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  2. Metabolism/Protease Compound Library

Metabolism/Protease Compound Library

Cat. No.: HY-L012
Library Contents: XLSX PDF

A unique collection of 431 Metabolism/Protease-related small molecules for high throughput screening (HTS) and high content screening (HCS).

Size (Pre-dissolved DMSO or Solid) Price Stock
30 μL/well (10 mM solution) Get quote In-stock
50 μL/well (10 mM solution) Get quote In-stock
100 μL/well (10 mM solution) Get quote In-stock
250 μL/well (10 mM solution) Get quote In-stock

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  • Description

  • Product Details

  • Composition

  • Contents

  • Documentation

& Advantages

•   A unique collection of 431 Metabolism/Protease-related small molecules for high throughput screening (HTS) and high content screening (HCS).

•   Targets such as PDE, Cytochrome P450, HMG-CoA Reductase, DPP4, Proteasome, HCV Protease, IDO, Cathepsin, MMP, etc.

•   A useful tool for drug discovery of metabolism-related diseases.

•   Bioactivity and safety confirmed by preclinical research and clinical trials. Some inhibitors have been approved by FDA.

•   Structurally diverse, medicinally active, and cell permeable.

•   More detailed compound information with structure, IC50, and brief introduction.

•   NMR and HPLC validated to ensure high purity and quality.

•   All compounds are in stock and continuously updated.

Product Details
A collection of 431 Metabolism/Protease related compounds supplied as pre-dissolved DMSO solutions or Solid
96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
Blue ice

Metabolism/Protease Compound Library

Source: MedChem Express

Contents of Metabolism/Protease Compound Library

Plate layout: HY-L012-1

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Ledipasvir (D-tartrate) Aliskiren (hemifumarate) 1-Aminobenzotriazole Allopurinol L-Hisidine 2-Deoxy-D-glucose 4-Butylresorcinol 3-Bromopyruvic acid Tioxolone Chlorzoxazone Empty
b Empty Gallic acid 2-Aminobenzenesulfonamide Fondaparinux (sodium) PMSF Edaravone DMOG Caffeic acid Theophylline Flopropione Sodium orthovanadate Empty
c Empty Deoxyarbutin Hexylresorcinol Hydralazine (hydrochloride) Thiabendazole Lipoic acid α-Lipoic Acid Milrinone Serotonin hydrochloride Salicylanilide PluriSln 1 Empty
d Empty Glucosamine (hydrochloride) Memantine (hydrochloride) Methoxsalen Bergapten Captopril Ethoxyquin IBMX Acetazolamide 2-PMPA Metyrapone Empty
e Empty Oltipraz Ozagrel Bivalirudin (Trifluoroacetate) Ibudilast Tartaric acid (disodium dihydrate) Stiripentol PRT4165 Methazolamide Zileuton PD 151746 Empty
f Empty AEBSF Tetramisole (hydrochloride) DKM 2-93 Oxyresveratrol (R)-Flurbiprofen BRL-50481 KNK437 Topiroxostat Ozagrel (sodium) Gemfibrozil Empty
g Empty ZLN005 AN-2728 FCCP Diphylline C75 (trans) Alrestatin Irsogladine Isoliquiritigenin AR7 Ethoxzolamide Empty
h Empty Acriflavine NSC 405020 Doxofylline Magnolol SPK-601 D609 Zardaverine Pentostatin LB-100 Baicalein Empty

Plate layout: HY-L012-2

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Apigenin Galangin IDO5L Arbutin ML346 Alpha-Estradiol Tolcapone (R)-(-)-Rolipram Rolipram (S)-(+)-Rolipram Empty
b Empty Tanshinone I Indirubin-3'-monoxime Pentoxifylline IDO-IN-7 Atglistatin Biochanin A Oroxylin A KRIBB11 Cladribine Olprinone (Hydrochloride) Empty
c Empty Shikonin Malotilate Androsterone Anagrelide (hydrochloride) Disulfiram Diosmetin TMS Retinoic acid Isotretinoin CL-82198 Empty
d Empty 2-Methoxyestradiol Vildagliptin Taxifolin Entacapone PD150606 SB-3CT TCS 401 SF1670 Orteronel LY2183240 Empty
e Empty Tebuconazole Bestatin U-104 Talabostat (mesylate) SYP-5 Carboxypeptidase G2 (CPG2) Inhibitor CPA inhibitor Saxagliptin Febuxostat BIIB021 Empty
f Empty Epalrestat FAAH-IN-2 Lonidamine NSC 663284 Alda-1 TOFA Levobupivacaine (hydrochloride) NQ301 Acitretin Teprenone Empty
g Empty Nepicastat (hydrochloride) Pimobendan Adjudin HTS01037 URB-597 Papaverine Cilomilast PKM2-IN-1 Ginkgolic Acid JNJ-42041935 Empty
h Empty D4-abiraterone Bexarotene TTNPB Tamibarotene AM580 Tazarotene PYZD-4409 FG-4592 IOX2 Chlorogenic acid Empty

Plate layout: HY-L012-3

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Xanthohumol CDD3505 Coptisine (chloride) Tolrestat Trelagliptin E-64 Benzophenonetetracarboxylic acid Fenofibrate Dorzolamide (hydrochloride) MLN2238 Empty
b Empty Clemizole (hydrochloride) EMD638683 Ganetespib Metolazone Cilostazol PYR-41 GMX1778 Arctigenin TEPP-46 Deoxycorticosterone (acetate) Empty
c Empty Finasteride Nortadalafil Papaverine (hydrochloride) DPP-IV-IN-2 Ro 28-1675 NVP-HSP990 Varespladib Carbosulfan GSK 650394 UAMC00039 (dihydrochloride) Empty
d Empty Anagliptin Brinzolamide MG-101 Bortezomib Enalaprilat (dihydrate) Racecadotril UK-371804 A939572 GM6001 TOK-001 Empty
e Empty CPI-613 Tadalafil Dalcetrapib Mevastatin Dafadine-A FK866 Abiraterone (acetate) Fenretinide 5-Iodotubercidin Chenodeoxycholic Acid Empty
f Empty Rotenone T863 PI-1840 PF-04620110 CD437 R-7128 TRO 19622 Roflumilast Lovastatin SR3335 Empty
g Empty Cabotegravir PF-05175157 Sitagliptin Omapatrilat AT13387 BMS-707035 JNJ-42165279 BMS-986205 PU-WS13 AHU-377 Empty
h Empty Balicatib ML-030 Adapalene SW033291 Stigmasterol N6022 ML228 ML348 Daidzin XMD16-5 Empty

Plate layout: HY-L012-4

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Ramipril NCT-501 Gabexate (mesylate) Simvastatin Dolutegravir Aminophylline DGAT-1 inhibitor 2 SZL P1-41 INT-747 Aldose reductase-IN-1 Empty
b Empty FIPI Choline Fenofibrate Fludrocortisone (acetate) LXR-623 AM-2394 Benzbromarone BMS-303141 CTS-1027 Teneligliptin TAK-063 Empty
c Empty A 922500 TM5441 Trandolapril SR1078 AHU-377 (hemicalcium salt) JZL195 Fluvastatin (sodium) Sivelestat LW6 Cilazapril (monohydrate) Empty
d Empty Rivaroxaban UVI 3003 Isavuconazole WWL70 INCB 024360 WAY-362450 Tiplaxtinin Ginkgolide C Pitavastatin (Calcium) Dolutegravir (sodium) Empty
e Empty Perindopril (erbumine) Imidapril (hydrochloride) Debio 0932 VX-222 Otamixaban Pravastatin (sodium) Elvitegravir Zofenopril (calcium) Celastrol Betrixaban Empty
f Empty DASA-58 PF-04457845 PF-3845 Apixaban Apremilast Benazepril (hydrochloride) GSK 2830371 Alogliptin (Benzoate) STF-118804 AGI-5198 Empty
g Empty Sal003 HA130 Skp2 Inhibitor C1 NVP-AUY922 TRC051384 Clinofibrate 18α-Glycyrrhetinic acid RVT-501 Linagliptin Quinacrine (dihydrochloride) Empty
h Empty Enasidenib P7C3 Sildenafil Quinapril (hydrochloride) Trelagliptin (succinate) Leupeptin (hemisulfate) Bay 60-7550 (20S)-Protopanaxatriol SR1001 VR23 Empty

Plate layout: HY-L012-5

1 2 3 4 5 6 7 8 9 10 11 12
a Empty PF-8380 AZD7545 Salubrinal NVP-BEP800 Paeoniflorin Doxycycline (hyclate) T0901317 AGI-6780 Raltegravir (potassium salt) Tilorone (dihydrochloride) Empty
b Empty Avanafil FTI-277 (hydrochloride) BAY-1436032 Enalapril (maleate) Orlistat Fexaramine Dabigatran (ethyl ester) Rosuvastatin (Calcium) Avasimibe SR12813 Empty
c Empty Dipyridamole Amprenavir BMS-779788 AKBA Temocapril (hydrochloride) Oglemilast Udenafil MLN9708 T-5224 GSK256066 Empty
d Empty Boceprevir JZL 184 CP-640186 (hydrochloride) Sitagliptin (phosphate monohydrate) Vardenafil (hydrochloride) BAY 87-2243 Odanacatib Argatroban (monohydrate) Sivelestat (sodium tetrahydrate) Dutasteride Empty
e Empty Ezatiostat Ketoconazole Oprozomib Moexipril (hydrochloride) Dabigatran (ethyl ester hydrochloride) Nafamostat (mesylate) GW 4064 TM5275 (sodium) Alvelestat Darunavir Empty
f Empty KML29 Aliskiren VER-155008 GSK864 Geldanamycin DMP 777 Mulberroside A KC7F2 Atorvastatin (hemicalcium salt) LY2955303 Empty
g Empty Naringin ONX-0914 Ivosidenib (R,S)-Ivosidenib Fosinopril (sodium) 17-AAG Chondroitin (sulfate) GLPG1690 GSK2033 Darunavir (Ethanolate) Empty
h Empty SR9238 RA190 Torcetrapib GW3965 (hydrochloride) Apoptozole SR9243 Dabigatran etexilate Lopinavir Teneligliptin (hydrobromide) GSK256066 (2,2,2-trifluoroacetic acid) Empty

Plate layout: HY-L012-6

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Anacetrapib Evacetrapib Lonafarnib Alvespimycin (hydrochloride) Nelfinavir (Mesylate) Sildenafil (citrate) Darapladib Saquinavir Icariin Telaprevir Empty
b Empty Indinavir (sulfate) Carfilzomib Ritonavir Dabigatran etexilate (mesylate) Danoprevir Edoxaban (tosylate monohydrate) Daclatasvir Clarithromycin Simeprevir LX1606 (Hippurate) Empty
c Empty Saquinavir (Mesylate) Cobicistat Astragaloside IV Atazanavir (sulfate) Daclatasvir (dihydrochloride) Velpatasvir Ledipasvir Angiotensin (1-7) Stibogluconate (sodium) Ledipasvir (acetone) Empty
d Empty LCZ696 Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
e Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
f Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
g Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
h Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty

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