2. Signaling Pathways
  3. GPCR/G Protein
  4. LPL Receptor
  5. LPAR1 Isoform
  6. LPAR1 Inhibitor

LPAR1 Inhibitor

LPAR1 Inhibitors (2):

Cat. No. Product Name Effect Purity
  • HY-117444
    ONO-9780307
    		Inhibitor 99.34%
    ONO-9780307 is a specific synthetic LPA1 (lysophosphatidic acid receptor 1) antagonist with an IC50 value of 2.7 nM.
  • HY-117959
    TAK-615
    		Inhibitor 98.97%
    TAK-615 is a negative allosteric modulator (NAM) of the LPA1 receptor for the research of pulmonary fibrosis. TAK-615 binds the LPA1 receptor with high affinity (Kd high affinity of 1.7 nM and Kd low affinity of 14.5 nM).