solubility

DMSO: ≥ 30 mg/mL

* "<1 mg/mL" means slightly soluble or insoluble. "≥" means soluble, but saturation unknown.

Inquiry Online

Your information is safe with us. * Required Fields.

Product name

 

Salutation

Applicant name *

 

Email address *

Phone number *

 

Organization name *

Country *

 

Requested quantity *

Remarks

Bulk Inquiry

Inquiry Information

Product Name:
Vorapaxar
Cat. No.:
HY-10119
Quantity: