1. Signaling Pathways
  2. GPCR/G Protein
  3. LPL Receptor
  4. LPAR1 Isoform
  5. LPAR1 Inhibitor

LPAR1 Inhibitor

LPAR1 Inhibitors (2):

Cat. No. Product Name Effect Purity
  • HY-117444
    Inhibitor 99.34%
    ONO-9780307 is a specific synthetic LPA1 (lysophosphatidic acid receptor 1) antagonist with an IC50 value of 2.7 nM.
  • HY-117959
    Inhibitor 98.97%
    TAK-615 is a negative allosteric modulator (NAM) of the LPA1 receptor for the research of pulmonary fibrosis. TAK-615 binds the LPA1 receptor with high affinity (Kd high affinity of 1.7 nM and Kd low affinity of 14.5 nM).