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Signaling Pathway

Capadenoson

HY-14917

(BAY 68-4986)

Capadenoson

Capadenoson Chemical Structure

Capadenoson (BAY 68-4986) is a new adenosine A1 receptor agonist.

Size Price Stock Quantity
10 mM * 1 mL in DMSO $327 In-stock
5 mg $286 In-stock
10 mg $369 In-stock
50 mg $996 In-stock
100 mg $1400 In-stock
200 mg Get quote
500 mg Get quote
Size Price Stock Quantity
10 mM * 1 mL in DMSO €320 In-stock
5 mg €280 In-stock
10 mg €362 In-stock
50 mg €976 In-stock
100 mg €1372 In-stock
200 mg Get quote
500 mg Get quote

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Inquiry Information
Product name: Capadenoson
Cat. No.: HY-14917

Capadenoson Data Sheet

  • View current batch:

    Purity: 99.62%

  • Pdf Version Network Version

    DataSheet

    Pdf Version Network Version

    MSDS

    Pdf Version

    COA

Related Compound Libraries

Biological Activity of Capadenoson

Capadenoson (BAY 68-4986) is a new adenosine A1 receptor agonist.
IC50 value:
Target:  adenosine A1 receptor
Studies showed that long-term therapy with Capadenoson improves phosphorylation and total protein level of PGC-1α in LV myocardium of HF dogs. Clinical trial found that in patients with stable angina Capadenoson lowers exercise HR at comparable maximum workload, which is associated with improved total exercise time and prolongation of time to ischaemia.

Chemical Information

M.Wt 520.03 Storage Please store the product under the recommended conditions in the Certificate of Analysis.
Formula C25H18ClN5O2S2
CAS No 544417-40-5
Solvent & Solubility

10 mM in DMSO

Preparing Stock Solutions

1 mg 5 mg 10 mg
1 mM 1.9230 mL 9.6148 mL 19.2297 mL
5 mM 0.3846 mL 1.9230 mL 3.8459 mL
10 mM 0.1923 mL 0.9615 mL 1.9230 mL

Clinical Information of Capadenoson

Product Name Sponsor Only Condition Start Date End Date Phase Last Change Date
Capadenoson Bayer AG Angina 31-MAR-08 01-NOV-08 Phase 2 12-SEP-13
Bayer AG Atrial fibrillation 23-JAN-08 31-DEC-08 Phase 2 12-JUN-13

References on Capadenoson

Inhibitor Kit

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