Blogs | MedChemExpress

Manzamine A, an Orally Active β-Carboline Alkaloid with Antiviru, Antimalarial and Anticancer Activities

AManzamine A is an orally active β-carboline alkaloid effective against HSV-1, Cancer, and Malaria.
STX-0119 is a Selective, Orally Active STAT3 Dimerization Inhibitor

STX-0119 is a selective, orally active STAT3 dimerization inhibitor. STX-0119 shows potent antitumor activity.
BNS-22 is a DNA Topoisomerase II Catalytic Inhibitor

BNS-22 is a potent and selective inhibitor of TOP2α and TOP2β that exhibits anti-proliferative activities.
Linzagolix is a potent, non-Peptide, and Orally Active GnRH Antagonist

Linzagolix is a potent, non-peptide, and orally active GnRH antagonist used for the research of endometriosis and uterine myomas.
Trolox, an Analogue of Vitamin E, Possesses Antioxidant Effect

Trolox is an analogue of vitamin E with a powerful antioxidant effect. Trolox is also a powerful inhibitor of membrane damage.
IMT1 is a First-in-Class Specific and Noncompetitive Human POLRMT Inhibitor

IMT1 is a first-in-class specific and noncompetitive human POLRMT inhibitor for mitochondrial transcription disorders related diseases.
TAS-119 is a Selective and Orally Active Aurora A Inhibitor

TAS-119 is an orally active, selective inhibitor of Aurora kinase A. A clinical candidate for efficacy testing in combination with taxanes.
Ro 90-7501, a Radiosensitizer, is an Aβ42 Fibril Assembly and PP5 Inhibitor

Ro 90-7501, an Aβ42 fibril assembly inhibitor, inhibits PP5 in a TPR-dependent manner and has radiosensitizing effects on cervical cancer cells.
COTI-2 is an Orally Available Mutant p53 Activator

COTI-2 is an orally available third generation activator of p53 mutant forms by inhibiting the PI3K/AKT/mTOR pathway. COTI-2 has has anti-cancer activity.
VERU-111 is an Orally Active Tubulin Inhibitor

VERU-111 (ABI-231) is a potent and orally bioavailable α and β tubulin inhibitor, which displays strong antiproliferative activity.

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Blogs (10)