1. Signaling Pathways
  2. Metabolic Enzyme/Protease
  3. Acyltransferase
  4. Acyltransferase Inhibitors

Acyltransferase Inhibitors

ACAT1

ACAT2

MGAT2

ACAT

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Acyltransferase Inhibitors
Product Name ACAT1 ACAT2 MGAT2 ACAT Purity
K-604 dihydrochloride
ACAT-1, IC50: 0.45 μM
ACAT-2, IC50: 102.85 μM
    ≥99.0%
Avasimibe
ACAT1, IC50: 24 μM
ACAT2, IC50: 9.2 μM
    99.50%
Nevanimibe hydrochloride
ACAT1, EC50: 9 nM
ACAT2, EC50: 368 nM
    98.07%
Pactimibe sulfate
ACAT1, IC50: 4.9 μM
ACAT2, IC50: 3.0 μM
 
ACAT, IC50: 2 μM (in the liver)
ACAT, IC50: 2.7 μM (in macrophages)
ACAT, IC50: 4.7 μM (in THP-1 cells)
98.22%
Pactimibe
ACAT1, IC50: 4.9 μM
ACAT2, IC50: 3.0 μM
 
ACAT, IC50: 2 μM (in the liver)
ACAT, IC50: 2.7 μM (in macrophages)
ACAT, IC50: 4.7 μM (in THP-1 cells)
98.07%
Beauvericin      
ACAT
99.11%
Nevanimibe
ACAT1, EC50: 9 nM
ACAT2, EC50: 368 nM
   
Glabrol      
ratACAT, IC50: 24.6 μM
99.95%
Enniatin B1      
ACAT
Enniatin B      
ACAT
99.10%
Phenylpyropene C      
ACAT, IC50: 16.0 μM
VULM 1457      
ACAT
99.95%
Enniatin A      
ACAT
MGAT2-IN-2    
MGAT2, IC50: 3.4 nM