1. Metabolic Enzyme/Protease
  2. Acyltransferase


Acyltransferase Related Products (18):

Cat. No. Product Name Effect Purity
  • HY-32219
    T863 Inhibitor 99.08%
    T-863(DGAT-1 inhibitor) is an orally active, selective and potent DGAT1 (Acyl-CoA:diacylglycerol acyltransferase 1) inhibitor that interacts with the acyl-CoA binding site of DGAT1, and inhibits triacylglycerol synthesis in cells.
  • HY-16278
    LCQ-908 Inhibitor
    LCQ-908 is a new generation of diacylglycerol acyltransferase 1 (DGAT1) inhibitor as anti-obesity and anti-diabetic agents.
  • HY-10038
    A 922500 Inhibitor 98.50%
    A 922500 is a potent, selective, and orally bioavailable DGAT-1 inhibitor exhibiting IC50 values of 9 and 22 nM against human and mouse DGAT-1, respectively.
  • HY-13215
    Avasimibe Inhibitor 99.25%
    Avasimibe is a ACAT inhibitor incluing ACAT-1 and ACAT-2 In vitro: 1) Avasimibe has beneficial on plasma lipids and direct antiatherosclerotic activity, independent of lipid effects, in various animal models of hypercholesterolemia 2) Avasimibe enhances the lipid lowering effect of atorvastatin in subjects with homozygousfamilial hypercholesterolemia.
  • HY-15497
    AZD7687 Inhibitor 98.09%
    AZD7687 is a potent and selective DGAT1 inhibitor with an IC50 value of 80 nM (hDGAT1).
  • HY-100400A
    K-604 dihydrochloride Inhibitor
    K-604 dihydrochloride is a potent and selective acyl-CoA:cholesterol acyltransferase 1 (ACAT-1) inhibitor with an IC50 of 0.45±0.06 μM.
  • HY-19183
    E-5324 Inhibitor
    E-5324 is a novel inhibitor of acyl-CoA:cholesterol acyltransferase (ACAT).
  • HY-U00430
    MGAT2-IN-2 Inhibitor
    MGAT2-IN-2 is a potent and selective acyl CoA:monoacylglycerol acyltransferase 2 (MGAT2) inhibitor with an IC50 of 3.4 nM.
  • HY-N1067
    Xanthohumol Inhibitor 99.68%
    Xanthohumol is one of the principal flavonoids isolated from hops, the inhibitor of diacylglycerol acetyltransferase (DGAT), COX-1 and COX-2, and shows anti-cancer and anti-angiogenic activities.
  • HY-13009
    PF-04620110 Inhibitor 99.37%
    PF-04620110 is an orally active, selective and potent diglyceride acyltransferase-1 (DGAT1) inhibitor with IC50 of 19 nM.
  • HY-50670
    DGAT-1 inhibitor 2 Inhibitor
    DGAT-1 inhibitor 2 is an effective inhibitor of DGAT-1;antiobesity agents.
  • HY-12425
    DGAT1-IN-1 Inhibitor
    DGAT1-IN-1 is a potent DGAT1 inhibitor with IC50 of < 10 nM(cell lysate from Hep3B cells overexpressing human DGAT1).
  • HY-101857
    MGAT2-IN-1 Inhibitor 98.63%
    MGAT2-IN-1 is an orally active inhibitor of monoacylglycerol acyltransferase (MGAT2) with IC50 of 7.8 and 2.4 nM for human and mouse MGAT2, respectively.
  • HY-101576
    RP 70676 Inhibitor
    RP 70676 is a potent inhibitor of ACAT, with IC50 of 25 and 44 nM for rat and rabbit ACAT.
  • HY-101627
    YM17E Inhibitor
    YM17E is an inhibitor of acyl CoA:cholesterol acyltransferase (ACAT), with IC50 of 44 nM in rabbit liver microsomes in vitro.
  • HY-16437
    RP-64477 Inhibitor
    RP-64477 is a potent inhibitor of the cholesterol esterifying enzyme Acyl-coenzyme A:cholesterol O-acyltransferase (ACAT).
  • HY-15197
    ABT-046 Inhibitor
    ABT-046 is a potent, selective, and orally bioavailable Diacylglycerol acyltransferase 1 (DGAT-1 ) inhibitor (IC50= 8 nM).
  • HY-101648
    ACAT-IN-1 cis isomer Inhibitor
    ACAT-IN-1 cis isomer is a potent ACAT inhibitor with an IC50 of 100 nM.