1. Screening Libraries
  2. Metabolism/Protease Compound Library

Metabolism/Protease Compound Library

Cat. No.: HY-L012
Library Contents: XLSX PDF

A unique collection of 404 Metabolism/Protease-related small molecules for high throughput screening (HTS) and high content screening (HCS).

Size (Pre-dissolved DMSO or Solid) Price Stock
30 μL/well (10 mM solution) Get quote In-stock
50 μL/well (10 mM solution) Get quote In-stock
100 μL/well (10 mM solution) Get quote In-stock
250 μL/well (10 mM solution) Get quote In-stock

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  • Description

  • Product Details

  • Composition

  • Contents

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Description
& Advantages

•   A unique collection of 404 Metabolism/Protease-related small molecules for high throughput screening (HTS) and high content screening (HCS).

•   Targets such as PDE, Cytochrome P450, HMG-CoA Reductase, DPP4, Proteasome, HCV Protease, IDO, Cathepsin, MMP, etc.

•   A useful tool for drug discovery of metabolism-related diseases.

•   Bioactivity and safety confirmed by preclinical research and clinical trials. Some inhibitors have been approved by FDA.

•   Structurally diverse, medicinally active, and cell permeable.

•   More detailed compound information with structure, IC50, and brief introduction.

•   NMR and HPLC validated to ensure high purity and quality.

•   All compounds are in stock and continuously updated.

Product Details
Formulation:
A collection of 404 Metabolism/Protease related compounds supplied as pre-dissolved DMSO solutions or Solid
Container:
96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
Storage:
-80°C
Shipping:
Blue ice
Composition

Metabolism/Protease Compound Library

Source: MedChem Express

Contents of Metabolism/Protease Compound Library

Plate layout: HY-L012-1

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Ledipasvir (D-tartrate) Aliskiren (hemifumarate) Allopurinol 2-Deoxy-D-glucose 4-Butylresorcinol 3-Bromopyruvic acid Tioxolone Chlorzoxazone Gallic acid 2-Aminobenzenesulfonamide Empty
b Empty Fondaparinux (sodium) PMSF Edaravone DMOG Caffeic acid Theophylline Flopropione Sodium orthovanadate Deoxyarbutin Hexylresorcinol Empty
c Empty Hydralazine (hydrochloride) Milrinone Salicylanilide PluriSln 1 Glucosamine (hydrochloride) Memantine (hydrochloride) Bergapten Methoxsalen Captopril Ethoxyquin Empty
d Empty IBMX Acetazolamide 2-PMPA Metyrapone Oltipraz Ozagrel Bivalirudin (Trifluoroacetate) Ibudilast Tartaric acid (disodium dihydrate) Stiripentol Empty
e Empty PRT4165 Methazolamide Zileuton PD 151746 AEBSF Tetramisole (hydrochloride) β-Lapachone DKM 2-93 Oxyresveratrol (R)-Flurbiprofen Empty
f Empty KNK437 HIV-1 integrase inhibitor Topiroxostat Ozagrel (sodium) ZLN005 AN-2728 Diphylline C75 (trans) Alrestatin Irsogladine Empty
g Empty Isoliquiritigenin AR7 Ethoxzolamide Acriflavine NSC 405020 Doxofylline Magnolol D609 SPK-601 Zardaverine Empty
h Empty Pentostatin LB-100 Baicalein Galangin IDO5L Arbutin Tolcapone (R)-(-)-Rolipram (S)-(+)-Rolipram Rolipram Empty

Plate layout: HY-L012-2

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Tanshinone I Indirubin-3'-monoxime Pentoxifylline NLG919 Atglistatin Biochanin A Oroxylin A KRIBB11 Cladribine Olprinone (Hydrochloride) Empty
b Empty Malotilate Anagrelide (hydrochloride) Disulfiram Diosmetin TMS Retinoic acid Isotretinoin CL-82198 2-Methoxyestradiol Vildagliptin Empty
c Empty Taxifolin Entacapone PD150606 SB-3CT TCS 401 SF1670 Orteronel LY2183240 Tebuconazole Bestatin Empty
d Empty U-104 Carboxypeptidase G2 (CPG2) Inhibitor CPA inhibitor Saxagliptin Febuxostat BIIB021 Epalrestat FAAH-IN-2 Lonidamine NSC 663284 Empty
e Empty Alda-1 TOFA Levobupivacaine (hydrochloride) NQ301 Acitretin Sobetirome Teprenone Nepicastat (hydrochloride) Pimobendan HTS01037 Empty
f Empty URB-597 Papaverine Cilomilast PKM2-IN-1 JNJ-42041935 Bexarotene TTNPB Tamibarotene AM580 Tazarotene Empty
g Empty PYZD-4409 FG-4592 IOX2 HIV-1 integrase inhibitor 2 Chlorogenic acid Xanthohumol CDD3505 BAY 73-6691 racemate Tolrestat Trelagliptin Empty
h Empty E-64 Benzophenonetetracarboxylic acid Fenofibrate Dorzolamide (hydrochloride) MLN2238 Clemizole (hydrochloride) EMD638683 Ganetespib Metolazone TZ9 Empty

Plate layout: HY-L012-3

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Cilostazol PYR-41 GMX1778 Arctigenin TEPP-46 Deoxycorticosterone (acetate) Finasteride Nortadalafil Papaverine (hydrochloride) H-Lys(4-nitro-Z)-pyrrolidide Empty
b Empty Ro 28-1675 NVP-HSP990 Varespladib Carbosulfan GSK 650394 UAMC00039 (dihydrochloride) Anagliptin Brinzolamide MG-101 Bortezomib Empty
c Empty Enalaprilat (dihydrate) Racecadotril UK-371804 A939572 GM6001 TOK-001 CPI-613 Tadalafil Dalcetrapib Mevastatin Empty
d Empty Dafadine-A FK866 Fenretinide Abiraterone (acetate) 5-Iodotubercidin Chenodeoxycholic Acid PX-478 PI-1840 T863 PF-04620110 Empty
e Empty R-7128 Roflumilast Lovastatin SR3335 Cabotegravir PF-05175157 Sitagliptin Omapatrilat AT13387 BMS-707035 Empty
f Empty JNJ-42165279 PU-WS13 AHU-377 Balicatib ML-030 Adapalene SW033291 Stigmasterol N6022 ML228 Empty
g Empty ML348 XMD16-5 Ramipril NCT-501 Gabexate (mesylate) Simvastatin Dolutegravir Aminophylline DGAT-1 inhibitor 2 SZL P1-41 Empty
h Empty INT-747 Aldose reductase-IN-1 FIPI Choline Fenofibrate Fludrocortisone (acetate) LXR-623 AM-2394 Benzbromarone BMS-303141 CTS-1027 Empty

Plate layout: HY-L012-4

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Teneligliptin TAK-063 A 922500 TM5441 SR1078 AHU-377 (hemicalcium salt) JZL195 Fluvastatin (sodium) Sivelestat LW6 Empty
b Empty Cilazapril (monohydrate) Rivaroxaban INCB 024360 WAY-362450 Tiplaxtinin Pitavastatin (Calcium) Dolutegravir (sodium) Perindopril (erbumine) Imidapril (hydrochloride) Debio 0932 Empty
c Empty VX-222 Otamixaban Pravastatin (sodium) Elvitegravir Zofenopril (calcium) Celastrol Betrixaban DASA-58 PF-04457845 PF-3845 Empty
d Empty Apixaban Apremilast Benazepril (hydrochloride) GSK 2830371 Alogliptin (Benzoate) STF-118804 AGI-5198 Sal003 HA130 Skp2 Inhibitor C1 Empty
e Empty NVP-AUY922 TRC051384 MK-8245 Clinofibrate 18α-Glycyrrhetinic acid RVT-501 Linagliptin Quinacrine (dihydrochloride) Enasidenib P7C3 Empty
f Empty Sildenafil Quinapril (hydrochloride) Trelagliptin (succinate) Leupeptin (hemisulfate) Bay 60-7550 SR1001 VR23 PF-8380 AZD7545 Salubrinal Empty
g Empty NVP-BEP800 Paeoniflorin Doxycycline (hyclate) T0901317 AGI-6780 Raltegravir (potassium salt) Tilorone (dihydrochloride) Avanafil FTI-277 (hydrochloride) Enalapril (maleate) Empty
h Empty Orlistat Fexaramine Dabigatran (ethyl ester) Rosuvastatin (Calcium) SR12813 Dipyridamole Amprenavir BMS-779788 AKBA Temocapril (hydrochloride) Empty

Plate layout: HY-L012-5

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Oglemilast Udenafil MLN9708 T-5224 GSK256066 Boceprevir JZL 184 CP-640186 (hydrochloride) Sitagliptin (phosphate monohydrate) Vardenafil (hydrochloride) Empty
b Empty BAY 87-2243 Odanacatib Argatroban (monohydrate) Sivelestat (sodium tetrahydrate) Dutasteride Ezatiostat Ketoconazole Oprozomib Moexipril (hydrochloride) Dabigatran (ethyl ester hydrochloride) Empty
c Empty Nafamostat (mesylate) GW 4064 TM5275 (sodium) Alvelestat Darunavir KML29 Aliskiren VER-155008 GSK864 Geldanamycin Empty
d Empty DMP 777 Mulberroside A KC7F2 Atorvastatin (hemicalcium salt) LY2955303 Naringin ONX-0914 (R,S)-Ivosidenib Ivosidenib Fosinopril (sodium) Empty
e Empty 17-AAG GLPG1690 Darunavir (Ethanolate) RA190 Torcetrapib GW3965 (hydrochloride) Apoptozole SR9243 Dabigatran etexilate Lopinavir Empty
f Empty Teneligliptin (hydrobromide) GSK256066 (2,2,2-trifluoroacetic acid) Anacetrapib Evacetrapib Lonafarnib Alvespimycin (hydrochloride) Nelfinavir (Mesylate) Sildenafil (citrate) Darapladib Saquinavir Empty
g Empty Telaprevir Pepstatin Indinavir (sulfate) Carfilzomib Ritonavir Dabigatran etexilate (mesylate) Danoprevir Edoxaban (tosylate monohydrate) Daclatasvir Clarithromycin Empty
h Empty Simeprevir LX1606 (Hippurate) Saquinavir (Mesylate) Cobicistat Astragaloside IV Atazanavir (sulfate) Daclatasvir (dihydrochloride) Velpatasvir Ledipasvir Angiotensin (1-7) Empty

Plate layout: HY-L012-6

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Stibogluconate (sodium) Ledipasvir (acetone) LCZ696 Sevelamer (hydrochloride) Empty Empty Empty Empty Empty Empty Empty
b Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
c Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
d Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
e Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
f Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
g Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
h Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
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