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  2. Metabolism/Protease Compound Library

Metabolism/Protease Compound Library

Cat. No.: HY-L012
Library Contents: XLSX PDF

A unique collection of 379 Metabolism/Protease-related small molecules for high throughput screening (HTS) and high content screening (HCS).

Size (Pre-dissolved DMSO or Solid) Price Stock
30 μL/well (10 mM solution) Get quote In-stock
50 μL/well (10 mM solution) Get quote In-stock
100 μL/well (10 mM solution) Get quote In-stock
250 μL/well (10 mM solution) Get quote In-stock

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  • Description

  • Product Details

  • Composition

  • Contents

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Description
& Advantages

•   A unique collection of 379 Metabolism/Protease-related small molecules for high throughput screening (HTS) and high content screening (HCS).

•   Targets such as PDE, Cytochrome P450, HMG-CoA Reductase, DPP4, Proteasome, HCV Protease, IDO, Cathepsin, MMP, etc.

•   A useful tool for drug discovery of metabolism-related diseases.

•   Bioactivity and safety confirmed by preclinical research and clinical trials. Some inhibitors have been approved by FDA.

•   Structurally diverse, medicinally active, and cell permeable.

•   More detailed compound information with structure, IC50, and brief introduction.

•   NMR and HPLC validated to ensure high purity and quality.

•   All compounds are in stock and continuously updated.

Product Details
Formulation:
A collection of 379 Metabolism/Protease related compounds supplied as pre-dissolved DMSO solutions or Solid
Container:
96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
Storage:
-80°C
Shipping:
Blue ice
Composition

Metabolism/Protease Compound Library

Source: MedChem Express

Contents of Metabolism/Protease Compound Library

Plate layout: HY-L012-1

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Ledipasvir (D-tartrate) Aliskiren (hemifumarate) Allopurinol 2-Deoxy-D-glucose 4-Butylresorcinol 3-Bromopyruvic acid Tioxolone Chlorzoxazone Fondaparinux (sodium) PMSF Empty
b Empty Edaravone DMOG Theophylline Sodium orthovanadate Sevelamer (hydrochloride) Deoxyarbutin Hexylresorcinol Hydralazine (hydrochloride) Milrinone PluriSln 1 Empty
c Empty Glucosamine (hydrochloride) Memantine (hydrochloride) Bergapten Methoxsalen Captopril Acetazolamide 2-PMPA Metyrapone Oltipraz Ozagrel Empty
d Empty Bivalirudin (Trifluoroacetate) Ibudilast Tartaric acid (disodium dihydrate) Stiripentol PRT4165 Methazolamide Zileuton PD 151746 AEBSF Tetramisole (hydrochloride) Empty
e Empty β-Lapachone DKM 2-93 Oxyresveratrol (R)-Flurbiprofen KNK437 HIV-1 integrase inhibitor Topiroxostat Ozagrel (sodium) ZLN005 AN-2728 Empty
f Empty Diphylline C75 (trans) Irsogladine Isoliquiritigenin AR7 Ethoxzolamide Acriflavine NSC 405020 Magnolol SPK-601 Empty
g Empty D609 Zardaverine Pentostatin LB-100 Baicalein Galangin IDO5L Arbutin Tolcapone (R)-(-)-Rolipram Empty
h Empty Rolipram (S)-(+)-Rolipram Pentoxifylline NLG919 Atglistatin Biochanin A Oroxylin A KRIBB11 Cladribine Olprinone (Hydrochloride) Empty

Plate layout: HY-L012-2

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Malotilate Anagrelide (hydrochloride) Disulfiram Diosmetin TMS Retinoic acid Isotretinoin CL-82198 2-Methoxyestradiol Vildagliptin Empty
b Empty Taxifolin Entacapone PD150606 SB-3CT TCS 401 SF1670 Orteronel LY2183240 Bestatin U-104 Empty
c Empty Carboxypeptidase G2 (CPG2) Inhibitor CPA inhibitor Saxagliptin Febuxostat BIIB021 Epalrestat FAAH-IN-2 Lonidamine Alda-1 Levobupivacaine (hydrochloride) Empty
d Empty NQ301 Acitretin Sobetirome Teprenone Nepicastat (hydrochloride) Pimobendan HTS01037 URB-597 Papaverine Cilomilast Empty
e Empty JNJ-42041935 Bexarotene TTNPB Tamibarotene AM580 Tazarotene PYZD-4409 FG-4592 IOX2 HIV-1 integrase inhibitor 2 Empty
f Empty Chlorogenic acid Xanthohumol CDD3505 Tolrestat Trelagliptin E-64 Benzophenonetetracarboxylic acid Fenofibrate Dorzolamide (hydrochloride) MLN2238 Empty
g Empty Clemizole (hydrochloride) EMD638683 Ganetespib Metolazone TZ9 Cilostazol PYR-41 GMX1778 Arctigenin Deoxycorticosterone (acetate) Empty
h Empty Finasteride (-)-p-Bromotetramisole (oxalate) Nortadalafil Papaverine (hydrochloride) Ro 28-1675 NVP-HSP990 Varespladib Carbosulfan GSK 650394 UAMC00039 (dihydrochloride) Empty

Plate layout: HY-L012-3

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Anagliptin Brinzolamide MG-101 Bortezomib Enalaprilat (dihydrate) UK-371804 A939572 GM6001 TOK-001 CPI-613 Empty
b Empty Tadalafil Dalcetrapib Mevastatin Dafadine-A FK866 Abiraterone (acetate) Fenretinide 5-Iodotubercidin Chenodeoxycholic Acid PX-478 Empty
c Empty T863 PI-1840 PF-04620110 R-7128 Roflumilast Lovastatin SR3335 Cabotegravir Sitagliptin Omapatrilat Empty
d Empty AT13387 BMS-707035 JNJ-42165279 PU-WS13 AHU-377 Balicatib ML-030 Adapalene SW033291 Stigmasterol Empty
e Empty N6022 ML228 ML348 XMD16-5 Ramipril NCT-501 Gabexate (mesylate) Simvastatin Dolutegravir Aminophylline Empty
f Empty DGAT-1 inhibitor 2 INT-747 Aldose reductase-IN-1 FIPI Choline Fenofibrate Fludrocortisone (acetate) LXR-623 AM-2394 Benzbromarone BMS-303141 Empty
g Empty CTS-1027 Teneligliptin TAK-063 A 922500 TM5441 AHU-377 (hemicalcium salt) SR1078 Fluvastatin (sodium) JZL195 Sivelestat Empty
h Empty LW6 Cilazapril (monohydrate) Rivaroxaban INCB 024360 WAY-362450 Tiplaxtinin Pitavastatin (Calcium) Dolutegravir (sodium) Perindopril (erbumine) Imidapril (hydrochloride) Empty

Plate layout: HY-L012-4

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Debio 0932 VX-222 Otamixaban Pravastatin (sodium) Elvitegravir Zofenopril (calcium) Celastrol Betrixaban DASA-58 PF-04457845 Empty
b Empty PF-3845 Apixaban Apremilast Benazepril (hydrochloride) GSK 2830371 Alogliptin (Benzoate) STF-118804 AGI-5198 Sal003 HA130 Empty
c Empty NVP-AUY922 TRC051384 MK-8245 Clinofibrate RVT-501 Linagliptin Quinacrine (dihydrochloride) Enasidenib P7C3 Quinapril (hydrochloride) Empty
d Empty Trelagliptin (succinate) Leupeptin (hemisulfate) Bay 60-7550 SR1001 VR23 PF-8380 AZD7545 Salubrinal NVP-BEP800 Paeoniflorin Empty
e Empty Doxycycline (hyclate) T0901317 AGI-6780 Raltegravir (potassium salt) Tilorone (dihydrochloride) Avanafil FTI-277 (hydrochloride) Enalapril (maleate) Orlistat Fexaramine Empty
f Empty Dabigatran (ethyl ester) Rosuvastatin (Calcium) SR12813 Dipyridamole Amprenavir BMS-779788 AKBA Temocapril (hydrochloride) Oglemilast Udenafil Empty
g Empty MLN9708 T-5224 GSK256066 Boceprevir JZL 184 Sitagliptin (phosphate monohydrate) Vardenafil (hydrochloride) BAY 87-2243 Odanacatib Argatroban (monohydrate) Empty
h Empty Sivelestat (sodium tetrahydrate) Dutasteride Ezatiostat Ketoconazole Oprozomib Moexipril (hydrochloride) Dabigatran (ethyl ester hydrochloride) LX-1031 Nafamostat (mesylate) GW 4064 Empty

Plate layout: HY-L012-5

1 2 3 4 5 6 7 8 9 10 11 12
a Empty TM5275 (sodium) Alvelestat Darunavir KML29 Aliskiren VER-155008 GSK864 DMP 777 Mulberroside A KC7F2 Empty
b Empty Atorvastatin (hemicalcium salt) Naringin ONX-0914 (R,S)-Ivosidenib Ivosidenib Fosinopril (sodium) 17-AAG GLPG1690 Darunavir (Ethanolate) RA190 Empty
c Empty Torcetrapib GW3965 (hydrochloride) Apoptozole SR9243 Dabigatran etexilate Lopinavir Teneligliptin (hydrobromide) GSK256066 (2,2,2-trifluoroacetic acid) Anacetrapib Evacetrapib Empty
d Empty Lonafarnib Alvespimycin (hydrochloride) Nelfinavir (Mesylate) Sildenafil (citrate) Darapladib Saquinavir Telaprevir Pepstatin Indinavir (sulfate) Carfilzomib Empty
e Empty Ritonavir Dabigatran etexilate (mesylate) Danoprevir Edoxaban (tosylate monohydrate) Daclatasvir Clarithromycin Simeprevir LX1606 (Hippurate) Saquinavir (Mesylate) Cobicistat Empty
f Empty Astragaloside IV Atazanavir (sulfate) Daclatasvir (dihydrochloride) Velpatasvir Ledipasvir Angiotensin (1-7) Stibogluconate (sodium) Ledipasvir (acetone) LCZ696 Empty Empty
g Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
h Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
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