1. GPCR/G Protein
  2. Adenosine Receptor

ZM241385 (Synonyms: ZM-241385; ZM 241385)

Cat. No.: HY-19532 Purity: 98.55%
Data Sheet SDS Handling Instructions

ZM 241385 is a novel non-xanthine adenosine receptor antagonist with selectivity for the A2a receptor subtype.

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ZM241385 Chemical Structure

ZM241385 Chemical Structure

CAS No. : 139180-30-6

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10 mM * 1 mL in DMSO $66 In-stock
5 mg $60 In-stock
10 mg $100 In-stock
50 mg $360 In-stock
100 mg $560 In-stock
200 mg $800 In-stock
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Description

ZM 241385 is a novel non-xanthine adenosine receptor antagonist with selectivity for the A2a receptor subtype. Target: adenosine receptor in vitro: ZM 241385 has high affinity for A2a receptors. In rat phaeochromocytoma cell membranes, ZM 241385 displaces binding of tritiated 5'-N-ethylcarboxamidoadenosine (NECA) with a pIC50 of 9.52. [1] in vivo: ZM 241385 has low potency at A2b receptors and antagonized the relaxant effects of adenosine in the guinea-pig aorta. ZM 241385 has a low affinity at A1 receptors. In rat cerebral cortex membranes it displaces tritiated R-phenylisopropyladenosine (R-PIA) with a pIC50 of 5.69. [2]

References
Preparing Stock Solutions
Concentration Volume (DMSO) Mass 1 mg 5 mg 10 mg
1 mM 2.9644 mL 14.8218 mL 29.6437 mL
5 mM 0.5929 mL 2.9644 mL 5.9287 mL
10 mM 0.2964 mL 1.4822 mL 2.9644 mL
References
M.Wt

337.34

Formula

C₁₆H₁₅N₇O₂

CAS No.

139180-30-6

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
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Room temperature in continental US; may vary elsewhere

Solvent & Solubility

DMSO: ≥ 30 mg/mL

* "<1 mg/mL" means slightly soluble or insoluble. "≥" means soluble, but saturation unknown.

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Product Name:
ZM241385
Cat. No.:
HY-19532
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