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  2. Metabolism/Protease Compound Library

Metabolism/Protease Compound Library

Cat. No.: HY-L012
Library Contents: XLSX PDF

A unique collection of 462 Metabolism/Protease-related small molecules for high throughput screening (HTS) and high content screening (HCS).

Metabolism/Protease Compound Library
Size (Pre-dissolved DMSO or Solid) Price Stock
30 μL/well (10 mM solution) Get quote In-stock
50 μL/well (10 mM solution) Get quote In-stock
100 μL/well (10 mM solution) Get quote In-stock
250 μL/well (10 mM solution) Get quote In-stock

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  • Description

  • Product Details

  • Composition

  • Contents

  • Documentation

Description
& Advantages

•   A unique collection of 462 Metabolism/Protease-related small molecules for high throughput screening (HTS) and high content screening (HCS).

•   Targets such as PDE, Cytochrome P450, HMG-CoA Reductase, DPP4, Proteasome, HCV Protease, IDO, Cathepsin, MMP, etc.

•   A useful tool for drug discovery of metabolism-related diseases.

•   Bioactivity and safety confirmed by preclinical research and clinical trials. Some inhibitors have been approved by FDA.

•   Structurally diverse, medicinally active, and cell permeable.

•   More detailed compound information with structure, IC50, and brief introduction.

•   NMR and HPLC validated to ensure high purity and quality.

•   All compounds are in stock and continuously updated.

Product Details
Formulation:
A collection of 462 Metabolism/Protease related compounds supplied as pre-dissolved DMSO solutions or Solid
Container:
96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
Storage:
-80°C
Shipping:
Blue ice
Composition

Metabolism/Protease Compound Library

Source: MedChem Express

Contents of Metabolism/Protease Compound Library

Plate layout: HY-L012-1

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Ledipasvir (D-tartrate) Aliskiren (hemifumarate) 1-Aminobenzotriazole Allopurinol L-Hisidine 2-Deoxy-D-glucose 4-Butylresorcinol 3-Bromopyruvic acid Tioxolone Chlorzoxazone Empty
b Empty Gallic acid 2-Aminobenzenesulfonamide Fondaparinux (sodium) PMSF Edaravone DMOG Theophylline Caffeic acid Flopropione Sodium orthovanadate Empty
c Empty Deoxyarbutin Hexylresorcinol Hydralazine (hydrochloride) Thiabendazole α-Lipoic Acid Lipoic acid Milrinone Salicylanilide PluriSln 1 Glucosamine (hydrochloride) Empty
d Empty Memantine (hydrochloride) Bergapten Methoxsalen Captopril Ethoxyquin IBMX Acetazolamide 2-PMPA Metyrapone Oltipraz Empty
e Empty Ozagrel Bivalirudin (Trifluoroacetate) Tartaric acid (disodium dihydrate) Stiripentol PRT4165 Methazolamide 1-(1-(Benzo[b]thiophen-2-yl)ethyl)-1-hydroxyurea PD 151746 AEBSF Tetramisole (hydrochloride) Empty
f Empty DKM 2-93 Oxyresveratrol (R)-Flurbiprofen BRL-50481 KNK437 Topiroxostat Ozagrel (sodium) Gemfibrozil ZLN005 AN-2728 Empty
g Empty FCCP Diphylline C75 (trans) Alrestatin Irsogladine Isoliquiritigenin AR7 Ethoxzolamide NSC 405020 Doxofylline Empty
h Empty Magnolol SPK-601 D609 Zardaverine Pentostatin Galangin Baicalein Apigenin IDO5L Arbutin Empty

Plate layout: HY-L012-2

1 2 3 4 5 6 7 8 9 10 11 12
a Empty ML346 Alpha-Estradiol Tolcapone (R)-(-)-Rolipram Rolipram (S)-(+)-Rolipram Tanshinone I Indirubin-3'-monoxime Pentoxifylline FG-2216 Empty
b Empty IDO-IN-7 Atglistatin Biochanin A Oroxylin A KRIBB11 Cladribine Olprinone (Hydrochloride) Shikonin Malotilate Androsterone Empty
c Empty Anagrelide (hydrochloride) Disulfiram Diosmetin TMS Retinoic acid Isotretinoin Nordihydroguaiaretic acid CL-82198 2-Methoxyestradiol Vildagliptin Empty
d Empty Taxifolin Entacapone PD150606 SB-3CT Vadadustat TCS 401 SF1670 Orteronel LY2183240 Tebuconazole Empty
e Empty Bestatin U-104 Talabostat (mesylate) GSTO1-IN-1 SYP-5 Carboxypeptidase G2 (CPG2) Inhibitor CPA inhibitor Saxagliptin Febuxostat BIIB021 Empty
f Empty Epalrestat FAAH-IN-2 Lonidamine NSC 663284 Alda-1 TOFA Levobupivacaine (hydrochloride) NQ301 Acitretin Mitochonic acid 5 Empty
g Empty Pyributicarb Teprenone Nepicastat (hydrochloride) Pimobendan Adjudin Dicoumarol HTS01037 URB-597 Canrenone Cilomilast Empty
h Empty PKM2-IN-1 Ginkgolic Acid JNJ-42041935 D4-abiraterone Bexarotene TTNPB Abiraterone Vinpocetine Tamibarotene AM580 Empty

Plate layout: HY-L012-3

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Tazarotene PYZD-4409 FG-4592 IOX2 Chlorogenic acid Xanthohumol 1-Linoleoyl Glycerol CDD3505 Coptisine (chloride) Gentiopicroside Empty
b Empty Tolrestat Trelagliptin E-64 Benzophenonetetracarboxylic acid Fenofibrate Dorzolamide (hydrochloride) MLN2238 Clemizole (hydrochloride) EMD638683 Apararenone Empty
c Empty Ganetespib Metolazone SR-18292 Cilostazol PYR-41 GMX1778 Tetrahydrocurcumin Arctigenin TEPP-46 Deoxycorticosterone (acetate) Empty
d Empty Finasteride (-)-p-Bromotetramisole (oxalate) Nortadalafil DPP-IV-IN-2 Ro 28-1675 NVP-HSP990 Varespladib Carbosulfan GSK 650394 UAMC00039 (dihydrochloride) Empty
e Empty Anagliptin Brinzolamide MG-101 Bortezomib Enalaprilat (dihydrate) Racecadotril UK-371804 A939572 GM6001 TOK-001 Empty
f Empty 6,8-Bis(benzylthio)octanoic acid CPDA Tadalafil Dalcetrapib Proadifen (hydrochloride) Mevastatin Dafadine-A FK866 Abiraterone (acetate) Fenretinide Empty
g Empty 5-Iodotubercidin Chenodeoxycholic Acid Daprodustat PX-478 Rotenone T863 PI-1840 PF-04447943 PF-04620110 CD437 Empty
h Empty R-7128 TRO 19622 GCN2-IN-1 Roflumilast Lovastatin SR3335 Cabotegravir PF-05175157 Sitagliptin Omapatrilat Empty

Plate layout: HY-L012-4

1 2 3 4 5 6 7 8 9 10 11 12
a Empty AT13387 BMS-707035 JNJ-42165279 BMS-986205 PU-WS13 AHU-377 Balicatib ML-030 Adapalene SW033291 Empty
b Empty Stigmasterol PF-05180999 N6022 Eplerenone ML228 ML348 Daidzin XMD16-5 Ramipril Schisandrin A Empty
c Empty NCT-501 Gabexate (mesylate) Simvastatin Dolutegravir Aminophylline DGAT-1 inhibitor 2 SZL P1-41 INT-747 Aldose reductase-IN-1 FIPI Empty
d Empty Choline Fenofibrate Fludrocortisone (acetate) LXR-623 AM-2394 Benzbromarone BMS-303141 CTS-1027 Teneligliptin TAK-063 A 922500 Empty
e Empty TM5441 AHU-377 (hemicalcium salt) Trandolapril SR1078 JZL195 Fluvastatin (sodium) Sivelestat Cilazapril (monohydrate) LW6 Rivaroxaban Empty
f Empty 5-R-Rivaroxaban UVI 3003 Isavuconazole WWL70 INCB 024360 WAY-362450 Tiplaxtinin Ginkgolide C Pitavastatin (Calcium) Dolutegravir (sodium) Empty
g Empty Perindopril (erbumine) Imidapril (hydrochloride) L-778123 (hydrochloride) Debio 0932 MK-8617 Raltegravir VX-222 Otamixaban Pravastatin (sodium) Elvitegravir Empty
h Empty Zofenopril (calcium) Celastrol Betrixaban DASA-58 PF-04457845 PF-3845 Apixaban Apremilast Benazepril (hydrochloride) GSK 2830371 Empty

Plate layout: HY-L012-5

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Alogliptin (Benzoate) STF-118804 AGI-5198 Sal003 HA130 Skp2 Inhibitor C1 NVP-AUY922 TRC051384 Clinofibrate RVT-501 Empty
b Empty Linagliptin Quinacrine (dihydrochloride) Enasidenib P7C3 BMS-309403 Quinapril (hydrochloride) Trelagliptin (succinate) Leupeptin (hemisulfate) Bay 60-7550 (20S)-Protopanaxatriol Empty
c Empty SR1001 VR23 PF-8380 AZD7545 Salubrinal NVP-BEP800 Paeoniflorin Doxycycline (hyclate) T0901317 AGI-6780 Empty
d Empty Tilorone (dihydrochloride) Avanafil FTI-277 (hydrochloride) Gemigliptin Tipifarnib BAY-1436032 Enalapril (maleate) Orlistat Fexaramine IDO-IN-2 Empty
e Empty Dabigatran (ethyl ester) Rosuvastatin (Calcium) Avasimibe SR12813 Dipyridamole Amprenavir BMS-779788 AKBA Temocapril (hydrochloride) Oglemilast Empty
f Empty Udenafil MLN9708 T-5224 GSK256066 Boceprevir JZL 184 CP-640186 (hydrochloride) Sitagliptin (phosphate monohydrate) Vardenafil (hydrochloride) BAY 87-2243 Empty
g Empty Odanacatib Argatroban (monohydrate) Sivelestat (sodium tetrahydrate) Dutasteride Ezatiostat Ketoconazole (+)-Ketoconazole Oprozomib Moexipril (hydrochloride) Dabigatran (ethyl ester hydrochloride) Empty
h Empty Nafamostat (mesylate) GW 4064 TM5275 (sodium) Alvelestat Darunavir KML29 Aliskiren VER-155008 GSK864 Geldanamycin Empty

Plate layout: HY-L012-6

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Mulberroside A Enasidenib (mesylate) KC7F2 KW-2478 LX1606 Atorvastatin (hemicalcium salt) LY2955303 Naringin ONX-0914 Ivosidenib Empty
b Empty (R,S)-Ivosidenib Fosinopril (sodium) 17-AAG GLPG1690 GSK2033 Darunavir (Ethanolate) SR9238 RA190 Torcetrapib GW3965 (hydrochloride) Empty
c Empty Ginsenoside C-K Apoptozole SR9243 Dabigatran etexilate Lopinavir Teneligliptin (hydrobromide) GSK256066 (2,2,2-trifluoroacetic acid) Anacetrapib Evacetrapib Lonafarnib Empty
d Empty Ginsenoside F1 Alvespimycin (hydrochloride) Nelfinavir (Mesylate) Sildenafil (citrate) Darapladib Saquinavir Icariin Telaprevir Indinavir (sulfate) Carfilzomib Empty
e Empty Ritonavir Dabigatran etexilate (mesylate) Danoprevir Edoxaban (tosylate monohydrate) Daclatasvir Clarithromycin Simeprevir LX1606 (Hippurate) Saquinavir (Mesylate) Cobicistat Empty
f Empty Astragaloside IV Pepstatin Trifluoroacetate Atazanavir (sulfate) Daclatasvir (dihydrochloride) Velpatasvir Ledipasvir Ombitasvir Angiotensin (1-7) Stibogluconate (sodium) Ledipasvir (acetone) Empty
g Empty Ginsenoside Rd LCZ696 Empty Empty Empty Empty Empty Empty Empty Empty Empty
h Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
Documentation

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