1. Screening Libraries
  2. CNS-Penetrant Compound Library

CNS-Penetrant Compound Library

Cat. No.: HY-L028
Library Contents: XLSX PDF

A unique collection of 329 bioactive CNS-penetrant compounds for high throughput screening (HTS) and high content screening (HCS).

CNS-Penetrant Compound Library
Size (Pre-dissolved DMSO or Solid) Price Stock
30 μL/well (10 mM solution) Get quote In-stock
50 μL/well (10 mM solution) Get quote In-stock
100 μL/well (10 mM solution) Get quote In-stock
250 μL/well (10 mM solution) Get quote In-stock

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Description
& Advantages

•   A unique collection of 329 bioactive CNS-penetrant compounds for high throughput screening (HTS) and high content screening (HCS).

•   Targets such as Kinases, GPCR and Ion Channels, and more.

•   A useful tool for the discovery of drugs used for brain diseases, such as brain tumors, mental disorders, and neurodegenerative diseases.

•   Bioactivity and safety confirmed by preclinical research and clinical trials. Some inhibitors have been approved by FDA.

•   Structurally diverse, medicinally active, CNS-penetrant and cell permeable.

•   More detailed compound information with structure, IC50, and brief introduction.

•   NMR and HPLC validated to ensure high purity and quality.

•   All compounds are in stock and continuously updated.

Product Details
Formulation:
A collection of 329 CNS-penetrant compounds supplied as pre-dissolved DMSO solutions or Solid
Container:
96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
Storage:
-80°C
Shipping:
Blue ice
Composition

CNS-Penetrant Compound Library

Source: MedChem Express

Contents of CNS-Penetrant Compound Library

Plate layout: HY-L028-1

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Flavopiridol Flavopiridol (Hydrochloride) SNS-032 SRI-011381 (hydrochloride) MRK-016 AEE788 Aprepitant Veliparib Olaparib Dasatinib Empty
b Empty Sorafenib Sorafenib (Tosylate) Tandutinib Cediranib Pazopanib Vorinostat Sunitinib Vandetanib (R)-Flurbiprofen Enzastaurin Empty
c Empty Vismodegib Nevirapine Delavirdine (mesylate) Efavirenz Gatifloxacin Flurbiprofen Valproic acid A-967079 NGP555 Lazertinib Empty
d Empty VER-155008 SB-590885 Pomalidomide Trametinib Rivastigmine (tartrate) Fingolimod SB 239063 3-Methyltoxoflavin LP-211 AZ32 Empty
e Empty Fingolimod (hydrochloride) Erlotinib (Hydrochloride) Pazopanib (Hydrochloride) BSI-201 Vatalanib (dihydrochloride) Vinorelbine (ditartrate) NS 1738 Nicardipine (Hydrochloride) Dantrolene (sodium hemiheptahydrate) Liproxstatin-1 Empty
f Empty Trimethobenzamide hydrochloride GNE-317 L-779450 PQR309 Laquinimod (+)-JQ-1 RJR-2403 (hemioxalate) Dacomitinib Oseltamivir (acid) Debio 0932 Empty
g Empty Chlorambucil Cisatracurium (besylate) Cladribine Cytarabine Epirubicin (hydrochloride) Ganciclovir Lomustine Procarbazine (Hydrochloride) Tamoxifen (Citrate) Tamoxifen Empty
h Empty Topotecan (Hydrochloride) Pemetrexed (disodium hemipenta hydrate) Tenofovir Escitalopram (oxalate) Vilazodone Indomethacin Methotrexate Haloperidol Clozapine Olanzapine Empty

Plate layout: HY-L028-2

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Quetiapine Aripiprazole Pimavanserin tartrate GTS-21 (dihydrochloride) Lopinavir Genistein Diethylstilbestrol Tramiprosate Clioquinol Rasagiline (mesylate) Empty
b Empty Dexamethasone Dexamethasone (acetate) Retinoic acid Aspirin Sulfasalazine Thalidomide Givinostat (hydrochloride monohydrate) Firategrast Diclofenac Diclofenac (Sodium) Empty
c Empty Lonafarnib Glibenclamide SB-269970 (hydrochloride) Vigabatrin Cabazitaxel Hoechst 34580 (tetrahydrochloride) Sodium phenylbutyrate SB-222200 Cilengitide RG2833 Empty
d Empty Irinotecan Irinotecan (hydrochloride trihydrate) AK-7 Rolipram SH-4-54 Miglustat (hydrochloride) Epothilone B Acamprosate (calcium) Dexmedetomidine (hydrochloride) Loratadine Empty
e Empty Pramipexole (dihydrochloride) Dimethyl fumarate Temozolomide Atazanavir (sulfate) Rivastigmine Rofecoxib Atorvastatin (hemicalcium salt) Metoclopramide Atomoxetine (hydrochloride) Rosiglitazone Empty
f Empty Loxapine Terbinafine Tolcapone Ziprasidone (hydrochloride monohydrate) Iloperidone Zidovudine Guanfacine (hydrochloride) Acyclovir Abacavir Abacavir (sulfate) Empty
g Empty Emtricitabine Amprenavir Mefloquine (hydrochloride) Prednisolone Metformin (hydrochloride) Atenolol Simvastatin Candesartan (Cilexetil) Itraconazole sn-Glycero-3-phosphocholine Empty
h Empty Pyrimethamine GNE-7915 (tosylate) Conivaptan (hydrochloride) L-701324 SC79 AZD3759 Roscovitine Selumetinib Palbociclib (hydrochloride) Gefitinib Empty

Plate layout: HY-L028-3

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Erlotinib Lapatinib Lapatinib (ditosylate) Imatinib (Mesylate) Rotigotine Voriconazole Etodolac Galanthamine Ibuprofen (R)-(-)-Ibuprofen Empty
b Empty Ritonavir Lenalidomide Ramelteon Paliperidone Palonosetron (Hydrochloride) Rufinamide Gabapentin Palbociclib (isethionate) Doxylamine (succinate) Perphenazine Empty
c Empty Fluphenazine (dihydrochloride) Cefotaxime (sodium salt) Trimethadione Sulindac Capecitabine D-Cycloserine Granisetron (Hydrochloride) Melatonin Bendamustine (hydrochloride) Edaravone Empty
d Empty Etomidate Etomidate (hydrochloride) Fluconazole Fluoxetine (hydrochloride) Fluvoxamine (maleate) Levetiracetam Oxcarbazepine Stavudine Sumatriptan (succinate) Topiramate Empty
e Empty Zonisamide Ofloxacin Aztreonam Ketorolac (tromethamine salt) Flucytosine Tranexamic acid Pregnenolone Salicylic acid Milnacipran (hydrochloride) Milnacipran ((1S-cis) hydrochloride) Empty
f Empty Antipyrine Sertraline (hydrochloride) Felbamate Lidocaine Lidocaine (hydrochloride) Alfuzosin Venlafaxine (hydrochloride) Naratriptan (hydrochloride) Candesartan Rizatriptan (benzoate) Empty
g Empty Pyridostigmine (bromide) Riluzole Prednisone Acetylcysteine Ketoprofen Adenosine Zolmitriptan Phenylbutazone Disulfiram Busulfan Empty
h Empty Carbamazepine Didanosine Lamivudine Piroxicam Methylprednisolone Meloxicam Methocarbamol Nimodipine Oxybutynin Pyrazinamide Empty

Plate layout: HY-L028-4

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Rifampicin Ethionamide Acetylcholine (chloride) (2S)-2-Amino-3-methyl-3-sulfanylbutanoic acid Hydroxyurea Vitamin B12 Metronidazole Sulfamethoxazole Isoniazid Levofloxacin Empty
b Empty Primidone Mirtazapine Dyclonine (hydrochloride) Memantine (hydrochloride) Cyproheptadine (hydrochloride) Orphenadrine (citrate) Almotriptan (malate) Probucol Amantadine (hydrochloride) Bupropion (hydrochloride) Empty
c Empty Clonidine (hydrochloride) Domperidone Ribavirin Vardenafil (hydrochloride) Phenytoin Phenytoin (sodium) Miconazole (nitrate) Clomipramine (hydrochloride) Amoxicillin (sodium) Amoxicillin (trihydrate) Empty
d Empty Streptomycin (sulfate) Trazodone (hydrochloride) Lamotrigine Benztropine (mesylate) Amitriptyline (hydrochloride) Trifluoperazine (dihydrochloride) Probenecid Hydroxyzine (dihydrochloride) Propranolol (hydrochloride) Cyclosporin A Empty
e Empty Tetrabenazine Ceftazidime Desvenlafaxine (succinate hydrate) Cefepime (Dihydrochloride Monohydrate) Ropinirole (hydrochloride) Dihydroergotamine (mesylate) Metaxalone Tiagabine (hydrochloride) Ceftriaxone (sodium salt) Cyclobenzaprine (hydrochloride) Empty
f Empty Acetazolamide Theophylline Protriptyline (hydrochloride) Thioridazine (hydrochloride) Amoxapine Halothane Molindone (hydrochloride) Phenelzine (sulfate) Sulpiride Fosfomycin (calcium) Empty
g Empty Buspirone (hydrochloride) L-Cycloserine Trimipramine (maleate) Prednisolone (21-acetate) Droperidol Salsalate Desipramine hydrochloride Trihexyphenidyl (hydrochloride) Piperacillin (sodium) Choline (chloride) Empty
h Empty Ethosuximide Sulfamethoxypyridazine Nefazodone (hydrochloride) 4-Aminoantipyrine Nortriptyline (hydrochloride) Chlorzoxazone Mezlocillin (sodium) Serotonin hydrochloride Imipramine (hydrochloride) Tranylcypromine (hemisulfate) Empty

Plate layout: HY-L028-5

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Fosphenytoin (disodium) Quinidine S-(+)-Ketoprofen Daidzein 5-Aminolevulinic acid (hydrochloride) Progesterone Lovastatin L-Aspartic acid Cytosporone B Empty Empty
b Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
c Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
d Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
e Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
f Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
g Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
h Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
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