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Metabolism/Protease Compound Library

Cat. No.: HY-L012
Library Contents: XLSX PDF

A unique collection of 800 Metabolism/Protease-related small molecules for high throughput screening (HTS) and high content screening (HCS).

Metabolism/Protease Compound Library
Size (Pre-dissolved DMSO or Solid) Price Stock
30 μL/well (10 mM solution) Get quote In-stock
50 μL/well (10 mM solution) Get quote In-stock
100 μL/well (10 mM solution) Get quote In-stock
250 μL/well (10 mM solution) Get quote In-stock

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  • Description

  • Product Details

  • Composition

  • Contents

  • Documentation

Description
& Advantages

•   A unique collection of 800 Metabolism/Protease-related small molecules for high throughput screening (HTS) and high content screening (HCS).

•   Targets such as PDE, Cytochrome P450, HMG-CoA Reductase, DPP4, Proteasome, HCV Protease, IDO, Cathepsin, MMP, etc.

•   A useful tool for drug discovery of metabolism-related diseases.

•   Bioactivity and safety confirmed by preclinical research and clinical trials. Some inhibitors have been approved by FDA.

•   Structurally diverse, medicinally active, and cell permeable.

•   More detailed compound information with structure, IC50, and brief introduction.

•   NMR and HPLC validated to ensure high purity and quality.

•   All compounds are in stock and continuously updated.

Product Details
Formulation:
A collection of 800 Metabolism/Protease related compounds supplied as pre-dissolved DMSO solutions or Solid
Container:
96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
Storage:
-80°C
Shipping:
Blue ice
Composition

Metabolism/Protease Compound Library

Source: MedChem Express

Contents of Metabolism/Protease Compound Library

Plate layout: HY-L012-1

1 2 3 4 5 6 7 8 9 10 11 12
a Empty BAY-1436032 NSC 663284 KNK437 RSL3 (1S,3R-) AM-2394 SZL P1-41 WWL70 CL-82198 A 922500 FCCP Empty
b Empty Odanacatib TM5275 (sodium) TPI-1 Benzophenonetetracarboxylic acid PD150606 CD437 Flopropione Ribitol (-)-(S)-Equol (±)-Equol Empty
c Empty Stibogluconate (sodium) Urolithin A BVT948 SYP-5 ML348 ML349 RA190 Norverapamil (hydrochloride) IDO-IN-2 2-PMPA Empty
d Empty CHS-828 SR12813 Hypotaurine Kynurenic acid Quinolinic acid (R)-Serine KRIBB11 GCN2-IN-1 CDD3505 MK-8617 Empty
e Empty Sarcosine NQ301 TOFA AR7 Allopregnanolone UK-371804 XMD16-5 Vadadustat DMU2139 Cilostamide Empty
f Empty Deoxycytidine triphosphate Cyclo(his-pro) N-(5-Aminopentyl)acetamide Nicotinamide N-oxide Docosatrienoic Acid O-Acetylserine SDMA 4-Acetamidobutanoic acid 2-(Methylamino)-1H-purin-6(7H)-one Iberin Empty
g Empty L-DABA Vanilpyruvic acid SR9238 SR0987 SR-18292 HTS01037 BMS-986205 TRC051384 TM5441 UAMC00039 (dihydrochloride) Empty
h Empty GLPG1690 DKM 2-93 BMS-309403 Prostaglandin E2 6-Biopterin Tanespimycin BIIB021 Luminespib Bortezomib PX-478 Empty

Plate layout: HY-L012-2

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Telaprevir Boceprevir Danoprevir Mericitabine Simeprevir Betrixaban Dabigatran etexilate Dabigatran etexilate (mesylate) Linagliptin Saxagliptin Empty
b Empty Tarenflurbil ML-030 ABT-702 dihydrochloride 1-Aminobenzotriazole Stiripentol Methylmalonate Raltegravir Raltegravir (potassium salt) PKM2-IN-1 3-Methoxytyramine hydrochloride Empty
c Empty 3-Methoxytyramine CTS-1027 L-Kynurenine BAY 73-6691 racemate Ixazomib citrate Ixazomib Delanzomib Carfilzomib Daclatasvir (dihydrochloride) Daclatasvir Empty
d Empty GSK256066 AM580 Cobicistat Tipifarnib Orteronel Darapladib Ro 28-1675 T0901317 GW3965 (hydrochloride) LXR-623 Empty
e Empty 4-Butylresorcinol Tetrahydrobiopterin UVI 3003 LY2955303 Cilomilast DPP-IV-IN-2 LY2183240 GSK2033 Apararenone Cilofexor Empty
f Empty Fexaramine Pifithrin-μ VER-155008 VER-82576 BRL-50481 Arachidonic acid D4-abiraterone Crisaborole CVT-12012 Diprotin A (TFA) Empty
g Empty Pyributicarb AZD5904 1-Linoleoyl Glycerol Tinoridine hydrochloride PF-05180999 1-Ethynylnaphthalene BAY-678 GSTO1-IN-1 Mitochonic acid 5 Retagliptin Phosphate Empty
h Empty TFAP BN82002 Maltotriose Elaidic acid N-Acetylornithine 1-Methyladenosine 25-Hydroxycholesterol 5-Methylcytidine Galactose 1-phosphate Potassium salt Asymmetric dimethylarginine Empty

Plate layout: HY-L012-3

1 2 3 4 5 6 7 8 9 10 11 12
a Empty p-Synephrine trans-trans-Muconic acid (3-Carboxypropyl)trimethylammonium chloride 3-Methyladipic acid Leucyl-phenylalanine Ureidopropionic acid 4-Guanidinobutanoic acid Citraconic acid Nicotinuric acid Anserine Empty
b Empty Petroselinic acid N-Methylhydantoin DL-Dopa 3-Hydroxyisovaleric acid 3-Methylglutaric acid Nepsilon-Acetyl-L-lysine N-Acetyl-L-aspartic acid 2-D08 ABX-1431 Alvespimycin (hydrochloride) Empty
c Empty Apremilast Torcetrapib Anacetrapib Oprozomib Aliskiren Aliskiren (hemifumarate) INT-747 T-5224 TCS 401 IBMX Empty
d Empty SB-3CT C75 C75 (trans) Angiotensin (1-7) Balipodect Oltipraz Velpatasvir Lotamilast ML228 FIPI Empty
e Empty STF-118804 AEBSF JNJ-42041935 PF-05175157 PF-04620110 Telotristat etiprate Telotristat ethyl Tripterin ONX-0914 Avasimibe Empty
f Empty Talabostat (mesylate) Dolutegravir Dolutegravir (sodium) BMS-707035 Nepicastat (hydrochloride) Vinpocetine PYR-41 PYZD-4409 Oseltamivir (acid) Evacetrapib Empty
g Empty PF-8380 Varespladib SR1001 Roxadustat KW-2478 Debio 0932 U-104 Clinofibrate Cladribine Dutasteride Empty
h Empty Ezatiostat Finasteride LW6 Quinacrine (dihydrochloride) Sitagliptin Sitagliptin (phosphate monohydrate) Ursodiol 2-Deoxy-D-glucose IDO-IN-7 Ombitasvir Empty

Plate layout: HY-L012-4

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Zileuton Bexarotene Milrinone Olprinone (Hydrochloride) Febuxostat Isavuconazole Entacapone Vildagliptin PF-04457845 PF-3845 Empty
b Empty SR3335 SR1078 Onalespib Lopinavir Biochanin A (S)-Glutamic acid Retinoic acid DHEA Tamibarotene Thalidomide Empty
c Empty Fluvastatin (sodium) Choline Fenofibrate Elvitegravir Olesoxime Palifosfamide Teneligliptin Teneligliptin (hydrobromide) Topiroxostat Anagliptin Gemigliptin Empty
d Empty Dalcetrapib N6022 Bay 60-7550 Sildenafil Sildenafil (citrate) Apoptozole Balicatib Isotretinoin O-Phospho-L-serine Lonafarnib Empty
e Empty Oglemilast NVP-HSP990 GSK 650394 EMD638683 Ganetespib Geldanamycin JZL 184 JZL195 Tiplaxtinin CP-640186 (hydrochloride) Empty
f Empty E-64 Nelfinavir (Mesylate) Fenretinide Sacubitril Sacubitril hemicalcium salt Trelagliptin Trelagliptin (succinate) 5-Iodotubercidin PF-04447943 Roflumilast Empty
g Empty IOX2 Zardaverine Salubrinal Cabotegravir Ledipasvir Ledipasvir (acetone) Ledipasvir (D-tartrate) FG-2216 Alvelestat Bivalirudin (Trifluoroacetate) Empty
h Empty TTNPB IDO5L Epacadostat PluriSln 1 AGI-6780 Ilomastat NSC 405020 GSK 2830371 BAY 87-2243 SF1670 Empty

Plate layout: HY-L012-5

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Atglistatin FTI-277 (hydrochloride) DMOG Sal003 P7C3 AZD7545 BMS-303141 L-778123 (hydrochloride) Tolrestat Skp2 Inhibitor C1 Empty
b Empty Dafadine-A Rolipram (R)-(-)-Rolipram 5'-Methylthioadenosine SW033291 SR9243 Saquinavir (Mesylate) Saquinavir Darunavir Darunavir (Ethanolate) Empty
c Empty Fenofibrate Clozapine (N-oxide) Atazanavir (sulfate) Dabigatran (ethyl ester) Atorvastatin (hemicalcium salt) Racecadotril Tolcapone Mevastatin Amprenavir Sivelestat Empty
d Empty Sivelestat (sodium tetrahydrate) Cortisone Cilostazol Simvastatin Rosuvastatin (Calcium) Clarithromycin ZLN005 sn-Glycero-3-phosphocholine 2'-Deoxyguanosine Daprodustat Empty
e Empty AGI-5198 LCZ696 Omapatrilat Leupeptin (hemisulfate) Avanafil Udenafil L-Thyroxine 3-Indoleacetic acid TZ9 TEPP-46 Empty
f Empty PU-WS13 CPDA Enasidenib Enasidenib (mesylate) Endoxifen (hydrochloride) Lipoic acid VR23 Ivosidenib (R,S)-Ivosidenib NCT-501 Empty
g Empty KC7F2 Alda-1 Aldose reductase-IN-1 KML29 Adjudin 3-Methyladenine HA130 DASA-58 TMS GSK864 Empty
h Empty BEC (hydrochloride) JNJ-42165279 (-)-p-Bromotetramisole (oxalate) PD 151746 Indirubin-3'-monoxime PRT4165 BMS-779788 3-Bromopyruvic acid AM 3112 Methoxsalen Empty

Plate layout: HY-L012-6

1 2 3 4 5 6 7 8 9 10 11 12
a Empty (S)-Leucic acid (S)-2-Hydroxy-3-phenylpropanoic acid Clemizole (hydrochloride) T863 Ethylmalonic acid L-Hydroxyproline Octanoic acid 5-Amino-3H-imidazole-4-Carboxamide D-Alanine (-)-Aspartic acid Empty
b Empty GW 4064 Apixaban DGAT-1 inhibitor 2 A939572 3-Methylxanthine FK866 Rivaroxaban WAY-362450 2-Amino-1-phenylethanol Epalrestat Empty
c Empty Carboxypeptidase G2 (CPG2) Inhibitor CPA inhibitor TOK-001 Abiraterone Otamixaban GSK256066 (2,2,2-trifluoroacetic acid) D609 SPK-601 Abiraterone (acetate) VX-222 Empty
d Empty L-Pyroglutamic acid Vitamin D2 Chenodeoxycholic Acid 5-R-Rivaroxaban Dabigatran (ethyl ester hydrochloride) FAAH-IN-2 Ritonavir Nortadalafil Tadalafil Pentostatin Empty
e Empty Alogliptin (Benzoate) Cilazapril (monohydrate) Malotilate N-Acetyl-D-glucosamine Adenosine monophosphate Doxofylline Melatonin Adapalene Benazepril (hydrochloride) Edaravone Empty
f Empty Ketoconazole (+)-Ketoconazole Acitretin Dorzolamide (hydrochloride) Diphylline Perindopril (erbumine) Bestatin Aminophylline Estradiol Alpha-Estradiol Empty
g Empty Niacin Pitavastatin (Calcium) Nicotinamide Pregnenolone Adenine Cytidine Pravastatin (sodium) Lithocholic acid Nafamostat (mesylate) Pimobendan Empty
h Empty Metolazone Acetylcysteine Ethynyl Estradiol Orlistat Allopurinol Adenosine Enalaprilat (dihydrate) Estrone Disulfiram Eplerenone Empty

Plate layout: HY-L012-7

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Gemfibrozil Thiabendazole Ramipril Dipyridamole Irsogladine Enalapril (maleate) Menadione Taurine Memantine (hydrochloride) Captopril Empty
b Empty Argatroban (monohydrate) Moexipril (hydrochloride) Fosinopril (sodium) Temocapril (hydrochloride) Gabexate (mesylate) Dextrose (S)-(+)-Rolipram Dichlorphenamide D-Sorbitol Estriol Empty
c Empty Ozagrel Ozagrel (sodium) Vardenafil (hydrochloride) NAD+ Dopamine (hydrochloride) Hydralazine (hydrochloride) Quinapril (hydrochloride) Tioxolone Lonidamine PMSF Empty
d Empty Creatinine Anagrelide (hydrochloride) Methazolamide Brinzolamide Trandolapril Fondaparinux (sodium) Levobupivacaine (hydrochloride) Zofenopril (calcium) Eicosapentaenoic Acid Indinavir (sulfate) Empty
e Empty Azelaic acid Pentoxifylline Ibudilast Teprenone Acetazolamide Theophylline Tebuconazole Hexylresorcinol L-SelenoMethionine 4-Aminobenzoic acid Empty
f Empty Tilorone (dihydrochloride) N-Acetylprocainamide Benzbromarone Cotinine Tetramisole (hydrochloride) Alrestatin Fludrocortisone (acetate) Histamine Carprofen Metyrapone Empty
g Empty Protoporphyrin IX 4-Aminohippuric acid Proadifen (hydrochloride) Retinol 4-Aminoantipyrine Salicylanilide i-Inositol Ethoxyquin Canrenone Uridin Empty
h Empty Imidapril (hydrochloride) Deoxyarbutin Chlorzoxazone Deoxycorticosterone (acetate) Serotonin hydrochloride Ethoxzolamide cAMP Corticosterone Pyridoxal phosphate Rotenone Empty

Plate layout: HY-L012-8

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Spermidine Carbosulfan Lactose Uric acid Tryptamine 2-Aminobenzenesulfonamide Docosahexaenoic Acid ATP Stearic acid 2'-Deoxycytidine Empty
b Empty 2'-Deoxyuridine Glutathione oxidized Tartaric acid (disodium dihydrate) Sodium orthovanadate Glycylglycine β-Nicotinamide mononucleotide Iloperidone metabolite Hydroxy Iloperidone Omeprazole metabolite Omeprazole sulfide Norgestimate metabolite Norelgestromin N-Desmethylclozapine Empty
c Empty Epiandrosterone N-Acetylneuraminic acid 6-Aminopyrimidin-2(1H)-one PCL 016 Regorafénib N-oxyde (M2) Uracil L-Alloisoleucine Icariin Daidzin Arctigenin Empty
d Empty Ginsenoside Rd Chlorogenic acid Ginkgolic Acid Dimethylfraxetin Hypoxanthine Inosine Guanosine Vanillin Isoliquiritigenin Coenzyme Q10 Empty
e Empty Diosmetin Stigmasterol Tanshinone I Taxifolin Theobromine Naringin Oleanolic Acid Orotic acid Magnolol Caffeic acid Empty
f Empty 18β-Glycyrrhetinic acid Arbutin Baicalein Nordihydroguaiaretic acid D-Galactose (-)-Epigallocatechin L-Alanine β-Alanine Cordycepin Paeoniflorin Empty
g Empty Stachydrine Salvianolic acid A Bilirubin Cholic acid L-Methionin Bergapten D-Mannitol D-Mannose Galangin Homovanillic acid Empty
h Empty L-Glutamine L-Citrulline L-Cystine β-Carotene Succinic acid Astragaloside IV Progesterone L-Arginine α-Lipoic Acid Gentiopicroside Empty

Plate layout: HY-L012-9

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Lovastatin Morroniside Xylose Allantoin Oroxylin A Doxycycline (hyclate) Umbelliferone Hydrocortisone Deoxycholic acid Ginsenoside F1 Empty
b Empty Cinnamic acid Mulberroside A Dicoumarol L-Serine L-Aspartic acid L-Asparagine Schisandrin A Linoleic acid Glucosamine (hydrochloride) Coptisine (chloride) Empty
c Empty Ginkgolide C Phytic acid Shikonin Palmitic acid L-Hisidine (20S)-Protopanaxatriol AKBA Tetrahydrocurcumin Ginsenoside C-K Androsterone Empty
d Empty Xanthohumol Thymidine Apigenin Squalene 2-Methoxybenzoic acid Glycocholic acid Glycoursodeoxycholic acid Citric acid Oxyresveratrol (-)-Fucose Empty
e Empty Loureirin B Pyrogallol 4',5-Dihydroxyflavone Propylparaben Taurochenodeoxycholic acid Isoginkgetin Glycochenodeoxycholic acid 11beta-Hydroxyprogesterone Cholesteryl behenate Palmitelaidic Acid Empty
f Empty p-Hydroxycinnamic acid D-Arabitol Pepstatin Trifluoroacetate [Leu5]-Enkephalin 3,4-Dihydroxybenzeneacetic acid 2,5-Dihydroxybenzoic acid Pyrrole-2-carboxylic acid 2,5-Furandicarboxylic acid L-Homoserine 4-Hydroxy-3-methylbenzoic acid Empty
g Empty 2-(4-Methoxyphenyl)acetic acid Pentadecanoic acid 5-Hydroxymethyluracil 5-Hydroxymethyl-2-furancarboxylic acid 3-Methyl-2-oxobutanoic acid Tyramine 3-Oxopentanedioic acid 2-Oxobutanoic acid H-Phe-Phe-OH 2-Hydroxy-3-methylbutanoic acid Empty
h Empty 5-Hydroxyindole-3-acetic acid H-HoArg-OH H-Tyr(3-I)-OH Glutaric acid 5-Methyluridine Terephthalic acid 4,6-Dioxoheptanoic acid 2-Methylsuccinic acid Creatine Thymine Empty

Plate layout: HY-L012-10

1 2 3 4 5 6 7 8 9 10 11 12
a Empty DL-Norvaline H-Abu-OH Adenosine 5'-diphosphate Xanthosine Dodecanedioic acid N-Acetyl-L-tyrosine H-D-Trp-OH 2-Oxo-3-phenylpropanoic acid 2,4-Dihydroxybenzoic acid 3-Amino-4-methylpentanoic acid Empty
b Empty H-HoPro-OH 4-Methylcatechol 4-Ethylphenol 3-Amino-2-methylpropanoic acid 3-Methylbutanoic acid 2-Ketoglutaric acid Undecanedioic acid Ac-Arg-OH Decanedioic acid 1,3-Dimethyluric acid Empty
c Empty 2-(2-Methylbenzamido)acetic acid 3-Indolepropionic acid Octanedioic acid 3-Hydroxymandelic Acid Desaminotyrosine N-Isovaleroylglycine 3,5-Dihydroxybenzoic acid 2-Hydroxyphenylacetic acid 2-Phenylpropionic acid L-(+)-Arabinose Empty
d Empty 2-Hydroxy-2-methylbutanoic acid Fumaric acid Glycolic acid Hippuric acid L-Gulono-1,4-lactone trans-Aconitic acid H-Gly-Pro-OH 1-Methyl-L-histidine 3-Methyl-L-histidine L-Ornithine Hydrochloride Empty
e Empty 7-Methylxanthine Xanthine Adipic acid 2-Methylpentanedioic acid L-Homocitrulline Hexadecanedioic acid 2-Guanidinoacetic acid L-Arabinitol 2'-Deoxyadenosine 3-Chloro-L-tyrosine Empty
f Empty Phenylacetylglutamine (S)-3-Hydroxybutanoic acid (R)-3-Hydroxybutanoic acid (±) Anabasine L-Norleucine 3-Hydroxypicolinic acid N-Acetylglycine 2-Naphthol NSC 16590 D(-)-2-Aminobutyric acid Empty
g Empty Pyrocatechuic acid L-Proline 4-Hydroxybenzoic acid p-Hydroxybenzaldehyde L-Cysteine Maleic Acid Dulcite L-Lactic acid N-Methylsarcosine Pipecolic acid Empty
h Empty 3-Methoxybenzoic acid 3,4-Dimethoxyphenylacetic acid Pyruvic acid 2,6-Dihydroxybenzoic acid Levulinic acid Glycine (S)-2-Hydroxysuccinic acid Hydrocinnamic acid Pimelic acid Malic acid Empty
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