1. Screening Libraries
  2. Kinase Inhibitor Library

Kinase Inhibitor Library

Cat. No.: HY-L009
Library Contents: XLSX PDF

A unique collection of 768 phosphorylation kinase inhibitors/regulators for high throughput screening (HTS) and high content screening (HCS).

Size (Pre-dissolved DMSO or Solid) Price Stock
30 μL/well (10 mM solution) Get quote In-stock
50 μL/well (10 mM solution) Get quote In-stock
100 μL/well (10 mM solution) Get quote In-stock
250 μL/well (10 mM solution) Get quote In-stock

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  • Description

  • Product Details

  • Composition

  • Contents

  • Documentation

Description
& Advantages

•   A unique collection of 768 phosphorylation kinase inhibitors/regulators for high throughput screening (HTS) and high content screening (HCS).

•   The library contains compounds targeting protein kinases (VEGFR, EGFR, BTK, CDK, Akt, etc.), lipid kinases (PI3K, PI4K, SK, etc.) and carbohydrate kinases (Hexokinase).

•   Kinase inhibitors have played an increasingly prominent role in the treatment of cancer and other diseases.

•   Bioactivity and safety confirmed by preclinical research and clinical trials. Some inhibitors have been approved by FDA.

•   Structurally diverse, medicinally active, and cell permeable.

•   Rich documentation with structure, IC50, and customer reviews.

•   NMR and HPLC validated to ensure high purity.

•   All compounds are in stock and continuously updated.

Product Details
Formulation:
A collection of 768 kinase inhibitors/regulators supplied as pre-dissolved DMSO solutions or Solid
Container:
96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
Storage:
-80°C
Shipping:
Blue ice
Composition

Kinase Inhibitor Library

Source: MedChem Express

Contents of Kinase Inhibitor Library

Plate layout: HY-L009-1

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Ginsenoside Rb1 Methylthiouracil 3-Methyladenine 5-Aminosalicylic Acid 7-Hydroxy-4-chromone 2-Deoxy-D-glucose Metformin (hydrochloride) 3-Bromopyruvic acid Poloxime AG 18 Empty
b Empty MNS 4μ8C Trapidil AG126 CID755673 trans-Zeatin SP600125 RIPA-56 TDZD-8 SC-514 Empty
c Empty Resveratrol NSC95682 SU5416 Danthron SU9516 Phenformin (hydrochloride) CGP 57380 Piceatannol SAR407899 IQ-1 Empty
d Empty NU2058 Y-27632 PHA-767491 (hydrochloride) kb NB 142-70 7-Methoxyisoflavone TPI-1 Chrysophanol BMS-345541 (free base) Bakuchiol AS-605240 Empty
e Empty AICAR Necrostatin-1 SMI-16a Anisomycin RG13022 Honokiol PD98059 Formononetin Genistein Emodin Empty
f Empty SAR245409 Butein LY-364947 Bikinin TCS-PIM-1-4a RG14620 GW 441756 TC-DAPK 6 SC66 Indirubin-3'-monoxime Empty
g Empty HA-100 TPCA-1 NU 7026 Compound 401 PP1 BX517 Tyrphostin A9 Wogonin PF-06651600 Scutellarein Empty
h Empty A 77-01 RepSox Zoledronic acid (monohydrate) BMS-345541 CHR-6494 IRAK inhibitor 1 AG-490 [6]-Gingerol SU 5402 JANEX-1 Empty

Plate layout: HY-L009-2

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Poloxin SKF-86002 ID-8 Amlexanox Hispidulin Salidroside Nocodazole PP2 Quercetin SKI II Empty
b Empty MCB-613 AG1024 AS-252424 PF-06447475 Tyrphostin AG 528 IRAK inhibitor 2 Ruxolitinib LY294002 Hydroxyfasudil AR-A014418 Empty
c Empty PP 242 LY3177833 INK-128 TSU-68 IC261 Thiazovivin Tofacitinib AT13148 STO-609 AG-1478 Empty
d Empty Isorhamnetin Tyrphostin AG 879 STF-083010 1-Naphthyl PP1 TWS119 Vps34-PIK-III PP121 Dihydromyricetin Y-27632 (dihydrochloride) Triciribine Empty
e Empty Lonidamine AG 555 PS-1145 XL413 (hydrochloride) RKI-1447 Peficitinib Kenpaullone FR 180204 Fasudil (Hydrochloride) PD158780 Empty
f Empty TTP 22 SB 202190 1-NM-PP1 APY29 KW-2449 TCS JNK 5a Oglufanide GSK1059615 ZM 306416 GDC-0879 Empty
g Empty Tideglusib SL327 SB-505124 Dicoumarol DPH CC-115 AT7867 Pim1/AKK1-IN-1 NVP-BVU972 PRT-060318 Empty
h Empty MSC2530818 PF-06409577 PQ401 SB 525334 Hydroxyfasudil (hydrochloride) ETC-1002 BMS-265246 SSR128129E TG100-115 NG 52 Empty

Plate layout: HY-L009-3

1 2 3 4 5 6 7 8 9 10 11 12
a Empty L-779450 PI-103 Ingenol AZD-1480 CP-466722 SRPIN340 CX-4945 IPA-3 TA-01 Ro-3306 Empty
b Empty K02288 ML347 BQR-695 SD-208 1-Naphthyl PP1 (hydrochloride) VS-5584 Roscovitine TPX-0005 ISCK03 CGP60474 Empty
c Empty BIO WP1066 AICAR (phosphate) CH5183284 R1530 TAS-301 SAR131675 SGX-523 SB 415286 LFM-A13 Empty
d Empty PD153035 PD 169316 A-769662 TCS 359 PF06650833 PHA-793887 ZLN024 (hydrochloride) AZD-7762 MLN1117 R-268712 Empty
e Empty BML-277 EMD638683 CZC24832 Oridonin TGX-221 SC79 GSK180736A GW2580 MLN120B TCS PIM-1 1 Empty
f Empty ZM39923 (hydrochloride) LJI308 SB 239063 VE-821 PD168393 LY2157299 Tivantinib Brivanib MSDC 0160 LDC000067 Empty
g Empty SB 216763 Baricitinib AIM-100 SU6656 AZD-5438 PF-04217903 SB1317 CC-115 (hydrochloride) Src Inhibitor 1 Motesanib Empty
h Empty GNF-2 CRT0066101 dihydrochloride Linifanib ENMD-2076 WHI-P154 GSK'481 IM-12 CH5132799 SB 203580 HG-10-102-01 Empty

Plate layout: HY-L009-4

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Ro 28-1675 CCT245737 BI-78D3 MLi-2 AZD1208 O-304 PF-4989216 DMH-1 ZINC00881524 SNS-032 Empty
b Empty BS-181 TAK-659 (hydrochloride) CL-387785 LJH685 AT9283 AT7519 PLX647 GDC-0326 GSK 650394 EAI045 Empty
c Empty AMG-208 Losmapimod GSK'872 IMD-0354 Chelerythrine Chloride WP1130 SB-431542 PI-103 (Hydrochloride) SNS-062 K145 (hydrochloride) Empty
d Empty AMG319 Acumapimod TIC10 MHY1485 APS-2-79 BIBX 1382 6,8-Bis(benzylthio)octanoic acid Purvalanol A T56-LIMKi Solcitinib Empty
e Empty ZM 336372 PIK-93 PF-4708671 BI-D1870 Icotinib 5-Iodotubercidin Dovitinib Fruquintinib Erlotinib Reversine Empty
f Empty A66 Deguelin IRAK-1-4 Inhibitor I KU-55933 PD-166866 Toceranib IRAK inhibitor 6 Dinaciclib PD153035 (Hydrochloride) CID 2011756 Empty
g Empty IC-87114 CC-223 D4476 GSK583 Sunitinib BLZ945 GSK2578215A EW-7197 TAK-715 CVT-313 Empty
h Empty ACHP (Hydrochloride) Acalisib WEHI-345 Flavopiridol Dehydrocorydaline (chloride) VX-702 Ruxolitinib (phosphate) NVP-ACC789 SGI-1776 PF-06463922 Empty

Plate layout: HY-L009-5

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Palomid 529 LDN-212854 LY3023414 ANA-12 SR-3677 AZD 6482 PHT-427 Telatinib PF-670462 NVP-BKM120 Empty
b Empty AT7867 (dihydrochloride) PQR309 GS-9973 BAY-1895344 (hydrochloride) NT157 INCB28060 BIX02188 AZ20 APY0201 KU-57788 Empty
c Empty PLX-4720 AXL1717 CYT387 LTURM34 GNE-317 Diosgenin GSK2256098 CAL-101 ITD-1 Tomatidine Empty
d Empty GSK2656157 KRN-633 Duvelisib JH-II-127 Duvelisib (R enantiomer) ZSTK474 CP-673451 Pexidartinib GNF-5 TP-3654 Empty
e Empty AT7519 (Hydrochloride) LDN-214117 Vatalanib (dihydrochloride) Protein kinase inhibitors 1 hydrochloride CHIR-124 Linsitinib URMC-099 HS-173 CHZ868 AVL-292 Empty
f Empty AM-2394 NVP-BAW2881 HMN-214 LY3009120 CC-401 (hydrochloride) PF-04691502 GSK-690693 GW788388 GLPG0634 Vps34-IN-1 Empty
g Empty U0126 Lenvatinib Afuresertib Icotinib (Hydrochloride) Wortmannin AZD5363 GSK2141795 BMS-3 AZ191 ON123300 Empty
h Empty Erlotinib (Hydrochloride) PRT062607 (Hydrochloride) AS703026 BMS-5 MK-8745 GSK429286A Isovitexin Torin 2 BMS-911543 LDC4297 Empty

Plate layout: HY-L009-6

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Purvalanol B VRT752271 GSK2636771 CUDC-101 LEE011 TBB LY3200882 VX-745 LY2603618 Pazopanib Empty
b Empty XL228 Flavopiridol (Hydrochloride) Sotrastaurin S49076 Ginkgolide C PCI-32765 BIX02189 AEE788 UNC2250 MEK162 Empty
c Empty BYL-719 SU14813 Go 6983 AZM475271 PD173955 GNE-7915 OSI-930 Crenolanib SAR405 LY2874455 Empty
d Empty Mitoxantrone A 83-01 sodium salt SAR-20347 Cerdulatinib Erdafitinib NVP-BKM120 (Hydrochloride) Gefitinib AZD2932 Amuvatinib Quercitrin Empty
e Empty PI3K inhibitor X AZD-3463 Crizotinib Cediranib ISRIB (trans-isomer) GSK2606414 AZ 628 SUN11602 SLx-2119 AZ3146 Empty
f Empty GDC-0349 Oclacitinib (maleate) AZD2858 SB-590885 ONO-4059 Tivozanib WHI-P97 SGI-7079 GDC-0623 BRAF inhibitor Empty
g Empty ONO-4059 (analog) AZD8186 AS 602801 Selumetinib GDC-0068 (-)-Epigallocatechin Gallate AZD3759 YU238259 NVP-LCQ195 GDC-0032 Empty
h Empty PHA-848125 AZD8330 Necrosulfonamide BMS-754807 AZD0156 Perifosine CX-6258 MK-5108 Scutellarin AZD2014 Empty

Plate layout: HY-L009-7

1 2 3 4 5 6 7 8 9 10 11 12
a Empty CEP-33779 GSK2334470 BAY 61-3606 (dihydrochloride) AMG-337 VE-822 AZD4547 UNC2881 Afuresertib (hydrochloride) BI-847325 Tozasertib Empty
b Empty MRT67307 Sorafenib CHIR-99021 Acalabrutinib KU-0063794 AZD-8055 JI-101 YM-201636 Pelitinib Mubritinib Empty
c Empty PF-04217903 (methanesulfonate) HTH-01-015 BMS-794833 NVP-TAE 226 Baricitinib (phosphate) Ki8751 AZD-8835 CP-724714 Dacomitinib LY2784544 Empty
d Empty R406 (free base) ETP-46464 MRT68921 (hydrochloride) BX-912 Ro 5126766 Dorsomorphin (dihydrochloride) Pacritinib Rigosertib (sodium) Sapitinib Pazopanib (Hydrochloride) Empty
e Empty PF-03814735 XMD8-92 Danusertib LX2343 Vandetanib UNC2025 DMAT MLN8054 GW843682X CI-1040 Empty
f Empty AZD7545 CCT241533 (hydrochloride) B-Raf inhibitor 1 SBE13 (Hydrochloride) NVS-PAK1-1 BMS-536924 MK 2206 (dihydrochloride) Irbinitinib Mps1-IN-2 PD0325901 Empty
g Empty Dovitinib (lactate) CH5424802 Regorafenib IKK 16 Palbociclib (hydrochloride) LY2409881 AZ-5104 Afatinib CHIR-98014 Olmutinib Empty
h Empty Crizotinib (hydrochloride) Dasatinib Bucladesine (calcium salt) CZC-25146 PIK-75 c-Kit-IN-1 PIK-294 Vemurafenib PF-3758309 Poziotinib Empty

Plate layout: HY-L009-8

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Bucladesine (sodium salt) PF-573228 EMD-1214063 Apatinib Imatinib WZ4002 WYE-354 WZ4003 GDC-0980 Masitinib Empty
b Empty CNX-774 CDK9-IN-1 AZD-9291 VX-11e MK-1775 Regorafenib (monohydrate) PND-1186 Cabozantinib PHA-680632 NVP-BHG712 Empty
c Empty AMG 900 TAK-733 KX2-391 (dihydrochloride) Tofacitinib (citrate) TAK-901 CZC-54252 GSK2126458 MLN 2480 PI-3065 PF-562271 Empty
d Empty AZD1152-HQPA JNK-IN-8 GSK-1070916 BLU9931 TG101209 Altiratinib Defactinib eCF506 LY2090314 BMS 777607 Empty
e Empty SCIO-469 UNC2025 (hydrochloride) FRAX486 CCT196969 ZM-447439 GDC-0941 Enzastaurin TP-0903 1,3-Dicaffeoylquinic acid MP7 Empty
f Empty Hesperadin Mitoxantrone (dihydrochloride) CEP-32496 MGCD-265 analog ALK inhibitor 2 RAF265 Alisertib CH5424802 (Hydrochloride) Regorafenib (Hydrochloride) H-89 (dihydrochloride) Empty
g Empty WYE-125132 GW 5074 BI 2536 Tauroursodeoxycholate (Sodium) PD173074 Dasatinib (hydrochloride) TG-101348 LOXO-101 (sulfate) SNS-314 KX2-391 (Mesylate) Empty
h Empty Doramapimod IPI549 ALK-IN-1 Nilotinib AST 487 Lck Inhibitor FLT3-IN-1 GDC-0068 (dihydrochloride) Cobimetinib NMS-1286937 Empty

Plate layout: HY-L009-9

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Ponatinib GZD824 GSK1838705A CFI-400945 (free base) GNF-5837 Mps1-IN-1 BIBF 1120 XL-147 Saracatinib PLX8394 Empty
b Empty GSK461364 CNX-2006 Defactinib (hydrochloride) GNF-7 KU-60019 TAK-285 Pluripotin CCT 137690 NPS-1034 AKT inhibitor VIII Empty
c Empty LDN193189 (Hydrochloride) LY2801653 DDR1-IN-1 LEE011 (succinate) Gilteritinib BPR1J-097 Hydrochloride DCC-2036 Ro 31-8220 (mesylate) TAK-632 CO-1686 Empty
d Empty CGK733 Ningetinib Cucurbitacin E Neratinib THZ531 LDK378 SU14813 (maleate) Canertinib (dihydrochloride) NVP-BGJ398 LDC1267 Empty
e Empty Entrectinib Quizartinib PD318088 BAY1217389 TAK-960 Flumatinib Tandutinib NVP-BSK805 (dihydrochloride) THZ1 Cediranib (maleate) Empty
f Empty BMS-599626 (Hydrochloride) SU11274 WH-4-023 Motesanib (Diphosphate) GSK269962A LEE011 (succinate hydrate) LRRK2-IN-1 TGR-1202 Refametinib Palbociclib (isethionate) Empty
g Empty CHIR-99021 (trihydrochloride) Bafetinib Belizatinib CGI-1746 CEP-37440 ASP3026 Lapatinib Nilotinib (monohydrochloride monohydrate) Brigatinib AZD1152 Empty
h Empty Aurora A inhibitor I CEP-40783 Imatinib (Mesylate) BX795 A 419259 (trihydrochloride) Masitinib (mesylate) AZD-9291 (mesylate) PI3K-IN-1 THZ1 (Hydrochloride) LY2835219 Empty

Plate layout: HY-L009-10

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Avitinib (maleate) KRCA-0008 CYT387 (sulfate salt) EG00229 Neohesperidin dihydrochalcone LY2228820 NVP-TAE 684 Trametinib GNE-7915 (tosylate) Dabrafenib (Mesylate) Empty
b Empty LY-2584702 (tosylate salt) Volasertib LYN-1604 hydrochloride R788(prodrug of R406) R406 Sitravatinib LDK378 (dihydrochloride) Centrinone-B Foretinib Centrinone Empty
c Empty X-396 hydrochloride TAK-960 (dihydrochloride) FIIN-2 CEP-28122 (mesylate salt) Cabozantinib (S-malate) CO-1686 (hydrobromide) Sorafenib (Tosylate) XMD17-109 PHA-665752 BEZ235 (Tosylate) Empty
d Empty Cobimetinib (hemifumarate) BIBF 1120 (esylate) NVP-BGT226 CFI-400945 (fumarate) Flumatinib (mesylate) GDC-0853 PF-562271 (besylate) Trametinib (DMSO solvate) SCR-1481B1 GDC-0941 (dimethanesulfonate) Empty
e Empty Afatinib (dimaleate) KN-62 Ningetinib Tosylate R788 (disodium hexahydrate) Astragaloside IV GSK1904529A Lapatinib (ditosylate) Ginsenoside Re Empty Empty Empty
f Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
g Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
h Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
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