1. Screening Libraries
  2. Membrane Transporter/Ion Channel Compound Library

Membrane Transporter/Ion Channel Compound Library

Cat. No.: HY-L011
Library Contents: XLSX PDF

A unique collection of 417 small molecule modulators used for Ion Channel and Membrane Transporter research.

Membrane Transporter/Ion Channel Compound Library
Size (Pre-dissolved DMSO or Solid) Price Stock
30 μL/well (10 mM solution) Get quote In-stock
50 μL/well (10 mM solution) Get quote In-stock
100 μL/well (10 mM solution) Get quote In-stock
250 μL/well (10 mM solution) Get quote In-stock

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  • Description

  • Product Details

  • Composition

  • Contents

  • Documentation

& Advantages

•   A unique collection of 417 small molecule modulators used for Ion Channel and Membrane Transporter research.

•   The library contains compounds targeting Membrane Transporters including Pgp, CRM1, BCRP, etc., and Ion Channels including CFTR, proton pump, sodium pump, calcium pump, etc.

•   A useful tool for the research of drug absorption and distribution.

•   Bioactivity and safety confirmed by preclinical research and clinical trials. Some inhibitors have been approved by FDA.

•   Structurally diverse, medicinally active, and cell permeable.

•   Rich documentation with structure, IC50, and summary.

•   NMR and HPLC validated to ensure high purity.

•   All compounds are in stock and continuously updated.

Product Details
A collection of 417 Membrane Transporter/Ion Channel related compounds supplied as pre-dissolved DMSO solutions or Solid
96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
Blue ice

Membrane Transporter/Ion Channel Compound Library

Source: MedChem Express

Contents of Membrane Transporter/Ion Channel Compound Library

Plate layout: HY-L011-1

1 2 3 4 5 6 7 8 9 10 11 12
a Empty SKF-96365 (hydrochloride) Vonoprazan Ko 143 JNJ-17203212 Pipequaline PAP-1 HC-067047 SKF89976A (hydrochloride) DMCM (hydrochloride) MRK-016 Empty
b Empty LY2365109 (hydrochloride) ZL006 A-804598 CaCCinh-A01 U93631 D-AP5 GSK2193874 Norverapamil (hydrochloride) gamma-DGG Kynurenic acid Empty
c Empty Isoguvacine (hydrochloride) 7-Chloro-4-hydroxyquinoline-2-carboxylic acid 7-Chlorokynurenic acid sodium salt YM-58483 Diphenyleneiodonium chloride NPPB Sarcosine Allopregnanolone Org-26576 DHBP (dibromide) Empty
d Empty ZD7288 PF-01247324 Picrotoxin ICA-069673 4-Acetamidobutanoic acid L-DABA Vanilpyruvic acid GAL-021 Bamaquimast NS-638 Empty
e Empty CDN1163 Polyoxyethylene stearate Gefapixant Ilaprazole AMG9810 EIPA ML213 PSB-12062 GYKI53655 hydrochloride Bepridil hydrochloride Empty
f Empty CGP52432 Gabazine ML335 Capsaicin Dapagliflozin Dapagliflozin ((2S)-1,2-propanediol, hydrate) Canagliflozin Fantofarone Tariquidar Tariquidar (methanesulfonate, hydrate) Empty
g Empty Ketanserin Ketanserin (tartrate) Eniporide hydrochloride SB-705498 AMG 517 Almitrine mesylate SN 6 Desformylflustrabromine hydrochloride Aminooxyacetic acid hemihydrochloride Mirogabalin besylate Empty
h Empty Bitopertin AM-0902 WS-12 A-967079 Pyr3 Fluxametamide Tulrampator Aniracetam Ampalex Farampator Empty

Plate layout: HY-L011-2

1 2 3 4 5 6 7 8 9 10 11 12
a Empty NS11394 Icilin A-803467 A-867744 NS 1738 PNU-120596 ABT-239 SB-366791 Rostafuroxin PEAQX (tetrasodium hydrate) Empty
b Empty ML277 NS-1619 Efonidipine (hydrochloride monoethanolate) CFM-2 Pyr6 Naspm Naspm (trihydrochloride) GSK-7975A PEPA Nicardipine (Hydrochloride) Empty
c Empty Dantrolene (sodium hemiheptahydrate) PNU-282987 GS967 Hexachlorophene R(+)-IAA-94 LDN-212320 AZD3965 YHO-13177 YHO-13351 (free base) Optovin Empty
d Empty Eliprodil Ifenprodil (tartrate) ML204 ML204 (hydrochloride) Ivacaftor SDZ 220-581 SDZ 220-581 (hydrochloride) Rivanicline hemioxalate Lumacaftor KN-62 Empty
e Empty Vinpocetine Tofogliflozin (hydrate) Zatebradine (hydrochloride) Zatebradine TRAM-34 Cisatracurium (besylate) HM30181 HM30181 mesylate Lansoprazole Methionine Empty
f Empty A 839977 Ro 25-6981 (Maleate) PPQ-102 Amiodarone (hydrochloride) Levcromakalim Nilvadipine Pinacidil monohydrate Tebanicline (hydrochloride) L-655708 AF-353 Empty
g Empty GTS-21 (dihydrochloride) Diltiazem (hydrochloride) Ataluren Phenylpiracetam Imepitoin HC-030031 Chembridge-5861528 CNQX DNQX NBQX Empty
h Empty Fanapanel Fanapanel hydrate Talampanel Dizocilpine (Maleate) (-)-Dizocilpine (Maleate) Bay-K-8644 ((S)-(-)-) Bay-K-8644 ((R)-(+)-) Glibenclamide Zosuquidar Lesinurad Empty

Plate layout: HY-L011-3

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Lesinurad (sodium) Vonoprazan Fumarate Vigabatrin Empagliflozin KB-R7943 (mesylate) NS309 Tezacaftor Ertugliflozin GW791343 (dihydrochloride) UK-5099 Empty
b Empty A 438079 (hydrochloride) Sotagliflozin S0859 E-4031 Mibefradil (dihydrochloride) A-317491 A-317491 (sodium salt hydrate) Capsazepine QNZ46 NS6180 Empty
c Empty CGP37157 BTB06584 Gabapentin enacarbil MDL-29951 Etifoxine (hydrochloride) Etifoxine CFTR(inh)-172 VU 0240551 SN 2 (S)-(-)-5-Fluorowillardiine (hydrochloride) Empty
d Empty Verinurad ICA-121431 NS1643 Flupirtine (Maleate) Dofequidar (fumarate) Acamprosate (calcium) (R)-Baclofen Valspodar Rosiglitazone Mitiglinide (Calcium) Empty
e Empty Ranolazine (dihydrochloride) Manidipine (dihydrochloride) Cilnidipine Vinblastine Flecainide (acetate) Clevidipine Omberacetam Bumetanide Pantoprazole (sodium) Sunifiram Empty
f Empty NMDA Coluracetam Meclofenoxate (hydrochloride) Nonivamide Radafaxine (hydrochloride) Bexagliflozin GlyH-101 IOWH-032 Azimilide (Dihydrochloride) RQ-00203078 Empty
g Empty SYM2206 L-701324 CIQ GlyT2-IN-1 Adjudin Lorediplon Pyr10 GSK1016790A Cariporide KS176 Empty
h Empty XEN907 BCTC KM11060 RN-1734 CRAC intermediate 2 (-)-Aspartic acid Transcrocetin meglumine salt Zosuquidar (trihydrochloride) Senicapoc A-740003 Empty

Plate layout: HY-L011-4

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Elacridar Proparacaine (Hydrochloride) (-)-Menthol Dronedarone (Hydrochloride) Gabapentin Gabapentin (hydrochloride) Verapamil (hydrochloride) Tetracaine Trimethadione Mexiletine (hydrochloride) Empty
b Empty Flumazenil Azelnidipine Vigabatrin (Hydrochloride) Etomidate Etomidate (hydrochloride) Levetiracetam Minoxidil Omeprazole Oxcarbazepine Vecuronium (bromide) Empty
c Empty Zonisamide Furosemide Prilocaine Felbamate Lidocaine Lidocaine (hydrochloride) Riluzole Riluzole hydrochloride Dofetilide Isradipine Empty
d Empty Trichlormethiazide Carbamazepine Glipizide Indapamide Nimodipine Acetylcholine (chloride) Nifedipine Amiloride (hydrochloride) Amiloride hydrochloride dihydrate Atracurium (besylate) Empty
e Empty Felodipine Amlodipine Amlodipine (maleate) Amlodipine (besylate) Cromolyn (sodium) Primidone Nefiracetam Nicorandil ATP (disodium salt) Lacidipine Empty
f Empty Chlormezanone Ginkgolide A Flunarizine (dihydrochloride) Dyclonine (hydrochloride) Memantine (hydrochloride) Orphenadrine (citrate) Adiphenine (hydrochloride) Ibutilide (fumarate) Tolbutamide Nitrendipine Empty
g Empty Pancuronium (dibromide) Propafenone (hydrochloride) Phenytoin Phenytoin (sodium) Neomycin (sulfate) Niflumic acid Lamotrigine Mepivacaine (hydrochloride) Amitriptyline (hydrochloride) Ouabain (Octahydrate) Empty
h Empty Probenecid Doxapram (hydrochloride hydrate) Dibucaine Dibucaine (hydrochloride) Ropivacaine (hydrochloride monohydrate) Ropivacaine hydrochloride Dequalinium (Chloride) Hexamethonium (Bromide) Decamethonium (Bromide) Zinc Pyrithione Empty

Plate layout: HY-L011-5

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Triamterene Piracetam Tetrabenazine Tetrabenazine (Racemate) Tetrabenazine ((+)-) 4-Aminopyridine Lercanidipine (hydrochloride) Rabeprazole (sodium) Tiagabine (hydrochloride) Eslicarbazepine (acetate) Empty
b Empty Gliclazide Lomerizine dihydrochloride Dihydroergotoxine (mesylate) Dinotefuran Meticrane Lobeline (hydrochloride) Fendiline (hydrochloride) Digoxin Penfluridol Cinnarizine Empty
c Empty N-Acetylprocainamide L-Cycloserine 3-Methyl-7-chloro-1,2,4-benzothiadiazine 1,1-dioxide Ajmaline Terfenadine Carbamoylcholine (chloride) Flufenamic acid Propoxycaine (hydrochloride) Mephenesin Quinidine hydrochloride monohydrate Empty
d Empty (-)-Sparteine (sulfate pentahydrate) Bemegride Digitoxin Ethosuximide Chlorpropamide Butamben Esomeprazole magnesium Benidipine (hydrochloride) Domiphen (bromide) Procyclidine (hydrochloride) Empty
e Empty Anabasine Benzamil hydrochloride (Z)-Capsaicin Oxiracetam Afloqualone 6-Methoxy-2-naphthoic acid Tannic acid Cloperastine fendizoate 7ACC1 Quinine Empty
f Empty Canagliflozin (hemihydrate) Ginsenoside Rb1 Ginsenoside Rc Ginsenoside Rd Eucalyptol γ-Aminobutyric acid Phloretin Phlorizin Piperine Caffeic acid Empty
g Empty Cytisine L-Phenylalanine (+)-Bicuculline Daurisoline Catharanthine Imperatorin Sinapine (thiocyanate) Acacetin Reserpine Reserpine (hydrochloride) Empty
h Empty Ginsenoside Rf Ginsenoside Rg3 Ginsenoside Ro Jujuboside A alpha-Asarone (20S)-Protopanaxadiol Camphor Shikonin DL-Borneol (+)-Borneol Empty

Plate layout: HY-L011-6

1 2 3 4 5 6 7 8 9 10 11 12
a Empty (-)-Borneol Loureirin B Acevaltrate (-)-Securinine Ibotenic acid Podocarpic acid Methyllycaconitine citrate 6,2'-Dihydroxyflavone 6-Methylflavone Phe-Met-Arg-Phe amide trifluoroacetate Empty
b Empty (+)-Sparteine 3,4,5-Trimethoxycinnamic acid WS-3 Traxoprodil Benzocaine p-Hydroxybenzaldehyde Glycine Empty Empty Empty Empty
c Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
d Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
e Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
f Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
g Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty
h Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty Empty

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