1. Metabolic Enzyme/Protease
  2. Drug Metabolite

Drug Metabolite

Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.

Drug Metabolite Related Products (26):

Cat. No. Product Name Effect Purity
  • HY-17366
    Clozapine N-oxide 99.98%
    Clozapine N-oxide (CNO) is a major metabolite of the anti-psychotic drug clozapine. Clozapine N-oxide is a agonist for the chemogenetic Designer Receptors Exclusively Activated by Designer Drug (DREADD) system.
  • HY-13318
    Oseltamivir acid 98.60%
    GS 4104, the ethyl ester prodrug of GS 4071, is an inhibitor of influenza virus neuraminidase with an IC50 of approximately 100 nM.
  • HY-100599
    Urolithin A 98.06%
    Urolithin A is an intestinal metabolite of ellagic acid with antioxidant and antiproliferative effects; inhibits T24 and Caco-2 cell growth with IC50 values of 43.9 and 49 μM, respectively.
  • HY-101406
    Thyroxine sulfate >98.0%
    Thyroxine sulfate is a thyroid hormone metabolite.
  • HY-101107
    Allopregnanolone >98.0%
    Allopregnanolone is a progesterone metabolite. Allopregnanolone is an allosteric modulator of the GABA receptor. Used to treat postpartum depression.
  • HY-G0002A
    Lurasidone metabolite 14326 hydrochloride Chemical 98.76%
    Lurasidone metabolite 14326 (hydrochloride) is an active metabolite of the atypical antipsychotic Lurasidone.
  • HY-G0014B
    Quetiapine sulfoxide hydrochloride
    Quetiapine sulfoxide hydrochloride (Quetiapine S-oxide hydrochloride) is a main metabolite of Quetiapinem. Quetiapine is a second-generation antipsychotic.
  • HY-100645
    Trimethoprim 3-oxide >98.0%
    Trimethoprim 3-oxide (Trimethoprim 3-N-oxide) is the primary metabolite of trimethoprim.
  • HY-12772
    Hydroxy Itraconazole 99.60%
    Hydroxy Itraconazole is an active metabolite of Itraconazole (ITZ), which is a triazole antifungal agent.
  • HY-B1398
    Ampyrone 98.86%
    Ampyrone is a reagent for glucose determination in the presence of peroxidase and phenol.
  • HY-101397
    Allopurinol riboside 99.04%
    Allopurinol riboside, a metabolite of allopurinol, shows potent activities against parasites.
  • HY-G0006
    Omeprazole metabolite Omeprazole sulfide 99.91%
    Omeprazole sulfide is a metabolite of Omeprazole, which is a proton pump inhibitor.
  • HY-G0014
    Quetiapine sulfoxide
    Quetiapine sulfoxide (Quetiapine S-oxide) is a main metabolite of Quetiapinem. Quetiapine is a second-generation antipsychotic.
  • HY-G0014A
    Quetiapine sulfoxide dihydrochloride >98.0%
    Quetiapine sulfoxide dihydrochloride (Quetiapine S-oxide dihydrochloride) is a main metabolite of Quetiapinem. Quetiapine is a second-generation antipsychotic.
  • HY-101407
    Nicotinamide N-oxide 99.45%
    Nicotinamide N-oxide, an in vivo nicotinamide metabolite, is a potent, and selective antagonist of the CXCR2 receptor.
  • HY-G0011S
    Netupitant N-oxide D6
    Netupitant N-oxide D6 is the deuterium labeled Netupitant N-oxide, which is a metabolite of Netupitant.
  • HY-G0007
    Omeprazole metabolite Omeprazole sulfone
    Omeprazole sulfone is a metabolite of Omeprazole, which is a proton pump inhibitor.
  • HY-G0010S
    N-desmethyl Netupitant D6
    N-desmethyl Netupitant D6 is the deuterium labeled N-desmethyl Netupitant, which is a metabolite of Netupitant.
  • HY-15793A
    Trans (2,3)-Dihydrotetrabenazine
    Trans (2,3)-Dihydrotetrabenazine, a metabolite of Tetrabenazine, shows remarkable inhibition activity on vesicular monoamine transporter (VMAT2).
  • HY-G0001S
    Lurasidone Metabolite 14283 D8
    Lurasidone Metabolite 14283 D8 is the deuterium labeled Lurasidone Metabolite 14283, which is a metabolite of Lurasidone.
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